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Home >> Signaling Pathways >> GPCR/G protein >> Adrenergic Receptor

Adrenergic Receptor(肾上腺素能受体)

Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.

Products for  Adrenergic Receptor

  1. Cat.No. 产品名称 Information
  2. GC36980 Propranolol

    普萘洛尔

     普萘洛尔(Propranolol)是一种非选择性的 β-adrenergic receptor (βAR) 拮抗剂,对 β1AR 和 β2AR 具有高亲和力,Ki值分别为 1.8 nM和0.8 nM。
  3. GC61208 Propranolol D7 hydrochloride

    盐酸普萘洛尔 d7 (盐酸盐)

     PropranololD7hydrochloride是Propranololhydrochloride的氘代物。Propranololhydrochloride是一种非选择性的β-adrenergicreceptor(βAR)拮抗剂，对β1AR和β2AR具有高亲和力，Ki值分别为1.8nM和0.8nM。Propranololhydrochloride抑制[3H]-DHA与大鼠脑膜制剂的结合，IC50为12nM。Propranololhydrochloride用于高血压，嗜铬细胞瘤，心肌梗塞，心律不齐，心绞痛和肥大心肌病的相关研究。
  4. GC11343 Propranolol HCl

    盐酸普萘洛尔

     A β-adrenergic receptor antagonist
  5. GC32631 QF0301B QF0301B是α1肾上腺素能受体(α1adrenergicreceptor)拮抗剂，也可阻断α2肾上腺素受体，5-HT2A和组胺H1受体。
  6. GC16250 Rauwolscine hydrochloride

    萝芙素盐酸盐; α-Yohimbine hydrochloride; Corynanthidine hydrochloride; Isoyohimbine hydrochloride

     A reversible α2-adrenergic receptor antagonist
  7. GC46212 Rec 15/2615 (hydrochloride)

    SB 216469

     An α1B-AR antagonist
  8. GC17812 Rec 15/2615 dihydrochloride α1B-adrenoceptor antagonist
  9. GC71070 Rezatomidine Rezatomidine（AGN-203818）是一种强效且选择性的α2-AR激动剂。
  10. GC60325 Rilmenidine

    利美尼啶

     An antihypertensive agent
  11. GC15657 Rilmenidine (hemifumarate)

    Oxaminozoline,S 3341

    An antihypertensive agent
  12. GC15063 Ritodrine HCl

    盐酸利托君; DU21220 hydrochloride

     A β2-AR agonist
  13. GC61871 Ro 363 hydrochloride Ro 363 hydrochloride，一种有效的正性肌力活化剂，是一种有效且高度选择性的 β1 肾上腺素受体 (β1-adrenoceptor) 激动剂。Ro 363 hydrochloride 是一种心血管调节剂，可降低舒张压并显着增加心肌收缩力。
  14. GC67683 Romifidine Romifidine 是 α2 肾上腺素受体激动剂。Romifidine 在体内显示出镇定作用。
  15. GC10614 Rotigotine

    罗替戈汀; N-0437; N-0923

     A non-selective dopamine receptor agonist
  16. GC16017 Rotigotine hydrochloride

    罗替戈汀盐酸盐; N-0923 Hydrochloride

     A non-selective dopamine receptor agonist
  17. GC13069 RS 100329 hydrochloride Subtype-selective α1A-adrenoceptor antagonist
  18. GC17070 RS 17053 hydrochloride

    RS-17053

     An α1A-adrenergic receptor antagonist
  19. GC10723 RS 79948 hydrochloride α2-adrenoreceptor antagonist
  20. GC10514 RWJ 52353 An α2D-adrenergic receptor agonist
  21. GC14463 RX 821002 hydrochloride

    RX821002 hydrochloride

     RX 821002 hydrochloride (RX821002 hydrochloride) 是一种高度选择性的 α 2-肾上腺素受体拮抗剂，几乎没有或没有咪唑啉拮抗剂作用。
  22. GC31059 Salbutamol (Albuterol)

    沙丁胺醇半硫酸盐; Albuterol hemisulfate; AH-3365 hemisulfate

     Salbutamol (Albuterol)是一种短效的β2-肾上腺素能受体激动剂（IC50 = 8.93μM），用于治疗哮喘和慢性阻塞性肺病（COPD）。
  23. GC13974 Salbutamol Sulfate

    沙丁胺醇半硫酸盐; Albuterol hemisulfate; AH-3365 hemisulfate

     A β2-AR agonist
  24. GC12188 Salmefamol

    AH 3923;AH-3923; AH3923

    β2-adrenergic receptor agonist
  25. GC30092 Salmeterol (GR33343X)

    沙美特罗; GR33343X

     Salmeterol (Astmerole, GR-33343X, SN408D) is a long-acting beta2-adrenergic receptor agonist with Ki value of 1.5 nM for WT β2AR and shows very high selectivity for the WT β2AR(β1Ki/β2Ki ratio of approximately 1500).
  26. GC11531 Salmeterol xinafoate

    沙美特罗昔萘酸酯; GR 33343X xinafoate

     A long-acting β2-adrenergic receptor agonist
  27. GC48067 Salmeterol-d3

    沙美特罗-D3

     An internal standard for the quantification of salmeterol
  28. GC14220 Scopine

    东莨菪醇,6,7-Epoxytropine

     A metabolite of scopolamine
  29. GC11373 Scopine HCl

    盐酸东莨菪醇,6,7-Epoxytropine hydrochloride

     A metabolite of scopolamine
  30. GC13623 SDZ 21009

    卡品多罗

     β-adrenoceptor and 5-HT1A/1B receptor antagonist
  31. GC13990 Setiptiline

    司普替林; Org-8282

     Setiptiline (Org-8282) 是一种血清素受体拮抗剂。
  32. GC13549 Setiptiline maleate

    马来酸司普替林; MO-8282

     Setiptiline maleate (MO-8282 maleate) 是一种血清素受体拮抗剂。
  33. GC15719 Silodosin

    西洛多辛; KAD 3213; KMD 3213

     A potent α1A-adrenoceptor antagonist
  34. GC12856 SKF 86466 hydrochloride An α2-AR antagonist
  35. GC15426 SNAP 5089 α1A-adrenoceptor antagonist
  36. GC34808 Solabegron

    3'-[[2-[(2R)-2-(3-氯苯基)-2-羟基乙基]氨基]乙基]氨基]-[1,1'-联苯基]-3-羧酸,GW 427353

    Solabegron(GW427353)是β3肾上腺素能受体(β3-AR)的选择性激动剂,在中国仓鼠卵巢细胞中测得的EC50值为22nM。目前正在被用于开发治疗膀胱过度活跃和肠易激综合征。
  37. GC13173 Sotalol

    索他洛尔,(R)-Sotalol

     An Analytical Reference Standard
  38. GC15631 Sotalol hydrochloride

    盐酸索他洛尔; MJ 1999

     A β-AR antagonist and a class III antiarrhythmic agent
  39. GC45893 Sotalol-d6 (hydrochloride)

    索他洛尔-D6,MJ 1999-d6 hydrochloride

     An internal standard for the quantification of sotalol
  40. GC31005 Spirendolol (Li 32-468)

    4'-[3-[(叔丁基)氨基]-2-羟基丙氧基]螺[环己烷-1,2'-[2H]茚]-1'(3'H)-酮,Li 32-468; S 32-468; Substance 32468

     Spirendolol (Li 32-468) is a ⋲肾上腺素受体拮抗剂。
  41. GC13338 Spiroxatrine

    三氮螺癸苯恶烷

     5-HT1A拮抗剂和α2C肾上腺素能受体拮抗剂
  42. GC16091 SR 58611A hydrochloride

    SR 58611A

     A selective β3-AR agonist
  43. GC12227 SR 59230A hydrochloride A β3-AR antagonist
  44. GC39725 SR59230A A β3-AR antagonist
  45. GC11913 ST 91 α2-adrenoceptor agonist
  46. GC38438 Synephrine

    辛弗林; Oxedrine

     Synephrine (Oxedrine), a natural protoalkaloid in the extract of bitter orange and other citrus species, is commonly used for weight loss.
  47. GC12715 Synephrine HCl

    辛弗林盐酸盐; Oxedrine hydrochloride

     An alkaloid
  48. GC39449 Tamsulosin

    坦索罗辛; (R)-(-)-YM12617 free base; LY253351 free base

     A potent α1-AR antagonist
  49. GC50035 Tamsulosin hydrochloride

    盐酸坦索罗辛; (R)-(-)-YM12617; LY253351

     A potent α1-AR antagonist
  50. GC65276 Tasipimidine sulfate Tasipimidine sulfate 是一种具有口服活性的、选择性的 α2A-adrenoceptor 激动剂，对人 α2A-adrenoceptor 的pEC50 为 7.57。Tasipimidine sulfate 可用于情境焦虑和恐惧的研究。
  51. GC16217 TC-G 1000 α2D-adrenoceptor agonist

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