S1P receptor(S1P受体)

S1P (sphinogosine-1-phosphate) receptor is a G-protein coupled receptor that involved in regulation of cells proliferation, survival, motility and adhesion etc.

Products for S1P receptor

Cat.No. 产品名称 Information
GC50275 Ex 26
S1P1-IN-Ex26
Ex 26 (S1P1-IN-Ex 26) 是一种有效的选择性 1-磷酸鞘氨醇受体 1 (S1P1) 拮抗剂 (IC50\u003d0.93 nM)。
GC42664 A-971432 A sphingosine-1-phosphate receptor 5 (S1P₅) agonist
GC16660 Ponesimod
ACT-128800
A potent S1P₁ receptor agonist
GC14360 Ozanimod (RPC1063)
奥扎莫德; RPC-1063
An S1P₁ and S1P₅ agonist
GC16701 SKI II
鞘氨醇激酶抑制剂
An SPHK1 inhibitor
GC17201 BAF312 (Siponimod)
辛波莫德; BAF-312
An S1P₁ and S1P₅ receptor agonist receptor modulator
GC14807 Fingolimod (FTY720) HCl
盐酸芬戈莫德; FTY720
芬戈莫德(FTY720)是一种免疫抑制剂,通常用于治疗多发性硬化症,也有抗癌作用,可以作为HDACi(组蛋白脱乙酰酶抑制剂)。
GC11917 PF-543
(2R)-1-[[4-[[3-甲基-5-[(苯磺酰基)甲基]苯氧基]甲基]苯基]甲基]-2-吡咯烷甲醇,PF543; PF 543
PF-543是一种强效、选择性、可逆和鞘氨醇竞争性SphK 1抑制剂，IC50值为2nM，Ki值为3.6 nM。