Adrenergic Receptor(肾上腺素能受体)
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
Products for Adrenergic Receptor
- Cat.No. 产品名称 Information
- GC31329 Ko-3290 Ko-3290是一种β-adrenoceptor拮抗剂,在动物试验中,具有心脏选择性和抗脂肪分解的特点。
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GC36413
L-(-)-α-Methyldopa hydrate
L-甲基多巴,L-(-)-α-Methyldopa hydrate; MK-351 hydrate
L-(-)-α-Methyldopa (Methyldopa, MK-351) hydrate, a potent antihypertensive drug, is a selective agonist for α2-adrenergic receptors. -
GC16401
L-(-)-α-Methyldopa hydrochloride
L-3-(3,4-二羟基苯基)-2-甲基丙氨酸盐酸盐,L-(-)-α-Methyldopa hydrochloride; MK-351 hydrochloride
A DOPA decarboxylase inhibitor - GC16939 L-748,337 A selective β3-adrenergic receptor antagonist
- GC15743 L-755,507 A selective β3-adrenergic receptor partial agonist
- GC32670 L-765314 L-765314 is a selective and potent α1b-adrenoceptor (α1b adrenergic receptor) antagonist with an IC50 of 1.90 nM and Kis of 5.4 and 2.0 for rat and human α1b adrenergic receptor, respectively.
- GC33410 L-771688 L-771688是一个选择性α1A-Adrenoceptor受体拮抗剂,Ki值为0.43±0.02nM。
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GC14816
L-Adrenaline
肾上腺素,L(-)-Epinephrine
An adrenergic receptor agonist -
GC17319
L-Phenylephrine
去氧肾上腺素; (R)-(-)-Phenylephrine; L-Phenylephrine
A selective adrenergic α1A receptor agonist -
GC64143
Labetalol
拉贝洛尔,AH5158; Sch-15719W free base
An antagonist of α- and β-adrenoreceptors -
GC10887
Labetalol HCl
盐酸拉贝洛尔; AH-5158 hydrochloride; Sch-15719W
An antagonist of α- and β-adrenoreceptors -
GC36422
Landiolol hydrochloride
盐酸兰地洛尔; ONO1101 hydrochloride
Landiolol hydrochloride (ONO-1101) is the hydrochloride salt form of Landiolol, which is an ultra-short-acting β1 selective adrenoceptor antagonist. -
GC17974
Latrepirdine dihydrochloride
2,3,4,5-四氢-2,8-二甲基-5-[2-(6-甲基-3-吡啶基)乙基]-1H-吡啶并[4,3-B]吲哚二盐酸盐,Dimebolin dihydrochloride
A neuroprotective agent -
GC36441
Levalbuterol tartrate
左旋沙丁胺醇酒石酸盐,Levosalbutamol tartrate
Levalbuterol HCl(Levosalbutamol tartrate) is a relatively selective beta2-adrenergic receptor agonist used for the treatment of asthma. -
GC17653
Levobetaxolol HCl
左旋倍他洛尔; (S)-Betaxolol hydrochloride; AL-1577A
A β1-adrenergic receptor antagonist -
GC30972
Lidanserin (ZK-33839)
利丹色林,ZK-33839
Lidanserin (ZK-33839) (ZK-33839) 作为 5-HT2A 和 α1-肾上腺素能受体拮抗剂起作用。 -
GC36477
Lofexidine
洛非西定
An α2-adrenergic receptor agonist -
GC17064
Lofexidine (hydrochloride)
盐酸洛非西定; Baq-168; MDL-14042
An α2-adrenergic receptor agonist -
GC67977
Lubabegron
LY-488756
Lubabegron 是一种有效的 β-肾上腺素受体 (β-AR) 调节剂。Lubabegron 在牛中表现出对 β1 和 β2 受体亚型的拮抗行为和对 β3 受体亚型的激动行为。Lubabegron 可减少动物或其废物的 NH3 气体排放。 -
GC31266
Lusaperidone (R107474)
R107474
Lusaperidone (R107474) (R107474) 是一种 α2 肾上腺素能受体拮抗剂,α2A 和 α2C 的 Kis 分别为 0.13 和 0.15 nM。 - GC69416 LY377604 LY377604 是一种人类 β3-肾上腺素受体激动剂,其 EC50 值为 2.4 nM,同时也是 β1 和 β2 肾上腺素能受体的拮抗剂。
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GC63054
Mabuterol-D9
马布特罗-D9
Mabuterol-D9 是 Mabuterol 的一种氘代化合物。Mabuterol 是 β2-肾上腺素能受体 (β2-adrenergic receptor) 激动剂。 -
GC12376
Maprotiline HCl
盐酸马普替林
A tricyclic antidepressant -
GC13144
Medetomidine
美托咪定
Medetomidine(Domtor) 是一种有效的、高选择性的 α2-adrenoceptor 激动剂(α2-和 α1-adrenoceptors 的 Ki 值分别为 1.08 和 1750 nM)。 -
GC12983
Medetomidine HCl
盐酸美托咪定; MPV785
Medetomidine (hydrochloride) 是一种有效的、选择性的和特异性的 α2-adrenoceptor 激动剂,适用于外周和中枢神经系统。 -
GC65874
Medroxalol
RMI81968
Medroxalol (RMI81968) 是一种具有口服活性的肾上腺素受体拮抗剂,可阻断 α- 和 β- 肾上腺素受体。Medroxalol 具有抗高血压和血管扩张的活性。 -
GC60243
Meranzin
橙皮内酯
A coumarin with diverse biological activities -
GC44169
Metaproterenol (hemisulfate)
硫酸奥西那林,Orciprenaline hemisulfate
A long-acting β2-adrenergic receptor agonist -
GC63067
Methoxyphenamine
甲氧那明,NSC-65644 free base
Methoxyphenamine Hydrochloride (2-methoxy-N-methylamphetamine, OMMA) is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.
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GC63068
Methoxyphenamine hydrochloride
盐酸甲氧那明,NSC-65644
An Analytical Reference Standard - GC71881 Methyl maslinate Methyl maslinate是一种β肾上腺素能拮抗剂。
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GC16490
Methyldopa
甲基多巴; L-(-)-α-Methyldopa; MK-351
A DOPA decarboxylase inhibitor -
GC17888
Metipranolol
美替洛尔
A β-AR antagonist -
GC44185
Metipranolol (hydrochloride)
Trimepranol
A β-AR antagonist -
GC36603
Metoprolol
美托洛尔
Metoprolol is a cardioselective β1-adrenergic blocking agent with log Kd values of ?7.26±0.07, ?6.89±0.09, ?5.16±0.12 for β1, β2, and β3 adrenoceptors, respectively. It is used for acute myocardial infarction, heart failure, angina pectoris and mild to moderate hypertension. -
GC17945
Metoprolol Succinate
琥珀酸美托洛尔
A potent, selective β1-adrenergic receptor blocker -
GC14536
Metoprolol Tartrate
酒石酸美托洛尔
An Analytical Reference Standard - GC71519 Metoprolol-d7 hydrochloride Metoprolol-d7 hydrochloride是氘标记的美托洛尔。
- GC34048 MG 1 MG1是α1肾上腺素能受体拮抗剂。
- GC72193 Mibenratide Mibenratide是一种小环肽,是一种肾上腺素能β1受体拮抗剂。
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GC67691
Midaglizole
(±)-DG5128 free base; DG5128 free base
Midaglizole ((±)-DG5128 free base, DG5128 free base) 是一种有效的 α2-adrenoceptor 拮抗剂。Midaglizole 是一种降血糖药。Midaglizole 在具有升高血压并降低血糖水平的作用。 -
GC31615
Midaglizole hydrochloride ((±)-DG5128)
(±)-DG5128; DG5128
Midaglizole hydrochloride ((±)-DG5128) (DG5128) 是一种优先的 α2-adrenoceptor 拮抗剂。 -
GC11239
Midodrine (hydrochloride)
盐酸米多君; (±)-Midodrine hydrochloride
A prodrug form of desglymidodrine -
GC11915
Mirabegron (YM178)
米拉贝隆; YM178
A β3-AR agonist -
GC48855
Mirtazapine (CRM)
米氮平; Org3770; 6-Azamianserin
An Analytical Reference Material - GC71647 Mirtazapine-d4 Mirtazapine-d4氘标记为米氮平。
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GC32485
Moxisylyte hydrochloride (Thymoxamine hydrochloride)
4-(2-二甲氨基乙氧基)-5-异丙基-2-甲基酯盐酸盐,Thymoxamine hydrochloride
Moxisylyte hydrochloride (thymoxamine) is an alpha-adrenergic blocking agent used for the treatment of Raynaud's disease. -
GC39740
Nadolol
纳多洛尔; SQ-11725
Nadolol (Corgard, Solgol, Anabet, SQ11725) is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities. -
GC36687
Nadolol D9
纳多洛尔 D9; SQ-11725-d9
Nadolol D9是Nadolol氘代化合物标准品。
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GC16836
Naftopidil
萘哌地尔; KT-611; BM-15275
Naftopidil (KT-611) 是一种选择性 alpha1-adrenoceptor 拮抗剂,对克隆的人 α1a-、α1b- 和 α1d-adrenoceptor 亚型的 Kis 分别为 3.7 nM、20 nM 和 1.2 nM。