Search results for: 'Peptide'

Cat.No. 产品名称 Information

GC26093 α-Conotoxin GI α-Conotoxin GI, a 13-residue peptide originally isolated from the venom of the fish-hunting cone snail Conus geographus, acts as a competitive antagonist for the muscle-type nicotinic acetylcholine receptor (nAChR) with excellent selectivity for α/δ receptor subunit binding over α/γ.

GC26066 WAY-383487 WAY-383487 is one of the Tat peptide derivatives and inhibits HIV-1 long terminal repeat-activated transcription.

GC26027 V-0219 V-0219 is an orally active, positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R), can be used for obesity-associated diabetes research.

GC25648 MOTS-c MOTS-c, a mitochondria-derived peptide (MDP), exerts antinociceptive and anti-inflammatory effects through activating AMPK pathway and inhibiting MAP kinases-c-fos signaling pathway.

GC25579 LL-37(human) LL-37, human is a 37-residue, amphipathic, cathelicidin-derived peptide, which exhibits a broad spectrum of antimicrobial activity.

GC25304 CP2 CP2 is a cyclic peptide that inhibits the JmjC histone demethylases KDM4 with IC50 values of 42 nM and 29 nM for KDM4A and KDM4C, respectively.

GC67887 Val-Cit-PAB-MMAF sodium Val-Cit-PAB-MMAF sodium 是抗体偶联药物 ADC 的一部分。Val-Cit-PAB-MMAF sodium 由 ADC linker (peptide Val-Cit-PAB) 和强效微管蛋白聚合抑制剂 MMAF 偶联而成。

GC67812 MC-VA-PAB-Exatecan MC-VA-PAB-Exatecan 是抗体偶联药物 ADC 的一部分。MC-VA-PAB-Exatecan 由 ADC linker (peptide MC-VA-PAB) 和 DNA 拓扑异构酶 I (topoisomerase I) 抑制剂 Exatecan 偶联而成。MC-VA-PAB-Exatecan 合成的 ADC 具有较好的抗肿瘤活性。

GC52506 Ghrelin (human) (trifluoroacetate salt)

Lenomorelin

A growth hormone releasing peptide

GC52490 Glucagon (hydrochloride) A peptide hormone

GC52488 Bz-FVR-AMC (trifluoroacetate salt)

Benzoyl-Phe-Val-Arg-AMC, Thrombin Fluorogenic Substrate III

A fluorogenic peptide substrate

GC52474 Arg-Gly-Asp (trifluoroacetate salt)

RGD

A synthetic peptide corresponding to an integrin cell adhesion sequence

GC52460 tcY-NH2 (trifluoroacetate salt)

tc-YPGKF-NH2, trans-cinnamoyl-YPGKF-amide, trans-cinnamoyl-YPGKF-NH2

A peptide antagonist of PAR4

GC52457 WRW4 (trifluoroacetate salt)

Trp-Arg-Trp-Trp-Trp-Trp-CONH2, Trp-Arg-Trp-Trp-Trp-Trp-NH2, WRWWWW-NH2

A peptide antagonist of FPR2 and FPR3

GC52453 Orexin A (17-33) (human, mouse, rat, bovine) (trifluoroacetate salt)

OXA (17-33)

A peptide orexin receptor 1 agonist

GC52443 Akt Substrate (trifluoroacetate salt)

RPRAATF

An Akt peptide substrate

GC52426 Chemerin-9 (human) (acetate)

Chemerin (149-157), YFPGQFAFS

A peptide agonist of CMKLR1 and CMKLR2

GC52423 10Panx (trifluoroacetate salt)

10Panx1, WRQAAFVDSY

A peptide inhibitor of PANX1

GC52419 MOG (35-55) (mouse, rat) (trifluoroacetate salt)

MEVGWYRSPFSRVVHLYRNGK, Myelin Oligodendrocyte Glycoprotein (35-55)

An MOG antigen peptide

GC52416 Histatin 5 (trifluoroacetate salt)

DSHAKRHHGYKRKFHEKHHSHRGY, Hst-5

An antimicrobial peptide

GC52414 [Ala17]-MCH (trifluoroacetate salt)

Ala17-Melanin-Concentrating Hormone

An MCH-derived peptide and MCH receptor agonist

GC52412 TT-232 (trifluoroacetate salt) A synthetic peptide derivative of somatostatin

GC52406 AMPR-22 (trifluoroacetate salt)

KKMMKKGGKFGTFMAIGGIR

An antimicrobial peptide

GC52397 SOR-C13 (trifluoroacetate salt) A peptide TRPV6 antagonist

GC52395 Indolicidin (trifluoroacetate salt)

ILPWKWPWWPWRR-NH2

An antimicrobial peptide

GC52390 Spexin 1 (human, mouse, rat, bovine) (acetate)

Neuropeptide Q, NPQ, NWTPQAMLYLKGAQ-NH2, SPX1

An endogenous peptide and agonist of GAL₂ and GAL₃

GC52387 Crosstide (trifluoroacetate salt)

Gly-Arg-Pro-Arg-Thr-Ser-Ser-Phe-Ala-Glu-Gly-OH, GRPRTSSFAEG-OH

A peptide substrate for Akt

GC52380 AOD-9604 (acetate) A synthetic lipolytic peptide

GC52378 Cecropin A (trifluoroacetate salt) An antimicrobial peptide

GC52369 Cecropin B (trifluoroacetate salt) An antimicrobial peptide

GC52355 BimS BH3 (51-76) (human) (trifluoroacetate salt)

DMRPEIWIAQELRRIGDEFNAYYARR-OH, Bims (51-76)

A Bim-derived peptide

GC52354 Tertiapin Q (trifluoroacetate salt)

TPN(M13Q), TPNQ

A peptide derivative of tertiapin

GC52346 IDR 1002 (trifluoroacetate salt) A synthetic cationic innate defense regulator peptide

GC52344 Bak BH3 (72-87) (human) (trifluoroacetate salt) A Bak-derived peptide

GC52338 α-Conotoxin PnIA (trifluoroacetate salt)

α-CtxPnIA, αPnIA

A peptide antagonist of α3β2-subunit containing and α7 nAChRs

GC66679 2,6-Dimethyl-L-tyrosine

Dmt

2,6-Dimethyl-L-tyrosine (Dmt) 是一种酪氨酸衍生物，可增强阿片肽（opioid peptides）的受体亲和力、功能性生物活性和体内镇痛作用。

GC66368 Defensin HNP-2 human An antimicrobial peptide

GC52128 AOD-9604 A synthetic lipolytic peptide

GC52127 Pexiganan (acetate)

培西加南

An antimicrobial peptide

GC65529 TRAP-6 amide A peptide PAR1 agonist

GC65451 RR-11a analog RR-11a analog 是一种有效且不可逆的 Schistosoma mansoni legumain 抑制剂。其 IC50 为 31 nM。RR-11a analog 是 aza-Asn 的衍生物和 aza-peptide Michael 的受体。

GC65109 MC-VA-PABC-MMAE MC-VA-PABC-MMAE 是抗体偶联药物 ADC 的一部分。MC-VA-PABC-MMAE 由 ADC linker (peptide MC-VA-PABC) 和强效微管蛋白聚合抑制剂 MMAE 偶联而成。

GC64908 Defensin HNP-1 human An antimicrobial peptide

GC64447 KRpep-2d KRpep-2d is a K-Ras(G12D) selective inhibitory cyclic peptide with selectivity against wild-type (WT) K-Ras and the K-Ras(G12C) mutant. The IC50 value is 1.6 nM.