Dopamine Receptor(多巴胺受体)
Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.
Products for Dopamine Receptor
- Cat.No. 产品名称 Information
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GC30375
Clomipramine D3
Chlorimipramine-d3; G-34586-d3; NSC-169865-d3
An Analytical Reference Standard -
GC30280
Chlorpromazine D6 hydrochloride
盐酸氯丙嗪 D6
An internal standard for the quantification of chlorpromazine -
GC30241
GSK598809
GSK598809是多巴胺D3受体(DRD3)的选择性拮抗剂,其pKi值为8.9。
- GC19176 GSK163090 GSK163090 是一种有效的、选择性的和具有口服活性的 5-HT1A/1B/1D 受体拮抗剂,pKi 值分别为 9.4/8.5/9.7。
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GC10260
cis-Flupenthixol (hydrochloride)
顺式-(Z)-氟哌噻吨二盐酸盐,cis-Flupentixol
A typical antipsychotic - GC12466 FAUC-365 A dopamine D3 receptor antagonist
- GC13786 (±)-Salsolinol (hydrochloride) A metabolite of ethanol that targets dopaminergic neurons
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GC11243
Halopemide
卤培米特,NSC 354856,R34301
Inhibitor of phospholipase D1 and D2 -
GC14281
L-DOPA methyl ester (hydrochloride)
盐酸左旋多巴甲酯,3,4-Dihydroxyphenylalanine methyl ester,LDME,Levodopa methyl ester,ST 41769
A dopamine precursor -
GC10643
Pimozide
匹莫齐特; R6238
A dopamine receptor antagonist -
GC17656
Chlorprothixene (hydrochloride)
氯普噻吨盐酸盐;泰尔登盐酸盐;氯丙硫蒽盐酸盐
A dopamine D2 receptor antagonist -
GC16782
Benocyclidine
N-[1-(2-苯并[B]噻嗯-2-基)环己基)]哌啶马来酸
An Analytical Reference Standard -
GC12293
Perphenazine
奋乃静
A typical antipsychotic -
GC14559
Fluphenazine dihydrochloride
盐酸氟奋乃静
A dopamine D1 and D2 receptor antagonist -
GC17729
SKF38393 HCl
(±)-SKF-38393 hydrochloride; SKF-38393A
SKF38393 HCl 是一种多巴胺 D1 受体 (D1DR) 的选择性激动剂,IC50 为 110 nM。 -
GC17047
Threo-methylphenidate hydrochloride
盐酸哌甲酯
盐酸苏哌甲酯(Threo-methylphenidate hydrochloride)是一种儿茶酚胺再摄取抑制剂,抑制多巴胺转运蛋白(DAT)和去甲肾上腺素转运蛋白(NET)。 - GC12800 PAOPA dopamine D2 receptor modulator
- GC14610 A 412997 dihydrochloride Selective D4 agonist
- GC13036 L-741,742 hydrochloride highly potent and selective D4 dopamine receptor antagonist
- GC14569 L-745,870 trihydrochloride L-745,870 trihydrochloride 是一种有效的、选择性的、脑渗透性和口服活性的多巴胺 D4 受体拮抗剂,Ki 为 0.43 nM。
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GC17527
(+)-Dihydrexidine hydrochloride
(+)-DAR-0100 hydrochloride
(+)-Dihydrexidine hydrochloride ((+)-DAR-0100 hydrochloride) 是一种多巴胺 D1 受体激动剂,EC50 为 72± 21 nM。
- GC14873 2-CMDO Dopamine D2-like receptor antagonist
- GC17841 JHW 007 hydrochloride Dopamine uptake inhibitor
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GC13183
SB 277011A dihydrochloride
SB-277011A dihydrochloride
A selective dopamine D3 antagonist -
GC12015
Sonepiprazole
PNU-101387G; U-101387G
A selective D4 receptor antagonist -
GC16730
Lisuride maleate
New Product
- GC14593 GSK 789472 hydrochloride dopamine D3 receptor antagonist and D2 partial agonist
- GC11810 PG 01037 dihydrochloride A selective dopamine D3 receptor antagonist
- GC14280 PD 168568 dihydrochloride PD 168568 dihydrochloride 是一种具有口服活性的选择性 D4 多巴胺受体拮抗剂,Ki 为 8.8 nM。
- GC15763 PNU 177864 hydrochloride dopamine D3 receptor antagonist
- GC14694 NGD 94-1 High affinity D4 receptor ligand
- GC11902 PNU 96415E PNU 96415E 是一种选择性 D4/5-HT2A 拮抗剂。
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GC13109
Fananserin
法南色林,RP 62203
Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂,对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。 - GC18068 NGB 2904 A selective D3 antagonist
- GC17238 OSU 6162 hydrochloride Dopamine stabilizer
- GC12428 Ro 10-5824 dihydrochloride Ro 10-5824 dihydrochloride 是一种选择性多巴胺 D4 受体部分激动剂,Ki 为 5.2 nM。
- GC16992 SCH 39166 hydrobromide A dopamine D1 receptor antagonist
- GC11795 ABT 724 trihydrochloride A dopamine D4 receptor agonist
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GC14826
Carmoxirole hydrochloride
EMD 45609 hydrochloride
Carmoxirole hydrochloride (EMD 45609 hydrochloride) 是一种选择性的、外周作用的多巴胺 D2 受体激动剂,在体内表现出抗高血压活性。 - GC11503 SKF 83822 hydrobromide SKF 83822 hydrobromide 是一种有效的多巴胺 D1 受体激动剂。
- GC11146 SKF 83959 hydrobromide A dopamine D1 and D5 receptor partial agonist
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GC12355
Eticlopride hydrochloride
依替必利盐酸盐
A dopamine D2 and D3 receptor antagonist -
GC16769
Raclopride
雷氯必利
A dopamine D2/D3 receptor antagonist -
GC12543
Nemonapride
顺-5-氯-2-甲氧基-4-(甲基氨基)-N-[2-甲基-2-(苯基甲基)-3-吡咯烷基]苯甲酰胺,YM-09151-2; Emilace; Emonapride
An antipsychotic - GC11183 A 77636 hydrochloride A dopamine D1 receptor agonist
- GC13169 SKF 77434 hydrobromide A dopamine D1 receptor partial agonist
- GC15016 SKF 83566 hydrobromide A dopamine D1 receptor antagonist
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GC10745
Roxindole hydrochloride
EMD 38362
Roxindole hydrochloride (EMD 38362) 是一种吲哚烷基哌啶,是一种有效的多巴胺自身受体激动剂,对低纳摩尔范围内的 D2 样亚型具有亲和力。 -
GC15498
A 68930 hydrochloride
1-(氨基甲基)-3,4-二氢-3-苯基-1H-2-苯并吡喃-5,6-二醇盐酸盐
A 68930 hydrochloride 作为多巴胺 D1 受体激动剂,可用于支气管扩张的研究。 -
GC12158
SKF 81297 hydrobromide
(±)6chloroPB
A selective dopamine D1-like receptor agonist