Sigma Receptor(Sigma受体)
Sigma receptors are non-opioid receptors that interacted with psychostimulants such as cocaine and methamphetamine. It is associated with central nervous systems diseases, cancer and neuropathic pain etc.
Products for Sigma Receptor
- Cat.No. 产品名称 Information
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GC13357
4-PPBP maleate
4-PPBP maleate 是一种有效的 σ 1 受体配体和激动剂。
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GC14960
PRE-084 hydrochloride
1-苯基环己烷羧酸2-(4-吗啉基)乙基酯盐酸盐
An Analytical Reference Standard
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GC16595
BD 1008 dihydrobromide
An Analytical Reference Standard
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GC16598
DTG
二邻甲苯胍,1,3-Di-o-tolylguanidine; DTG
A σ receptor ligand
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GC13911
S1RA hydrochloride
4-[2-[[5-甲基-1-(2-萘基)-1H-吡唑-3-基]氧基]乙基]吗啉盐酸盐(1:1),E-52862 hydrochloride
A σ1 receptor antagonist
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GC10407
S1RA
E-52862
A σ1 receptor antagonist
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GC13083
Siramesine
Lu 28-179
A selective σ2 receptor agonist
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GC15222
Siramesine hydrochloride
西拉美新盐酸盐; Lu 28-179 hydrochloride
Siramesine (Lu 28-179) hydrochloride 是一种有效的 sigma-2 受体激动剂。 Siramesine hydrochloride 对 sigma-2 受体具有亚纳摩尔亲和力 (IC50=0.12 nM)，对 sigma-2 受体的选择性是 sigma-1 受体的 140 倍 (IC50=17 nM)。盐酸西拉美新通过破坏线粒体而不是溶酶体触发细胞死亡。抗癌活性。