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Cancer Biology(癌症生物学)

  1. Cat.No. 产品名称 Information
  2. GC91432 CAY10799

    Di-tert-butyl (((S)-1-(tert-butoxy)-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)carbamoyl)-L-glutamate

    CAY10799是合成前体,用于制备前列腺特异性膜抗原(PSMA)配体和荧光探针。这些配体和探针已被用于检测LNCaP和PC3细胞中的PSMA。
  3. GC91419 CYY292 CYY292是一种PDGFRα、PDGFRβ、FGFR1、-2和-3的抑制剂,它们的IC50分别为5.35、4.6、28、28和78 nM。
  4. GC91406 UK 122 (trifluoroacetate salt) UK 122是一种尿激酶型纤溶酶原激活剂(uPA)抑制剂(IC50 = 0.2 uM)。它选择性地作用于uPA,而不影响组织型纤溶酶原激活剂(tPA)、胰蛋白酶、纤溶酶和凝血酶(所有的IC50均大于100uM)。
  5. GC26181 (±)-Catechin

    rel-Cianidanol; rel-Catechuic acid

    (±) - Catechin (rel Xianidanol) is the racemate of Catechin.

  6. GC91297 Cholesterol-Doxorubicin

    Chol-DOX

    一种阿霉素的前药形式。

  7. GC91294 S-Geranylgeranyl-L-glutathione

    GGG

    一种P2RY8配体

  8. GC91124 Lipid III-45

    Cationic Lipid A

    一种可离子化的阳离子脂质

  9. GC91096 S-72

    一种微管聚合抑制剂。

  10. GC91083 Tiopronin-Cysteine Disulfide

    α-Mercaptopropionylglycine-Cysteine Disulfide

    一种硫普罗宁的代谢产物。

  11. GC91061 UNC8153 (trifluoroacetate salt)

    NSD2的降解剂

  12. GC91050 Bactobolin A (hydrochloride)

    BN-183B

    一种具有抗生素和抗癌活性的微生物代谢产物。

  13. GC91039 TG2-179-1

    一种BAP1抑制剂

  14. GC91030 Biotin-Cholesterol

    Biotin-Provitamin D

    一种生物素化的胆固醇

  15. GC90982 STING Agonist D61

    D61, Stimulator of Interferon Genes Agonist D61

    STING激动剂

  16. GC90981 Lipid 10

    ?EA-PIP

    一种可离子化的阳离子脂质

  17. GC90964 Lipid Catechol

    一种用于构建脂质前药纳米组装体的脂质。

  18. GC90829 1-Palmitoyl-2-Pyropheophorbide a-sn-glycero-3-PC

    1-Palmitoyl-2-Pyropheophorbide a-sn-glycero-3-Phosphocholine, 1-Palmitoyl-2-Pyropheophorbide a-sn-glycero-3-Phosphatidylcholine, Porphyrin-lipid, Pyro-PtdCho

    一种磷脂-卟啉共轭物

  19. GC90822 LAU-0901

    一种PAF受体拮抗剂

  20. GC90811 1-Palmitoyl-d9-2-Arachidonoyl-sn-glycero-3-PC

    1-Palmitoyl-d9-2-Arachidonoyl-sn-glycero-3-Phosphocholine, PAPC-d9, PC-d9(16:0/20:4)

    一种用于量化1-棕榈酰基-2-花生四烯酸基-sn-甘油3-磷脂胆碱的内部标准。

  21. GC90794 Adenosine 5'-methylenediphosphate (sodium salt)

    Adenosine 5'-(α,β-methylene)diphosphate, AMP-CP, APCP, 5'-APCP

    一种外切5'-核苷酸酶的抑制剂

  22. GC90784 STING Agonist 12L

    Stimulator of Interferon Genes Agonist 12L

    STING激动剂

  23. GC90779 Shepherdin (trifluoroacetate salt)

    Lys-His-Ser-Ser-Gly-Cys-Ala-Phe-Leu-OH, Survivin (79-87)

    一种抑制survivin-Hsp90相互作用的物质

  24. GC90774 1-Linoleoyl Lysophosphatidic Acid (sodium salt)

    1-Linoleoyl-2-hydroxy-sn-glycero-3-PA, 1-Linoleoyl-2-hydroxy-sn-glycero-3-phosphate, 1-Linoleoyl LPA

    一种甘油磷脂

  25. GC90745 1,2-Dioleoyl-3(S)-trimethylammoniumpropane (chloride)

    (S)-DOTAP, (S)-N,N,N-Trimethyl-2,3-bis(oleoyloxy)propan-1-aminium

    一个阳离子脂质

  26. GC90653 ERX-41

    一种内质网应激诱导剂

  27. GC90611 RTDLDSLRTYTL (trifluoroacetate salt)

    一种αVβ6整合素配体

  28. GC90496 β-Cortolone

    20β-Cortolone, NSC 56997

    一种皮质醇的代谢产物。

  29. GC90492 5-Dibromomethyl Anastrozole

    阿那曲唑的合成中间体。

  30. GC90030 Demethoxycurcumin

    DMC

    天然的姜黄素在癌症和炎症中扮演重要角色。

  31. GC70062 Tri-GalNAc(OAc)3 TFA Tri-GalNAc(OAc)3 TFA 是一种 tri-GalNAc 配体,可用于合成 GalNAc-LYTAC。GalNAc-LYTAC 利用去唾液酸糖蛋白受体进行靶向蛋白降解。
  32. GC20228 α-Amyrin

    α-香树脂醇

    α-香树脂醇是一种五环三萜类化合物。

  33. GC52505 Ganglioside GT1b (bovine) (sodium salt)

    Ganglioside G1, Trisialoganglioside GT1b

    A sphingolipid
  34. GC52504 Human Vitamin D Receptor Reporter Assay System

    NR1I1, VDR

    A nuclear receptor cell-based reporter assay
  35. GC52484 Purified Ganglioside Mixture (bovine) (ammonium salt) A mixture of purified bovine gangliosides
  36. GC52483 Fucosylated Ganglioside GM1 (porcine) (ammonium salt)

    Fucosylated Monosialoganglioside GM1, Fucosyl GM1

    A sphingolipid
  37. GC52472 Inostamycin A (sodium salt)

    Inostamycin

    A bacterial metabolite with anticancer activity
  38. GC52460 tcY-NH2 (trifluoroacetate salt)

    tc-YPGKF-NH2, trans-cinnamoyl-YPGKF-amide, trans-cinnamoyl-YPGKF-NH2

    A peptide antagonist of PAR4
  39. GC52412 TT-232 (trifluoroacetate salt) A synthetic peptide derivative of somatostatin
  40. GC52404 γ-Glu-Phe (trifluoroacetate salt)

    γ-Glutamylphenylalanine

    A dipeptide with metabolism-altering activity
  41. GC52397 SOR-C13 (trifluoroacetate salt) A peptide TRPV6 antagonist
  42. GC52392 Biotin-H10 (trifluoroacetate salt)

    Biotin-GGGSGMKMQVRIYLV-OH, Biotin-Gly-Gly-Gly-Ser-Gly-Met-Lys-Met-Gln-Val-Arg-Ile-Tyr-Leu-Val-OH

    A biotinylated form of H10
  43. GC52371 Vimentin (G146R) (139-159)-biotin Peptide

    Biotin-GQGKSRLRDLYEEEMRELRRQ, Biotin-GQGKSRLRDLYEEEMRELRRQ (X=Citrulline), VIM (G146R) (139-159)-biotin

    A biotinylated mutant vimentin peptide
  44. GC52370 Citrullinated Vimentin (R144) (139-159)-biotin Peptide

    Biotin-GQGKS(Cit)LGDLYEEEMRELRRQ, Biotin-GQGKSXLGDLYEEEMRELRRQ (X=Citrulline), Citrullinated VIM (R144)-biotin

    A biotinylated and citrullinated vimentin peptide
  45. GC52367 Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide

    Biotin-GQGKS(Cit)L(Cit)DLYEEEMRELRRQ, Biotin-GQGKSXLXDLYEEEMRELRRQ (X=Citrulline), Citrullinated VIM (G146R) (R144 + R146)-biotin

    A biotinylated and citrullinated mutant vimentin peptide
  46. GC52364 Vimentin (139-159)-biotin Peptide

    VIM (139-159)-biotin

    A biotinylated vimentin peptide
  47. GC52338 α-Conotoxin PnIA (trifluoroacetate salt)

    α-CtxPnIA, αPnIA

    A peptide antagonist of α3β2-subunit containing and α7 nAChRs
  48. GC52333 DSPE-PEG(2000)-NHS

    A PEGylated derivative of DSPE

  49. GC52324 3-(3-Hydroxyphenyl)propionic Acid sulfate

    3-HPPA sulfate

    A metabolite of certain phenols and glycosides
  50. GC52316 Deferitrin

    GT-56-252, (S)-4'-Hydroxydesazadesferrithiocin

    An iron chelator and derivative of desferrithiocin
  51. GC52314 Lysyllysyllysine (trifluoroacetate salt)

    Trilysine

    A tripeptide

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