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Home >> Signaling Pathways >> Neuroscience >> AChR

AChR(乙酰胆碱受体)

AChR, also known as acetylcholine receptor, is an integral membrane protein that responds to the binding of acetylcholine.

Products for  AChR

  1. Cat.No. 产品名称 Information
  2. GC26093 α-Conotoxin GI α-Conotoxin GI, a 13-residue peptide originally isolated from the venom of the fish-hunting cone snail Conus geographus, acts as a competitive antagonist for the muscle-type nicotinic acetylcholine receptor (nAChR) with excellent selectivity for α/δ receptor subunit binding over α/γ.
  3. GC26032 Varenicline (CP 526555) dihydrochloride

    Chantix, Champix,CP 526555 dihydrochloride

     Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation.
  4. GC25994 Thonzylamine

    Neohetramine

     Thonzylamine (Neohetramine) is an antihistamine and anticholinergic drug.
  5. GC25583 Lobelin sulphate

    Lobeline sulfate, Bantron

     Lobelin sulphate (Lobeline sulfate, Bantron) is an alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has a variety of therapeutic uses including in respiratory disorders, peripheral vascular disorders, insomnia, and smoking cessation.
  6. GC25387 Ethyl (triphenylphosphoranylidene) acetate

    (Carbethoxymethylene)triphenylphosphorane, Triphenylcarbethoxymethylenephosphorane, Ethyl 2-(triphenylphosphoranylidene)acetate

     Ethyl (triphenylphosphoranylidene) acetate (Triphenylcarbethoxymethylenephosphorane, (Carbethoxymethylene)triphenylphosphorane) may act as an inhibitor of cholinesterase that inhibits AChE and BChE.
  7. GC17885 VU0364572 (trifluoroacetate salt) A selective muscarinic M1 receptor agonist
  8. GC13314 L-Acetylcarnitine (hydrochloride)

    乙酰左旋肉碱,Acetyl-L-Carnitine,ALCAR

     A mitochondrial metabolite
  9. GC12507 ML352 An inhibitor of the presynaptic choline transporter
  10. GC13445 LY2119620

    3-氨基-5-氯-N-环丙基-4-甲基-6-[2-(4-甲基-1-哌嗪基)-2-氧代乙氧基]-噻吩并[2,3-B]吡啶-2-甲酰胺

     A positive allosteric modulator of M2 and M4 mAChRs
  11. GC17627 Nitenpyram

    烯啶虫胺

     An insecticide
  12. GC11128 (±)-Vesamicol hydrochloride

    (±)-AH5183 hydrochloride

     (±)-Vesamicol hydrochloride ((±)-AH5183 hydrochloride) 是一种有效的囊泡乙酰胆碱转运抑制剂，Ki 为 2 nM。
  13. GC13361 Flavoxate hydrochloride

    盐酸黄酮哌酯,Rec-7-0040; DW61

     An internal standard for the quantification of flavoxate
  14. GC10508 Solifenacin hydrochloride

    索利那新盐酸盐,YM905 hydrochloride

     Solifenacin hydrochloride (YM905 hydrochloride) 是一种毒蕈碱受体拮抗剂，对 M1、M2 和 M3 受体的 pKis 分别为 7.6、6.9 和 8.0。
  15. GC14419 Bethanechol chloride

    氯贝胆碱; Carbamyl-β-methylcholine chloride

     A muscarinic acetylcholine receptor agonist
  16. GC14142 Acetylcholine Chloride

    氯化乙酰胆碱; ACh chloride

     A neurotransmitter
  17. GC11773 Pancuronium dibromide

    泮库溴铵

     Pancuronium dibromide 是一种双季铵盐类固醇，是一种神经肌肉松弛剂。
  18. GC10972 Gallamine Triethiodide

    三碘季胺酚

     An allosteric modulator of muscarinic acetylcholine receptors
  19. GC17483 Trospium chloride

    曲司氯铵

     An antagonist of muscarinic receptors
  20. GC13134 Tiotropium Bromide hydrate

    噻托溴铵一水合物,BA-679 BR (hydrate)

     A muscarinic receptor antagonist
  21. GC17229 Paroxetine HCl

    盐酸帕罗西汀; BRL29060 hydrochloride; BRL29060A

     A selective serotonin reuptake inhibitor
  22. GC17825 Methscopolamine

    甲溴东莨菪碱

     A muscarinic acetylcholine receptor antagonist
  23. GC13779 Orphenadrine Citrate

    枸酸芬那君

     Orphenadrine citrate 是一种具有口服活性且非竞争性的 NMDA 受体拮抗剂（穿过血脑屏障），Ki 为 6.0 μM。
  24. GC15150 Tropicamide

    托吡卡胺; Ro 1-7683

     A selective muscarinic M4 antagonist
  25. GC12453 Succinylcholine Chloride Dihydrate

    司可林

     An agonist of muscle-type nAChRs
  26. GC16056 Neostigmine Bromide

    溴化新斯的明; Eustigmin bromide; Neoserine bromide

     溴化新斯的明是一种胆碱酯酶抑制剂，用于治疗重症肌无力。
  27. GC10863 Otilonium Bromide

    奥替溴铵; Octylonium bromide; SP63

     An L- and T-type calcium channel inhibitor and mAChR antagonist
  28. GC11035 Hyoscyamine

    L-莨菪碱; Daturine

     A muscarinic receptor antagonist
  29. GC17908 Homatropine Methylbromide

    溴甲后马托品,Homatropine methobromide

     An anticholinergic agent
  30. GC13897 Homatropine Bromide

    氢溴酸后马托品

     An anticholinergic agent
  31. GC15178 Hexamethonium Bromide

    六甲溴铵

     A nondepolarizing neuromuscular blocking agent
  32. GC16255 Decamethonium Bromide

    十烃溴铵

     A depolarizing neuromuscular blocking agent
  33. GC14703 Oxybutynin chloride

    盐酸奥昔布宁

     An antagonist of muscarinic acetylcholine receptors
  34. GC12920 Pregnenolone

    孕烯醇酮; 3β-Hydroxy-5-pregnen-20-one

     A natural steroid hormone
  35. GC11219 (R)-(+)-Tolterodine

    托特罗定; (R)-(+)-Tolterodine; (+)-Tolterodine; (R)-Tolterodine; PNU-200583

     (R)-(+)-Tolterodine(PNU-200583) 是一种有效的毒蕈碱受体拮抗剂，在体内对膀胱的选择性优于唾液腺。
  36. GC15029 Glycopyrrolate

    格隆溴铵; Glycopyrronium bromide; Glycopyrrolate bromide

     A muscarinic acetylcholine receptor antagonist
  37. GC16059 Tarafenacin D-tartrate

    SVT-40776 D-tartrate

     Tarafenacin D-tartrate (SVT-40776 D-tartrate) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM)，选择性是 M2 受体的约 200 倍。
  38. GC13618 Tarafenacin

    他利那新,SVT-40776

     Tarafenacin(SVT-40776) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM)，选择性比 M2 受体高约 200 倍。
  39. GC16819 VU0152100

    3-氨基-N-[(4-甲氧基苯基)甲基]-4,6-二甲基噻吩并[2,3-B]吡啶-2-甲酰胺,VU152100

     A muscarinic M4 receptor positive allosteric modulator
  40. GC11643 PNU-120596

    NSC 216666

     An α7 neuronal nAChR modulator
  41. GC12717 Ipratropium Bromide

    异丙托溴铵; Sch 1000

     A muscarinic receptor antagonist
  42. GC16635 Diphemanil Methylsulfate

    甲硫二苯马尼,Diphemanil mesylate

     An anticholinergic agent
  43. GC12994 Rivastigmine Tartrate

    酒石酸卡巴拉汀; ENA 713; SDZ-ENA 713

     A cholinesterase inhibitor
  44. GC14113 Oxybutynin

    奥昔布宁

     An antagonist of muscarinic acetylcholine receptors
  45. GC16526 Atropine

    阿托品; Tropine tropate; DL-Hyoscyamine

     A non-selective muscarinic acetylcholine receptor antagonist
  46. GC11786 Acetylcysteine

    乙酰半胱氨酸; N-Acetylcysteine; N-Acetyl-L-cysteine; NAC

     乙酰半胱氨酸是半胱氨酸的 N-乙酰基衍生物。
  47. GC10948 Varenicline Tartrate

    酒石酸伐尼克兰; CP 526555-18

     An agonist of α7 and α4β2 nAChRs
  48. GC11210 Vecuronium Bromide

    维库溴铵; ORG NC 45

     A non-depolarizing muscle relaxant
  49. GC14624 Galanthamine HBr

    氢溴酸加兰他敏

     An alkaloid with AChE inhibitory and nAChR potentiating activities
  50. GC13449 Rocuronium Bromide

    罗库溴铵; ORG 9426 Bromide

     A non-depolarizing muscle relaxant
  51. GC12554 Tiotropium Bromide

    噻托溴铵; BA679 BR

     A muscarinic receptor antagonist

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