Membrane Transporter/Ion Channel(跨膜转运)

Cat.No. 产品名称 Information

GC35421 ATP synthase inhibitor 1 ATP synthase inhibitor 1 是一种 F1/FO-ATP 合酶复合物 c 亚基的有效抑制剂，抑制线粒体通透性转换孔的开放，但不影响 ATP 的水平。

GC35407 Asivatrep

PAC-14028

Asivatrep (PAC-14028) 是高效的选择性的瞬时受体电位香草酸亚型1 (TRPV1) 拮抗剂。

GC35325 Amlodipine maleate

马来酸氨氯地平

Amlodipine (Amvaz, UK-48340) maleate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.

GC35322 Amiodarone

胺碘酮

Amiodarone (NSC 85442,Amiodar,Amiodarone hydrochloride,Nexterone) HCl is a sodium/potassium-ATPase inhibitor and an autophagy activator, used to treat various types of cardiac dysrhythmias.

GC35316 AMG2850 AMG2850 是一个有效的、有口服活性的TRPM8 的选择性拮抗剂。

GC35293 Allocryptopine

别隐品碱

An isoquinoline alkaloid with antimicrobial activity

GC35273 Ajmaline

NSC 15627

Ajmaline是一种生物碱, 是一种Ia类的抗心律失常药。

GC35222 ABT-239 ABT-239 是一种新颖的，高效的，非咪唑类的 H3R 拮抗剂，也是 TRPV1 的拮抗剂。

GC35211 A-317491 sodium salt hydrate A P2X₃ and P2X_2/3 receptor antagonist

GC35147 5-(N,N-Hexamethylene)-amiloride

阿米洛利,Hexamethylene amiloride; HMA

An amiloride derivative with diverse biological activities

GC35108 3-Deoxyaconitine

3-脱氧乌头碱

3-Deoxyaconitine is a diterpenoid alkaloid isolated from the root of Aconitum Carmichaeli Debx.

GC35075 20-HETE

20-羟基二十碳-5Z,8Z,11Z,14Z-四烯酸

A cytochrome P450 (CYP450) metabolite of arachidonic acid

GC35010 (Z)-Capsaicin

(Z)-辣椒素; Zucapsaicin; Civamide; cis-Capsaicin

Zucapsaicin, the cis-isomer of capsaicin, is a topical analgesic used to treat osteoarthritis of the knee and other neuropathic pain. It is also a TRPV-1 modulator.

GC34998 (S)-(-)-5-Fluorowillardiine hydrochloride

(5S)-Fluorowillardiine hydrochloride; (S)-5-Fluorowillardiine hydrochloride

(S)-(-)-5-Fluorowillardiine hydrochloride 是AMPAR高效选择性激动剂。

GC34986 (R)-Baclofen hydrochloride

(R)-巴氯芬盐酸盐; Arbaclofen hydrochloride; STX 209 hydrochloride

A GABA_B receptor agonist

GC34959 (+)-Sparteine

(+)-鹰爪豆碱

A quinolizidine alkaloid

GC34954 (+)-Borneol

(+)-冰片

A bicyclic monoterpene with diverse biological activities

GC34952 (-)-Sparteine sulfate pentahydrate

五水合硫酸司巴丁,(+)-Lupinidine sulfate pentahydrate

Sparteine Sulfate, a quinolizidine alkaloid, is the sulfate form of sparteini, which is a sodium channel blocker used as an oxytocic and an anti-arrhythmia agent.