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Home >> Signaling Pathways >> Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel(跨膜转运)

Cat.No. 产品名称 Information
GC16924 Eniporide
N-(二氨基亚甲基)-2-甲基-5-(甲基磺酰基)-4-(1H-吡咯-1-基)苯甲酰胺
A NHE-1 inhibitor
GC13289 Barnidipine (hydrochloride)
盐酸巴尼地平,YM 09730-5
A calcium channel blocker
GC12700 Ivermectin B1a
伊维菌素 B1a
An anthelmintic
GC17065 Estradiol 3-(β-D-Glucuronide) (sodium salt)
E23G,β-Estradiol 3-(β-D-Glucuronide),17β-Estradiol 3-(β-D-Glucuronide),17β-Oestradiol 3-(β-D-Glucuronide)
An isomer of estradiol-(β-D-glucuronide)
GC10391 Hypophyllanthin
(7S,8S,9R)-9-(3,4-二甲氧基苯基)-6,7,8,9-四氢-4-甲氧基-7,8-双(甲氧基甲基)萘并[1,2-D]-1,3-二恶茂,NSC 619044
A P-glycoprotein inhibitor
GC16409 Oligomycin B
寡霉素 B
A nonselective inhibitor of the mitochondrial F₁F_O ATP synthase
GC15824 Ethyl 3-Aminobenzoate (methanesulfonate)
3-氨基苯甲酸乙酯甲基磺酸盐,Ethyl m-Aminobenzoate, NSC 93790, Tricaine methanesulfonate , MS-222
A fish anesthetic
GC12469 2,3-Butanedione-2-monoxime
2,3-丁烷二酮一肟,BDM|Diacetyl Monoxime|NSC 660|NSC 116103
A non-selective myosin ATPase inhibitor
GC15126 Zoniporide (hydrochloride)
CP 597,396
A selective NHE-1 inhibitor
GC10898 5-(N,N-dimethyl)-Amiloride (hydrochloride)
DMA,L-591,605,MK-685
An inhibitor of Na⁺/H⁺ exchangers
GC16823 Enniatin Complex
恩镰孢菌素复合物
A complex mixture of ionophores
GC16221 Oligomycin C
寡霉素C
A mitochondrial F₁F_O ATP synthase inhibitor
GC11124 Lanicemine
拉尼西明; AZD6765
A low-trapping NMDA channel blocker
GC15795 Rhodamine 123 (chloride)
罗丹明123; RH-123; R-22420
Rhodamine 123 (chloride)是一种细胞渗透性阳离子荧光探针，特异性识别线粒体膜电位，最大激发光/发射光为507/529nm。
GC17693 Enniatin B
恩镰孢菌素 B
A natural inhibitor of Pdr5p in yeast
GC11695 Cinnarizine
桂利嗪
A calcium channel inhibitor and histamine H₄ receptor antagonist
GC10497 Hexachlorophene
Nabac, NSC 9887, NSC 49115

KCNQ1/KCNE1 potassium channel activator
GC11143 NS 11394
3'-[5-(1-羟基-1-甲基乙基)-1H-苯并咪唑-1-基]-[1,1'-联苯]-2-甲腈
A subunit-selective positive allosteric modulator of the GABA_A receptor
GC13490 E-4031 An antiarrhythmic, ERG potassium channel blocker
GC13353 Spadin An inhibitor of K_2P2.1/TREK1
GC13930 N-(p-amylcinnamoyl) Anthranilic Acid
2-(3-(4-戊基苯基)丙烯酰胺基)苯甲酸,ACA
A TRP channel blocker and PLA₂ inhibitor
GC10949 Calcium Ionophore I
钙离子载体,ETH 1001
A Ca²⁺-selective ionophore
GC15858 MYK-461
玛伐凯泰,MYK461; SAR439152
A cardiac myosin ATPase inhibitor
GC13781 QX-314 A selective sodium channel blocker
GC14761 Mavatrep
JNJ-39439335
Mavatrep (JNJ-39439335) 是一种具有口服活性、选择性和有效的 TRPV1 拮抗剂，对 hTRPV1 通道具有高亲和力 (Ki=6.5 nM)。
GC10234 GSK1014802(CNV1014802)
GSK-1014802; CNV1014802
GSK1014802(CNV1014802) (GSK-1014802)是一种新型的小分子状态依赖性钠通道阻滞剂； Nav1.7 钠通道抑制剂。
GC17842 CARIPORIDE
卡立泊来德; HOE-642
An NHE-1 inhibitor
GC12413 Rostafuroxin (PST 2238)
PST 2238
An endogenous ouabain blocker at the Na⁺/K⁺ ATPase
GC14029 Retigabine
瑞替加滨
An Analytical Reference Standard
GC14635 RQ-00203078 A TRPM8 antagonist
GC10830 GS967 A selective inhibitor of cardiac late sodium current
GC14705 Tolbutamide Sodium A SUR1/K_ir6.2 channel inhibitor
GC14059 ML 240 A selective inhibitor of the ATPase p97
GC14642 7ACC2 An MCT1 and MPC inhibitor
GC13691 7ACC1
香豆素D1421; DEAC; Coumarin D 1421; D 1421
A fluorescent probe
GC14515 Azimilide
阿齐利特,NE-10064
A class III antiarrhythmic agent
GC16562 PEAQX
NVP-AAM077
PEAQX(NVP-AAM 077) 是一种有效的、具有口服活性的 NMDA 拮抗剂，对人 NMDA 受体的 1A/2A(IC50=270 nM) 比 1A/2B(29,600 nM) 高 15 倍。
GC10906 RBC8 A Ral inhibitor
GC12805 Procainamide HCl
盐酸普鲁卡因胺
An Analytical Reference Standard
GC11025 (+)-MK 801 Maleate
(+)-MK801顺丁烯二酸盐,Dizocilpine Maleate
(+)-MK 801 Maleate是一种强效、选择性和非竞争性的 N-甲基-D-天冬氨酸(NMDA)受体拮抗剂(Ki = 30.5nM)。(+)-MK 801 Maleate已被证明在各种缺血模型中具有保护作用，并能抑制对某些精神兴奋剂的行为敏感化。
GC18027 Huwentoxin XVI Huwentoxin XVI 是一种镇痛剂，是一种来自中国狼蛛 Ornithoctonus huwena 的高度可逆和选择性的哺乳动物 N 型钙通道 (IC50 为 ~60 nM) 拮抗剂。
GC15323 TRAM 39 Potent KCa3.1 blocker
GC11963 Oxiracetam
奥拉西坦,ISF2522
An Analytical Reference Standard
GC10913 GTS 21 dihydrochloride
(3E)-3-[(2,4-二甲氧基苯基)亚甲基]-3,4,5,6-四氢-2,3'-联吡啶二盐酸盐,DMXB-A; DMBX-anabaseine
An agonist of α7-containing nAChRs
GC16315 D-AP5
(R)-(-)-2-氨基-5-膦酰戊酸,D-2-Amino-5-Phosphonovaleric acid; D-APV
D-AP5是一种选择性N-甲基-D-天门冬胺酸（NMDA）受体拮抗剂，K_d 值为1.4μM。
GC11862 LY 233053 Competitive NMDA receptor antagonist
GC12703 Philanthotoxin 74
PhTx 74 dihydrochloride
An AMPA receptor antagonist
GC15678 STO-609 acetate A CaMKK inhibitor
GC13032 (RS)-AMPA hydrobromide
(R,S)-Α-氨基-3-羟基-5-甲基-4-二唑酸氢溴酸
AMPAR agonist
GC14480 CNQX disodium salt
FG9065 disodium
A non-NMDA glutamate receptor antagonist