Other Apoptosis(其他细胞凋亡)
- Cat.No. 产品名称 Information
-
GC11655
Moexipril HCl
莫昔普利盐酸盐,RS-10085
A prodrug form of moexiprilat -
GC15550
Lacidipine
拉西地平
An L-type calcium channel blocker -
GC12105
Etidronate
羟基乙叉二膦酸,Etidronate; HEDPA; HEDP
A bisphosphonate bone resorption inhibitor -
GC17121
Mycophenolic acid
霉酚酸; Mycophenolate
An immunosuppressive microbial metabolite -
GC13210
Flubendazole
氟苯咪唑
An anthelmintic -
GC11670
Pranoprofen
普拉洛芬
An NSAID and COX-1 inhibitor -
GC11532
Lonidamine
氯尼达明; AF-1890; Diclondazolic Acid; DICA
An inhibitor of hexokinase -
GC15271
Tyrphostin AG 879
AG 879
A non-specific tyrphostin ErbB2 inhibitor -
GC14273
TTNPB (Arotinoid Acid)
Ro 13-7410; Arotinoid acid; AGN191183
A potent, selective RAR agonist -
GC17096
STF-118804
烟酰胺磷酸核糖基转移酶
A Nampt inhibitor -
GC13616
Sodium ascorbate
维生素C钠; Sodium ascorbate; Sodium L-ascorbate; Vitamin C sodium salt
抗坏血酸钠(Sodium L-ascorbate)是一种电子供体,是一种内源性抗氧化剂。抗坏血酸钠选择性抑制 Cav3.2 通道,IC50 为 6.5 μM.抗坏血酸钠也是一种胶原蛋白沉积增强剂和弹性生成抑制剂。 -
GC11107
PF-573228
6-[(4-((3-(甲磺酰基)苄基)氨基)-5-三氟甲基嘧啶-2-基)氨基]-3,4-二氢-1H-喹啉-2-酮
A selective focal adhesion kinase inhibitor -
GC13246
Ibandronate sodium
伊班膦酸钠
A bisphosphonate bone resorption inhibitor -
GC15178
Hexamethonium Bromide
六甲溴铵
A nondepolarizing neuromuscular blocking agent -
GC12940
Fidaxomicin
非达霉素; OPT-80; PAR-101
A natural antibiotic -
GC14499
Fenoprofen calcium hydrate
非诺洛芬钙盐二水合物,Fenoprofen calcium salt dihydrate
An NSAID -
GC11383
CYT997 (Lexibulin)
CYT-997
An inhibitor of microtubule polymerization -
GC13502
Cysteamine HCl
半胱胺盐酸盐; 2-Aminoethanethiol hydrochloride; 2-Mercaptoethylamine hydrochloride
A radioprotective aminothiol -
GC10813
Clofibric Acid
氯贝酸; Chlorofibrinic acid
A PPARα agonist and the active metabolite of clofibrate -
GC12733
C646
C646是一种有效的选择性p300/CBP组蛋白乙酰转移酶抑制剂(Ki 400 nM),已被证明具有多效性,包括神经保护、抗癌和抗上皮间质转化(anti-EMT)作用。
-
GC14987
GSK-3 Inhibitor IX (BIO)
(2'Z,3'E)-6-溴靛玉红-3'-肟,GSK-3 Inhibitor IX
A potent, selective, and reversible GSK3 inhibitor -
GC14930
Benzbromarone
苯溴马隆
An inhibitor of URAT1 -
GC14314
Aloperine
苦豆碱
An alkaloid with diverse biological activities -
GC11528
Orotic acid
乳清酸; 6-Carboxyuracil; Vitamin B13
乳清酸 (6-Carboxyuracil) 是嘧啶核苷酸和 RNA 生物合成的前体,从线粒体二氢乳清酸脱氢酶 (DHODH) 中释放出来,通过细胞质 UMP 合酶转化为 UMP。 -
GC15760
Ramipril
雷米普利; HOE-498
A prodrug from of ramiprilat -
GC15033
Azathioprine
硫唑嘌呤; BW 57-322
An immunosuppressive purine analog -
GC13339
Ketoprofen
酮洛芬; RP-19583
A non-selective COX inhibitor -
GC16450
Prednisone
强的松; Dehydrocortisone
A synthetic glucocorticoid -
GC13906
Nebivolol hydrochloride
盐酸奈必洛尔; R 065824 hydrochloride
A β1-AR antagonist -
GC12013
Sodium salicylate
水杨酸钠; Salicylic acid sodium salt; 2-Hydroxybenzoic acid sodium salt
水杨酸钠(水杨酸钠盐)抑制环加氧酶 2(COX-2)活性,与转录因子(NF-κB)激活无关。 -
GC11332
Pitavastatin
匹伐他汀; NK-104
Pitavastatin (NK-104) 是一种有效的羟甲基戊二酰辅酶A (HMG-CoA) 还原酶抑制剂。 -
GC12830
Stavudine (d4T)
司他夫定; d4T
An inhibitor of HIV reverse transcriptase -
GC15578
Dienogest
地诺孕素; STS 557
A synthetic progestin and PR agonist -
GC13835
Toremifene Citrate
枸橼酸托瑞米芬; Z-Toremifene citrate; NK 622; FC-1157a
A selective estrogen receptor modulator -
GC14123
GW441756
A potent inhibitor of TrkA
-
GC16077
Deracoxib
地拉考昔; SC 046; SC 46; SC 59046
An NSAID and selective COX-2 inhibitor -
GC16772
Cortisone acetate
醋酸可的松; Cortisone 21-acetate
A synthetic glucocorticoid -
GC12308
Fosbretabulin (Combretastatin A4 Phosphate (CA4P)) Disodium
CA 4DP; CA 4P; Combretastatin A4 disodium phosphate
A potent inhibitor of tubulin polymerization -
GC11895
Mevastatin
美伐他汀; Compactin; ML236B
An HMG-CoA reductase inhibitor -
GC13667
Temozolomide
替莫唑胺; NSC 362856; CCRG 81045; TMZ
替莫唑胺是一种口服活性烷化剂,可诱导 DNA 中 O6-甲基鸟嘌呤的形成,其在随后的 DNA 复制周期中与胸腺嘧啶错配,从而激活细胞凋亡途径,替莫唑胺可穿过血脑屏障并适用于恶性神经胶质瘤和转移性黑色素瘤。 -
GC14699
CPI-203
A bioavailable inhibitor of BET bromodomains
-
GC14247
GDC-0623
RG 7421; MEK inhibitor 1
A potent, ATP-uncompetitive inhibitor of MEK1 -
GC14756
EI1
6-氰基-N-[(1,2-二氢-4,6-二甲基-2-氧代-3-吡啶基)甲基]-1-(1-乙基丙基)-1H-吲哚-4-甲酰胺,KB-145943
A selective inhibitor of EZH2 -
GC17331
Salubrinal
Salubrinal是有效的选择性真核翻译起始因子2α(eIF2α)去磷酸化抑制剂。
-
GC17430
2-Deoxy-D-glucose
2-脱氧-D-葡萄糖; 2-DG; 2-Deoxy-D-arabino-hexose; D-Arabino-2-deoxyhexose
2-Deoxy-D-glucose (2DG),是一种葡萄糖类似物,作为竞争性糖酵解抑制剂。 -
GC14063
GSK1324726A
I-BET726
A selective inhibitor of BET family proteins -
GC11648
BML-277
Chk2 Inhibitor II
A selective DNA damage control kinase inhibitor -
GC13359
Topotecan HCl
盐酸拓扑替康; SKF 104864A Hydrochloride; NSC 609669 Hydrochloride
A potent inhibitor of DNA topoisomerase I -
GC11669
Tamoxifen Citrate
他莫昔芬柠檬酸盐; ICI 46474; (Z)-Tamoxifen Citrate; trans-Tamoxifen Citrate
A selective estrogen receptor modulator -
GC17865
Lomustine
洛莫司汀; CCNU; NSC 79037
A DNA alkylating agent