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Home >> Signaling Pathways >> GPCR/G protein >> Adrenergic Receptor

Adrenergic Receptor(肾上腺素能受体)

Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.

Products for  Adrenergic Receptor

  1. Cat.No. 产品名称 Information
  2. GC44311 Naftopidil (hydrochloride)

    KT-611 hydrochloride; BM-15275 hydrochloride

     An α1-adrenergic receptor antagonist
  3. GC17765 Naftopidil DiHCl

    盐酸萘哌地尔,KT-611 dihydrochloride; BM-15275 dihydrochloride

     Naftopidil DiHCl (KT-611 dihydrochloride) 是一种选择性 alpha1-adrenoceptor 拮抗剂，对克隆人 α1a-, ⋱1b- 和 α1d-adrenoceptor subtypes 的 Kis 分别为 3.7 nM，20 nM 和 1.2 nM。 Naftpidil DiHCl 具有抗增殖作用。 Naftpidil DiHCl可用于前列腺增生的研究。
  4. GC14988 Naphazoline HCl

    盐酸萘甲唑啉; Naphthazoline hydrochloride

     A vasoconstrictor
  5. GC25663 Nebivolol

    Bystolic,R 065824

     Nebivolol (Bystolic,R 065824) is a β1 receptor blocker with nitric oxide-potentiating vasodilatory effect used in treatment of hypertension and also for left ventricular failure.
  6. GC13906 Nebivolol hydrochloride

    盐酸奈必洛尔; R 065824 hydrochloride

     A β1-AR antagonist
  7. GC15786 Nedaplatin

    奈达铂,NSC 375101D

     An anticancer agent
  8. GC16324 Nefazodone hydrochloride

    萘法唑酮盐酸盐,BMY-13754; MJ-13754-1

     A serotonin, norepinephrine, and dopamine reuptake inhibitor
  9. GC70256 Neldazosin Neldazosin是一种有效的α - 1肾上腺素受体拮抗剂。
  10. GC16141 Nicergoline

    尼麦角林

     An α1-AR antagonist
  11. GC14919 Niguldipine (hydrochloride)

    B 844-39,NSC 617553

     An α1A-adrenoceptor antagonist
  12. GC50113 Noradrenaline bitartrate

    L-去甲肾上腺素酒石酸氢盐(酯),Levarterenol tartrate; L-Noradrenaline tartrate

     Norepinephrine (Levarterenol; L-Noradrenaline) tartrate 是一种有效的肾上腺素能受体 (AR) 激动剂。
  13. GC10976 Noradrenaline bitartrate monohydrate

    酒石酸去甲肾上腺素; Levarterenol bitartrate monohydrate; L-Noradrenaline bitartrate monohydrate

     An adrenoceptor agonist
  14. GC30744 Norepinephrine (Adrenor)

    去甲肾上腺素; Levarterenol; L-Noradrenaline

    (-)-Norepinephrine (Arterenol, Levarterenol, L-Noradrenaline) is a natural neurotransmitter and hormone. It is an agonist of adrenergic receptors with Ki values of 330, 56, and 740 nM for α1, α2, and β1 adrenoceptors, respectively.
  15. GC36758 Norepinephrine hydrochloride

    去甲肾上腺素盐酸盐; Levarterenol hydrochloride; L-Noradrenaline hydrochloride

    A racemic mixture of of L-norepinephrine and D-norepinephrine
  16. GC71059 NP10679 NP10679是一种选择性、pH依赖性的GluN2B亚基特异性N-甲基-D-天冬氨酸（NMDA）受体抑制剂，具有高口服生物利用度和良好的脑渗透性。
  17. GC15704 NPEC-caged-noradrenalin Adrenergic receptor agonist
  18. GC31015 NRA-0160 NRA-0160是一种选择性的dopamineD4receptor拮抗剂，Ki值为0.48nM；同时对dopamineD2receptor，D3receptor，大鼠5-HT2Areceptor和α1adrenoceptor分别具有不同程度的亲和度，Ki值分别为>10000nM，39nM，180nM和237nM。
  19. GC61813 O-Desmethyl Mebeverine alcohol hydrochloride

    Mebeverine metabolite O-desmethyl Mebeverine alcohol hydrochloride

     O-DesmethylMebeverinealcoholhydrochloride是Mebeverine的代谢物，Mebeverine是一种有效的α1受体(α1repector)抑制剂，用作消化道的一种解痉药。
  20. GC61809 Olanzapine D3

    奥氮平 D3; LY170053-d3

     OlanzapineD3(LY170053D3)是Olanzapine的氘代物。Olanzapine是一种选择性单胺能拮抗剂，高亲和力结合5-羟色胺H1，5HT2A/2C，5HT3，5HT6(Ki分别为7、4、11、57和5nM)，多巴胺D1-4(Ki=11-31nM)，毒蕈碱M1-5(Ki=1.9-25nM)和肾上腺素α1受体(Ki=19nM)。Olanzapine是一种非典型的抗精神病剂。
  21. GC62219 Olodaterol hydrochloride

    盐酸奥达特罗,BI1744 hydrochloride

     Olodaterol hydrochloride (BI-1744) is the hydrochloride salt form of Olodaterol, which is a long-acting beta2-adrenergic agonist.
  22. GC32543 OPC-28326 OPC-28326是一种外周血管扩张药，同时为α2-adrenergicreceptor的拮抗剂，对α2A-，α2B-和α2C肾上腺素受体的Ki值分别为2040，285和55 nM。
  23. GC10818 Oxprenolol hydrochloride

    盐酸氧烯洛尔,Ba 39089

     A non-selective β-adrenergic receptor antagonist
  24. GC13844 p-iodo-Clonidine (hydrochloride) An α2-adrenergic receptor partial agonist
  25. GC32532 Pamatolol

    氨甲酯心定

     Pamatolol是一种心选择性的beta-adrenoceptor拮抗剂，没有拟交感活性。
  26. GC31069 Pardoprunox (SLV-308)

    SLV-308; DU-126891

     Pardoprunox hydrochloride (DU-126891, SME-308) is a potent but partial dopamine D2 receptor agonist with pEC50 of 8.0, and a partial agonist in the induction of [35S]GTPγS binding with pEC50 of 9.2 and a serotonin 5-HT1A receptor agonist, with pEC50 of 6.3, respectively.
  27. GC30980 Pardoprunox hydrochloride (SLV-308 hydrochloride)

    盐酸帕多芦诺,SLV-308 hydrochloride; DU-126891 hydrochloride

     A dopamine D2 and D3 receptor partial agonist and 5-HT1A agonist
  28. GC31009 Pargolol hydrochloride (Ko 1400 hydrochloride)

    帕高洛尔盐酸盐,Ko 1400 hydrochloride

     Pargolol hydrochloride (Ko 1400 hydrochloride) 是 β；肾上腺素受体拮抗剂。
  29. GC32494 Penbutolol sulfate ((-)-Terbuclomine)

    喷布特罗硫酸盐,(-)-Terbuclomine

     A β-adrenergic and 5-HT1A receptor antagonist
  30. GC12293 Perphenazine

    奋乃静

     A typical antipsychotic
  31. GC36875 Perphenazine D8 Dihydrochloride

    奋乃静 D8 二盐酸盐

     Perphenazine D8二盐酸盐是Perphenazine氘代化合物标准品。
  32. GC12724 Phenoxybenzamine HCl

    盐酸酚苄明

     An α-AR antagonist
  33. GC16291 Phentolamine Mesylate

    甲磺酸酚妥拉明; Phentolamine methanesulfonate

     A reversible α-adrenergic receptor antagonist
  34. GC11272 Phenylephrine HCl

    盐酸去氧肾上腺素; (R)-(-)-Phenylephrine hydrochloride; L-Phenylephrine hydrochloride

     Phenylephrine HCl（盐酸去氧肾上腺素）是一种选择性的α1-肾上腺素能受体激动剂。
  35. GC69700 Phenylephrine-2,4,6-d3 hydrochloride

    (R)-(-)-Phenylephrine-2,4,6-d3 (hydrochloride); L-Phenylephrine-2,4,6-d3 (hydrochloride)

     Phenylephrine-2,4,6-d3 (hydrochloride) 是 Phenylephrine hydrochloride 的氘代物。(R)-(-)-Phenylephrine hydrochloride是一种选择性的α1-肾上腺素能受体激动剂，对α1D，α1B 和α1A 受体的pKis 分为5.86，4.87和4.70。
  36. GC63947 Phenylephrine-d3 hydrochloride

    (R)-(-)-Phenylephrine-d3 hydrochloride; L-Phenylephrine-d3 hydrochloride

     Phenylephrine-d3 (R)-(-)-Phenylephrine-d3) hydrochloride 是 Phenylephrine hydrochloride 的氘代物。(R)-(-)-Phenylephrine hydrochloride是一种选择性的α1-肾上腺素能受体激动剂，对α1D，α1B 和α1A 受体的pKis 分为5.86，4.87和4.70。
  37. GC68407 Phenylethanolamine A-d3 Phenylethanolamine A-D3 是 Phenylethanolamine A 的一种氘代化合物。Phenylethanolamine A 是一种 β-肾上腺素 (β-adrenergic) 激动剂。是 Ractopamine 合成过程中的副产物。
  38. GC10643 Pimozide

    匹莫齐特; R6238

     A dopamine receptor antagonist
  39. GC45756 Pimozide-d4

    R6238-d4

     An internal standard for the quantification of pimozide
  40. GC17734 Pindolol

    吲哚洛尔; LB-46

     A β1- and β2-AR antagonist
  41. GC31782 Piperoxan hydrochloride (Benodaine hydrochloride)

    盐酸哌罗克生; Benodaine hydrochloride

     An α2-adrenergic receptor antagonist
  42. GC36929 Piribedil

    吡贝地尔; 双哌嘧啶

     A dopamine receptor agonist
  43. GC30396 Piribedil D8 (ET-495 D8)

    吡贝地尔D8,ET-495 D8

     Piribedil D8 (ET-495 D8) (ET-495 D8) 是氘标记的 Piribedil，它是一种抗帕金森病药物。
  44. GC61789 Practolol

    普拉洛尔

     Practolol是一种有效和选择性的β1肾上腺素能受体拮抗剂。Practolol可用于心律失常的研究。
  45. GC16785 Prazosin

    哌唑嗪

     哌唑嗪是一种 α-肾上腺素能阻滞剂，是一种用于治疗高血压和焦虑症、创伤后应激障碍和恐慌症的交感神经药物。
  46. GC18072 Prazosin HCl

    哌唑嗪盐酸盐

     An α1-adrenergic receptor antagonist
  47. GC64843 Prenalterol

    普瑞特罗

     Prenalterol 是一种选择性 β1- 肾上腺素能受体激动剂。Prenalterol 对肠道平滑肌收缩活动无影响。Prenalterol 可用于心血管疾病的研究。
  48. GC17085 Procaterol hydrochloride

    盐酸丙卡特罗

     A β2-adrenergic receptor agonist
  49. GC32538 Pronethalol ((±)-Pronethalo)

    丙萘洛尔; (±)-Pronethalo

     Pronethalol ((±)-Pronethalo) ((±)-Pronethalo) 是一种非选择性的 β-肾上腺素能拮抗剂。
  50. GC10536 Pronethalol hydrochloride

    盐酸丙萘洛尔,(±)-Pronethalo hydrochloride

     Pronethalol ((±)-Pronethalo) 是一种非选择性 β-肾上腺素能拮抗剂。
  51. GC25786 Propafenone

    SA-79

     Propafenone (SA-79) is an orally active sodium channel blocking agent and a beta-adrenoceptor (β-adrenergic receptor) antagonist. Propafenone offers a broad spectrum of activity in the treatment of cardiac arrhythmias.

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