GluR(谷氨酸受体)
GluR (glutamate receptor) is a group of synaptic receptors located primarily on the membranes of neuronal cells.
Products for GluR
- Cat.No. 产品名称 Information
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GC17079
ACDPP hydrochloride
mGlu5 receptor antagonist
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GC11223
3-MATIDA
mGlu1 receptor antagonist
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GC13126
DMeOB
Negative allosteric modulator of mGlu5
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GC15385
DCB
DCB (3,3'-dichlorobenzaldazine) 是代谢型谷氨酸受体代谢型谷氨酸受体亚型 5 (mGluR5) 的中性变构调节剂。
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GC10739
(S)-HexylHIBO
Group I mGlu receptor antagonist
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GC17446
HexylHIBO
HexylHIBO 是一种有效的 I 组 mGluR 拮抗剂,对 mGlu1a 和 mGlu5a 受体的 Kb 值分别为 140 和 110 μM。
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GC11246
DFB
DFB
A positive allosteric modulator of mGluR5 -
GC14227
MNI-caged-L-glutamate
MNI-caged-L-glutamate是L-谷氨酸的稳定光释放剂。
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GC17722
(R)-3,4-DCPG
AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors
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GC16542
(RS)-3,4-DCPG
antagonist of AMPA receptors and agonist of mGluR8
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GC13046
UBP1112
group III mGlu receptor antagonist
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GC14639
(S)-3,4-DCPG
(S)-3,4-二甲酸苯基甘氨酸,(S)-3,4-Dicarboxyphenylglycine
A selective agonist of mGluR8 -
GC12831
LY 367385
An antagonist of mGluR1α
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GC11433
(RS)-PPG
4-磷酰基苯甘氨酸
(RS)-PPG 是 III 组 mGluR 的有效选择性激动剂。 -
GC11233
SIB 1757
An antagonist of mGluR5a
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GC10452
SIB 1893
2-甲基-6-(2-苯乙烯基)吡啶
SIB 1893 是 (E)-SIB-1893 和 (Z)-SIB-1893 异构体的外消旋化合物。 -
GC11379
(2R,4R)-APDC
(2R,4R)-APDC 是一种选择性 II 族代谢型谷氨酸受体 (mGluRs) 激动剂。
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GC11771
(RS)-APICA
(RS)-APICA 是一种选择性 II 组代谢型谷氨酸受体 (mGluR II) 拮抗剂。
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GC12532
CHPG
Chlorohydroxyphenylglycine, CHPG
A potent and selective mGluR5 agonist -
GC18134
CPCCOEt
An mGluR1b antagonist
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GC17383
PHCCC
N-苯基-7-(羟基亚胺基)环丙烯并[B]苯并吡喃-1A-甲酰胺
PHCCC 是 I 组 mGluR 拮抗剂,IC50 为 3 μM。 PHCCC 是 mGlu4 受体的选择性正调节剂。抗帕金森效应。 -
GC13192
E4CPG
(RS)-ECPG
An antagonist of mGluR1 and mGluR2 -
GC12100
CPPG
(RS)-CPPG
An antagonist of group II and group III mGluRs -
GC17326
EGLU
(2S)-α-Ethylglutamic acid; (2S)-α-EGLU
EGLU ((2S)-α-Ethylglutamic acid; (2S)-α-EGLU) 是一种有效的竞争性 mGluR-2 受体拮抗剂。 -
GC14146
AIDA
AIDA
AIDA (AIDA) 是一种刚性(羧基苯基)甘氨酸衍生物,是一种相对有效和选择性的 I 组代谢型谷氨酸受体 (mGlu1a) 拮抗剂,IC50 为 214 μM. -
GC11428
MTPG
MTPG 是一种有效的 mGluR2 和 mGluR3 拮抗剂。
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GC13548
MSPG
mGlu receptor antagonist
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GC15769
MPPG
MPPG 是一种有效的选择性 L-AP4 敏感受体拮抗剂,kD 值为 9.2 μM,正在新生大鼠脊髓上进行测试。
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GC16858
(S)-3,5-DHPG
(S)-3,5-二羟基苯基甘氨酸
A selective agonist of group I mGluRs -
GC17185
MSOP
MSOP 是一种选择性 III 族代谢型谷氨酸受体拮抗剂,对 L-AP4 敏感的突触前 mGluR 的表观 KD 为 51 μM。
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GC11571
MAP4
(S)-2-氨基-2-甲基-4-磷酰丁酸
MAP4 在某些电生理系统中是一种选择性 III 组 mGluR 拮抗剂。 -
GC11269
Salsolinol-1-carboxylic acid
Salsolinol-1-carboxy acid 是中枢神经系统 (CNS) 中的一种内源性生物碱。
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GC13222
N-Acetylglycyl-D-glutamic acid
Excitatory peptide that induces seizures
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GC15136
L-AP6
DL-2-氨基-6-膦酰己酸
selective agonist for 'quis'-sensitized site -
GC16349
(S)-MCPG
(+)-MCPG
An mGluR antagonist -
GC12279
(RS)-MCPG
alpha-MCPG
(RS)-MCPG (alpha-MCPG) 是一种竞争性和选择性的 I 组/II 组代谢型谷氨酸受体 (mGluR) 拮抗剂。 -
GC11536
(S)-3-Carboxy-4-hydroxyphenylglycine
group I metabotropic glutamate receptor antagonist and group II mGlu agonist
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GC14124
(R)-3-Carboxy-4-hydroxyphenylglycine
NMDA and AMPA/kainate receptor antagonist
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GC16234
(S)-3-Hydroxyphenylglycine
(S)-3-羟基苯甘氨酸
group I metabotropic glutamate receptors agonist -
GC12985
(RS)-3-Hydroxyphenylglycine
3-羟基苯甘氨酸
PI-linked metabotropic glutamate receptors agonist -
GC14176
(S)-4-Carboxyphenylglycine
group I metabotropic glutamate receptor antagonist
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GC13773
(RS)-4-Carboxyphenylglycine
broad spectrum EAA ligand
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GC12012
(S)-4-Carboxy-3-hydroxyphenylglycine
group I mGlu1a/1a receptor antagonist and mGluR2 agonist
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GC13288
(RS)-4-Carboxy-3-hydroxyphenylglycine
(RS)-4-羧基-3-羟基苯甘氨酸
broad spectrum EAA agonist/antagonist -
GC16207
(1S,3R)-ACPD
反-(1S,3R)-1-氨基-1,3-环戊烷二羧酸
group I and II mGlu receptor agonist -
GC14752
2,4-Dihydroxyphenylacetyl-L-asparagine
glutamate receptors blocker
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GC12394
(±)-trans-ACPD
Trans-(±)-ACP
An mGluR agonist -
GC10026
S-Sulfo-L-cysteine sodium salt
EAA receptor agonist
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GC12063
D-AP4
D(-)-2-氨基-4-磷酸基丁酸,D-APB; D-2-Amino-4-phosphonobutyric acid
D-AP4 (D-APB; D-2-Amino-4-phosphonobutyric acid) 是一种谷氨酸的膦酰基类似物,是一种 NMDA 广谱兴奋性氨基酸受体拮抗剂。 -
GC15435
RuBi-Glutamate
Ruthenium-bipyridine-trimethylphosphine caged glutamate