Dopamine Receptor(多巴胺受体)
Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.
Products for Dopamine Receptor
- Cat.No. 产品名称 Information
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GC16903
GR 103691
A dopamine D3 receptor antagonist
-
GC17634
PD 168077 maleate
A dopamine D4 receptor agonist
-
GC17877
(-)-Quinpirole hydrochloride
(-)-LY 171555
(-)-Quinpirole hydrochloride ((-)-LY 171555) 是一种多巴胺 D2/D3 受体的高亲和力激动剂。 -
GC11602
Piribedil dihydrochloride
盐酸吡贝地尔;盐酸双哌嘧啶;盐酸泰舒达
A dopamine receptor agonist -
GC15619
L-741,626
A dopamine D2 receptor antagonist
-
GC10892
SCH 23390 hydrochloride
R-(+)-SCH-23390 hydrochloride
SCH 23390 hydrochloride 是一种高效的选择性多巴胺 D1 样受体拮抗剂,对 D1 和 D5 多巴胺受体亚型的 K(i) 分别为 0.2 和 0.3 nM。 -
GC15606
3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride
dopamine uptake and transport inhibitor
-
GC12641
3-CPMT
dopamine uptake inhibitor
-
GC14822
Remoxipride hydrochloride
瑞莫必利盐酸盐
An atypical antipsychotic -
GC12870
(+)-UH 232 maleate
顺-(+)-5-甲氧基-1-甲基-2-(二正丙基氨基)萘满马来酸
D2 antagonist -
GC14311
4-Phenyl-1,2,3,4-tetrahydroisoquinoline hydrochloride
dopamine release inhibitor
-
GC16916
7-Hydroxy-PIPAT maleate
D3 receptor agonist
-
GC16574
7-Hydroxy-DPAT hydrobromide
A dopamine D3 receptor agonist
-
GC11945
BTCP maleate
dopamine reuptake inhibitor
-
GC15856
3'-Fluorobenzylspiperone maleate
ligand for the D2 receptor
-
GC13156
(+)-AJ 76 hydrochloride
Dopamine receptor antagonist
-
GC16049
AMI-193
螺哌丙苯,AMI-193
AMI-193 (AMI-193) 是一种有效的、选择性的 5-HT2 和多巴胺 D2 受体拮抗剂,Kis 分别为 2 nM 和 3 nM。 -
GC12456
GBR 12783 dihydrochloride
GBR 12783 dihydrochloride 是一种特异性、有效和选择性的多巴胺摄取抑制剂,抑制大鼠和小鼠纹状体突触体对 [3H] 多巴胺的摄取,IC50 分别为 1.8 nM 和 1.2 nM。
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GC12179
GBR 13069 dihydrochloride
dopamine uptake inhibitor
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GC14865
RuBi-Dopa
dopamine receptor activator
-
GC15326
Flupenthixol dihydrochloride
盐酸氟哌噻吨,Flupenthixol dihydrochloride
Flupentixol 是一种具有口服活性的 D1/D2 多巴胺受体拮抗剂和新型 PI3K 抑制剂(PI3Kα;IC50=127 nM)。 -
GC17075
NPEC-caged-dopamine
Dopamine receptor agonist
-
GC16267
6-Hydroxydopamine hydrobromide
6-羟基多巴胺氢溴酸盐; 6-Hydroxydopamine hydrobromide; 6-OHDA hydrobromide
6-Hydroxydopamine hydrobromide (6-OHDA) 是儿茶酚胺、多巴胺和去甲肾上腺素的结构类似物,对儿茶酚胺能神经元发挥毒性作用。 -
GC13573
Nomifensine
诺米芬辛; (±)-Nomifensin
An inhibitor of norepinephrine and dopamine reuptake -
GC17890
LE 300
A dopamine D1-like and 5-HT2A receptor antagonist
-
GC17192
Quinelorane hydrochloride
LY163502
Quinelorane hydrochloride (LY163502) 是一种有效的多巴胺 D3/D2 受体激动剂。 -
GC14048
SKF 38393 hydrobromide
(±)-SKF-38393 hydrobromide
A partial agonist of dopamine D1-like receptors -
GC10349
(RS)-(±)-Sulpiride
舒必利
An atypical antipsychotic -
GC13931
Bromocriptine mesylate
甲磺酸溴隐亭; CB-154
A dopamine receptor agonist -
GC13853
GBR 12935 dihydrochloride
An inhibitor of dopamine uptake
-
GC14657
Rotundine
罗通定; (-)-Tetrahydropalmatine; L-Tetrahydropalmatine
An antinociceptive alkaloid -
GC10441
Cabergoline
卡麦角林; FCE-21336
A potent and selective dopamine D2 receptor agonist -
GC11028
Dopamine HCl
盐酸多巴胺,ASL279
An endogenous catecholamine -
GC10144
Domperidone
多潘立酮; R33812
A dopamine D2 receptor antagonist -
GC15107
Clomipramine HCl
盐酸氯米帕明; Chlorimipramine hydrochloride; G-34586 hydrochloride; NSC-169865 hydrochloride
A tricyclic antidepressant -
GC14216
Chlorpromazine HCl
盐酸氯丙嗪
Chlorpromazine HCl是一种口服有效的、可透过血脑屏障的吩噻嗪类抗精神病药,能够有效抑制D2多巴胺受体和5-HT2A,具有很强的镇静作用。 -
GC15546
Alizapride HCl
盐酸阿立必利
A dopamine D2 receptor antagonist -
GC14759
Fenoldopam
非诺多泮; SKF 82526
An agonist of dopamine D1A and D1B receptors -
GC15470
Levosulpiride
左舒必利; RV-12309; S-(-)-Sulpiride
左舒必利 (RV-12309) 是舒必利的 (S)-对映异构体,是一种 D2 受体拮抗剂,是苯甲酰胺类的非典型抗精神病药物。 -
GC16783
Pramipexole 2HCl Monohydrate
普拉克索盐酸盐水合物
Pramipexole 2HCl Monohydrate 是一种选择性和血脑屏障 (BBB) 渗透性多巴胺 D2 型受体激动剂,对 D2 型受体、D2、D3 和 D4 受体的 Kis 分别为 2.2 nM、3.9 nM、0.5 nM 和 1.3 nM . -
GC11960
Pramipexole
普拉克索
Pramipexole 是一种选择性和血脑屏障 (BBB) 渗透性多巴胺 D2 型受体激动剂,对 D2 型受体、D2、D3 和 D4 受体的 Kis 分别为 2.2 nM、3.9 nM、0.5 nM 和 1.3 nM。 -
GC10105
Amantadine HCl
盐酸金刚烷胺; 1-Adamantanamine hydrochloride; 1-Adamantylamine hydrochloride; 1-Aminoadamantane hydrochloride
An NMDA receptor antagonist and antiviral agent -
GC15754
WAY-100635 Maleate
A serotonin 5-HT1A antagonist
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GC13031
Trifluoperazine 2HCl
盐酸三氟拉嗪;甲哌氟丙嗪;三氟吡拉嗪
An anti-adrenergic and anti-dopaminergic agent -
GC11462
Ropinirole HCl
盐酸罗匹尼罗; SKF 101468 hydrochloride
A dopamine D2 receptor agonist -
GC16615
Pergolide mesylate
甲磺酸培高利特; Pergolide methanesulfonate; LY127809
A dopamine D1 and D2 receptor agonist -
GC17600
PD128907 HCl
A potent D3 receptor agonist
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GC10808
Droperidol
氟哌啶; Dehydrobenzperidol
A dopamine D2 and D4 receptor antagonist -
GC16229
Azaperone
阿扎哌隆,R-1929
An Analytical Reference Standard -
GC17593
Lurasidone HCl
盐酸鲁拉西酮; SM-13496 Hydrochloride
An atypical antipsychotic