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Home >> Signaling Pathways >> Neuroscience >> Dopamine Receptor

Dopamine Receptor(多巴胺受体)

Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.

Products for  Dopamine Receptor

  1. Cat.No. 产品名称 Information
  2. GC35848 Dexpramipexole dihydrochloride

    右旋普拉克索二盐酸盐; (R)-Pramipexole dihydrochloride; R-(+)-Pramipexole dihydrochloride; KNS-760704 dihydrochloride

     An anti-apoptotic antioxidant
  3. GC35847 Dexpramipexole

    右旋普拉克索; (R)-Pramipexole; R-(+)-Pramipexole; KNS-760704

     Dexpramipexole(KNS-760704)也叫R-(+)-Pramipexole，是神经保护剂，是弱的非麦角类多巴胺受体激动剂。
  4. GC35610 Cariprazine hydrochloride

    盐酸卡利拉嗪; RGH188 hydrochloride

     An atypical antipsychotic
  5. GC35492 Benzamide Derivative 1 Benzamide Derivative 1是来自专利EP0213775A1，化合物18，的苯甲酰胺衍生物。Benzamide Derivative 1可能用于治疗胃肠疾病的研究。
  6. GC35323 Amisulpride hydrochloride

    氨磺必利盐酸盐; DAN 2163 hydrochloride

     A dopamine D2 and D3 and 5-HT2B, 5-HT7, and 5-HT7A receptor antagonist
  7. GC35252 Adoprazine

    阿哆嗪; SLV313

     Adoprazine是5-HT1A受体的完全激动剂和D2/3受体的拮抗剂。
  8. GC34949 (-)-Isocorypalmine

    (-)-异延胡索单酚碱,Tetrahydrocolumbamine; (S)-Tetrahydrocolumbamine

     An isoquinoline alkaloid and metabolite of L-THP with diverse biological activities
  9. GC45188 Zuclopenthixol

    珠氯噻醇,(Z)-Clopenthixol

     A dopamine receptor antagonist
  10. GC43660 Fenoldopam (mesylate)

    非诺多泮甲磺酸盐; Fenoldopam methanesulfonate; SKF-82526 mesylate

     An agonist of dopamine D1A and D1B receptors
  11. GC41486 Glaucine

    海罌粟鹼,O,O-Dimethylisoboldine; S-(+)-Glaucine; NSC 34396

     An Analytical Reference Standard
  12. GC19499 A-381393 A-381393 是一种有效的、选择性的脑穿透多巴胺 D4 受体拮抗剂，对人多巴胺 D4.4、D4.2 和 D4.7 受体的 Kis 分别为 1.5、1.9 和 1.6 nM，比选择性高 2700 倍以上D1、D2、D3 和 D5 多巴胺受体。
  13. GC33730 Pentiapine (CGS 10746)

    喷硫平,CGS 10746

     Pentiapine (CGS 10746) (CGS 10746) 是一种多巴胺释放抑制剂，不与突触多巴胺受体位点结合。
  14. GC33727 SKF 82958 ((±)-SKF 82958)

    (+/-)-6-氯-7,8-二羟基-3-烯丙基-1-苯基-2,3,4,5-四氢-1H-3-苯氮杂卓氢溴酸,(±)-SKF-82958; Chloro-APB

     SKF 82958 ((±)-SKF 82958) ((±)-SKF 82958) 是一种多巴胺 D1 受体完全激动剂 (K0.5=4 nM)，对 D1 的选择性优于对 D2 受体 (K0.5=73 nM) ）。
  15. GC33664 SKF-82958 hydrobromide ((±)-SKF 82958 hydrobromide)

    (±)-SKF-82958 hydrobromide; Chloro-APB hydrobromide

     A dopamine D1 receptor agonist
  16. GC33552 ABT-670

    ABT-670是一种具有选择性，可口服的dopamineD4受体抑制剂。
  17. GC33544 (±)-Methotrimeprazine (D6) (dl-Methotrimeprazine D6)

    (±)-Methotrimeprazine-d6; dl-Methotrimeprazine-d6

     (±)-Levomepromazine D6 ((±)-Methotrimeprazine D6) 是氘标记的 Methotrimeprazine，它是一种 D3 多巴胺和组胺 H1 受体拮抗剂。
  18. GC33527 Trimethobenzamide hydrochloride (Ro 2-9578)

    盐酸三甲氧苯酰胺,Ro 2-9578

     A dopamine D2 receptor antagonist and antiemetic
  19. GC33510 Org-10490 Org-10490是一种dopamineD1受体和dopamineD2受体的拮抗剂，常用于治疗神经疾病。
  20. GC31418 Clebopride malate

    苹果酸氯波必利

     Clebopride is a dopamine antagonist drug and is used to treat functional gastrointestinal disorder such as nausea or vomiting.
  21. GC31287 U91356 U91356是一种多巴胺受体(dopaminereceptor)激动剂。
  22. GC31278 BP 897

    N-[4-[4-(2-甲氧基苯基)-1-哌嗪基]丁基]-2-萘甲酰胺单盐酸盐

     A dopamine D3 receptor partial agonist
  23. GC31225 PF-592379 PF-592379是一种有效的多巴胺D3受体激动剂，EC50为21nM。
  24. GC31214 A-437203 (Lu201640)

    Lu201640; A37203

     A-437203 (Lu201640) 是一种选择性 D3 受体拮抗剂，对 D2、D3 和 D4 受体的 Ki 分别为 71、1.6 和 6220 nM。
  25. GC31188 Sultopride (LIN-1418)

    舒托必利; LIN-1418

     Sultopride (LIN-1418) (LIN-1418) 是多巴胺 D2 受体的选择性拮抗剂。
  26. GC31183 Piperidine-MO-1 Piperidine-MO-1是来自专利WO/2005/121087A1化合物实例2的多巴胺受体(dopaminereceptor)调节剂，在大鼠纹状体中增加DOPAC的ED50值为68μmol/kg。
  27. GC31173 Ocaperidone (R79598)

    奥卡哌酮,R79598

     Ocaperidone (R79598) 是一种有效的抗精神病药，作为有效的 5-HT2 和多巴胺 D2 拮抗剂和 5-HT1A 激动剂，对 5-HT2 的 Kis 分别为 0.14 nM、0.46 nM、0.75 nM、1.6 nM 和 5.4 nM 、a1-肾上腺素受体、多巴胺 D2、组胺 H1 和 a2-肾上腺素受体，h5-HT1A 的 pEC50 和 pKi 分别为 7.60 和 8.08。
  28. GC31111 NMI 8739

    DHA-DA, NMI 8739

     A conjugate of DHA and dopamine
  29. GC31069 Pardoprunox (SLV-308)

    SLV-308; DU-126891

     Pardoprunox hydrochloride (DU-126891, SME-308) is a potent but partial dopamine D2 receptor agonist with pEC50 of 8.0, and a partial agonist in the induction of [35S]GTPγS binding with pEC50 of 9.2 and a serotonin 5-HT1A receptor agonist, with pEC50 of 6.3, respectively.
  30. GC31055 Abaperidone

    阿巴哌酮

     Abaperidone是一种有效的5-HT2A受体和多巴胺D2受体拮抗剂，IC50分别为6.2和17nM。
  31. GC31047 Bromopride

    溴必利；溴灭吐灵

     A dopamine D2 receptor antagonist
  32. GC31037 Clocapramine (Clocarpramine)

    Clocarpramine; 3-Chlorocarpipramine

    Clocapramine是多巴胺D2和5-HT2A受体拮抗剂。
  33. GC31018 NEO 376 (SPI-376)

    SPI-376

     NEO 376 (SPI-376) 是 5-HT1 受体、GABA 受体和多巴胺受体的选择性调节剂，具有抗精神病活性。
  34. GC31015 NRA-0160 NRA-0160是一种选择性的dopamineD4receptor拮抗剂，Ki值为0.48nM；同时对dopamineD2receptor，D3receptor，大鼠5-HT2Areceptor和α1adrenoceptor分别具有不同程度的亲和度，Ki值分别为>10000nM，39nM，180nM和237nM。
  35. GC30995 CGP 25454A CGP25454A是一个新颖和选择性的突触前多巴胺自受体拮抗剂。
  36. GC30980 Pardoprunox hydrochloride (SLV-308 hydrochloride)

    盐酸帕多芦诺,SLV-308 hydrochloride; DU-126891 hydrochloride

     A dopamine D2 and D3 receptor partial agonist and 5-HT1A agonist
  37. GC30975 Tiapride hydrochloride

    盐酸硫必利

     Tiapride is a drug that selectively blocks D2 and D3 dopamine receptors in the brain and is used to treat a variety of neurological and psychiatric disorders.
  38. GC30974 Promazine hydrochloride

    盐酸丙嗪; Romtiazin hydrochloride; Ampazine hydrochloride; Berophen hydrochloride

     Promazine (Romtiazin, Sinophenin) is an antagonist at types 1, 2, and 4 dopamine receptors, 5-HT receptor types 2A and 2C, muscarinic receptors 1 through 5, alpha(1)-receptors, and histamine H1-receptors with antipsychotic effects.
  39. GC30944 Sultopride hydrochloride (LIN-1418 hydrochloride)

    盐酸舒必利; LIN-1418 hydrochloride

     Sultopride hydrochloride (LIN-1418 hydrochloride) (LIN-1418 hydrochloride) 是多巴胺 D2 受体的选择性拮抗剂。
  40. GC30926 Lurasidone (SM-13496)

    鲁拉西酮; SM-13496

     An atypical antipsychotic
  41. GC30904 Molindone hydrochloride (EN-1733A)

    EN-1733A

     A dopamine receptor antagonist
  42. GC30871 Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride)

    6-羟基多巴胺盐酸盐; 6-Hydroxydopamine hydrochloride; 6-OHDA hydrochloride

     Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride)（6-OHDA）是神经递质多巴胺的拮抗剂。
  43. GC30854 Pridopidine (ACR16)

    4-[3-(甲磺酰基)苯基]-1-丙基哌啶,ACR16; ASP2314; FR310826

     Pridopidine (ACR16, ASP2314, FR310826) , a dopamine (DA) stabilizer, acts as an antagonist against sigma 1 receptor (S1R) and dopamine D2 receptor (D2R).
  44. GC30848 (+)-PD 128907 hydrochloride

    (+)-PD128907,盐酸盐

    A potent D3 receptor agonist
  45. GC30840 Quinagolide hydrochloride (CV205-502 hydrochloride)

    盐酸喹高利特; CV205-502 hydrochloride

    Quinagolide hydrochloride (CV205-502 hydrochloride) 是一种选择性多巴胺 D2 受体激动剂，也是一种催乳素抑制剂。
  46. GC30824 Veralipride ((±)-Veralipride)

    维拉必利,(±)-Veralipride; LIR166

    Veralipride ((±)-Veralipride) 是一种 D2 受体拮抗剂。
  47. GC30797 lumateperone Tosylate (ITI-007)

    1-(4-氟苯基)-4-[(6BR,10AS)-2,3,6B,9,10,10A-六氢-3-甲基-1H-吡啶并[3',4':4,5]吡咯并[1,2,3-DE]喹喔啉-8(7H)-基]-1-丁酮对甲苯磺酸盐,ITI-007 tosylate

    An atypical antipsychotic
  48. GC30790 Triflupromazine hydrochloride

    盐酸三氟丙嗪

     A phenothiazine with diverse biological activities
  49. GC30787 Sertindole (Lu 23-174)

    舍吲哚; Lu 23-174

     An atypical antipsychotic
  50. GC30772 Dopamine serotonin antagonist-1

    氯氮平杂质,Deschloroclozapine

     Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs (muscarinic Designer Receptors Exclusively Activated by Designer Drugs) agonist, and binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively.
  51. GC30396 Piribedil D8 (ET-495 D8)

    吡贝地尔D8,ET-495 D8

     Piribedil D8 (ET-495 D8) (ET-495 D8) 是氘标记的 Piribedil，它是一种抗帕金森病药物。

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