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Calcium Channel(钙离子通道)

Calcium channel is an ion channel that selectively permeable to calcium ions. It serves vital functions in cellular signal transduction.

Products for  Calcium Channel

  1. Cat.No. 产品名称 Information
  2. GC11678 PD 173212

    N-[[4-叔丁基苯基]甲基]-N-甲基-L-亮氨酰-N-叔丁基-O-苄基-L-酪氨酰胺

    An N-type calcium channel blocker
  3. GC12608 ω-Agatoxin TK ω-Agatoxin TK 是 Agelenopsis aperta 毒液的肽基毒素,是一种有效的选择性 P/Q 型 Ca2+ 通道阻滞剂。
  4. GC15513 ω-Agatoxin IVA

    OMEGA-漏斗网蛛毒素IVA

    A P-type calcium channel blocker
  5. GC14326 Calmidazolium chloride

    钙调蛋白抑制剂,R 24571

    An inhibitor of calmodulin
  6. GC16911 CGS 9343B

    CGS-9343B; KW 5617

    A calmodulin inhibitor
  7. GC15446 Ionomycin free acid

    离子霉素,SQ23377

    Ionomycin free acid 是一种选择性的强效钙离子载体,可作为活性 Ca2+ 载体。
  8. GC11082 Paxilline

    蕈青霉素

    Paxilline是一种致震颤真菌生物碱,可有效抑制高电导Ca2+ 激活K+ (BK)通道,IC50约为10nM,Ki=1.9nM。
  9. GC10351 SR 33805 oxalate Ca2+ channel antagonist
  10. GC15099 Autocamtide-2-related inhibitory peptide A CaMKII inhibitor
  11. GC16766 Ruthenium Red

    钌红; Ammoniated ruthenium oxychloride

    A polycationic dye that blocks Ca2+ release
  12. GC14484 (-)-Xestospongin C

    XeC, Araguspongine E

    A membrane-permeable antagonist of the inositol-1,4,5-triphosphate receptor
  13. GC11200 A23187

    离子载体(钙镁盐混合物),Calcimycin

    A23187自由酸是一种Ca2+离子载体。

  14. GC11482 Thapsigargin

    毒胡萝卜素

    他普西加林是一种肌浆网/内质网Ca2+ ATP酶泵的抑制剂。
  15. GC10786 DHBP dibromide

    二溴化-1,1ˊ-二庚基-4,4ˊ-联吡啶鎓,Diheptylviologen dibromide

    DHBP 二溴化物是一种钙释放抑制剂和一种肌肉松弛剂。
  16. GC15868 Dantrolene, sodium salt

    丹曲林钠,F 440

    An inhibitor of calcium release
  17. GC11178 A-7 hydrochloride A cell-permeable antagonist of calmodulin
  18. GC17496 W-7 hydrochloride

    N-(6-氨基己基)-5-氯-1-萘磺胺盐酸盐

    A cell-permeable antagonist of calmodulin
  19. GC16962 W-5 hydrochloride

    W-5盐酸盐

    A low-affinity calmodulin antagonist
  20. GC13869 Fasudil

    法舒地尔; HA-1077; AT877

    Fasudil(法舒地尔;HA-1077;AT877)是一种非特异性RhoA/ROCK抑制剂,对ROCK1的Ki为0.33μM,IC50为0.158μM,对ROCK2和PKA、PKC、PKG的IC50分别为4.58μM、12.30μM、1.650μM。
  21. GC17625 Lercanidipine

    乐卡地平

    乐卡地平是一种亲脂性第三代二氢吡啶-钙通道阻滞剂(DHP-CCB)。
  22. GC10590 Lercanidipine hydrochloride

    盐酸乐卡地平

    An L-type calcium channel blocker
  23. GC14142 Acetylcholine Chloride

    氯化乙酰胆碱; ACh chloride

    A neurotransmitter
  24. GC17587 Manidipine

    马尼地平

    An L- and T-type calcium channel blocker
  25. GC13888 Benidipine HCl

    盐酸贝尼地平,KW-3049

    An L-, T-, and N-type calcium channel blocker
  26. GC15550 Lacidipine

    拉西地平

    An L-type calcium channel blocker
  27. GC16532 Flunarizine 2HCl

    盐酸氟桂利嗪

    A calcium antagonist
  28. GC13352 Neomycin sulfate

    硫酸新霉素

    An antibiotic used in tissue culture studies

  29. GC13146 Amlodipine Besylate

    苯磺酸氨氯地平; Amlodipine benzenesulfonate

    An L-type calcium channel blocker
  30. GC13523 Amlodipine

    氨氯地平

    An L-type calcium channel blocker
  31. GC16999 Nitrendipine

    尼群地平; BAY-E-5009

    An L-type calcium channel blocker
  32. GC15024 Nifedipine

    硝苯地平; BAY-a-1040

    An L-type calcium channel blocker
  33. GC12911 Tetracaine HCl

    盐酸丁卡因,Amethocaine hydrochloride

    An Analytical Reference Standard
  34. GC13466 Flufenamic acid

    氟芬那酸

    An NSAID and COX inhibitor
  35. GC15860 Ibutilide Fumarate

    富马酸伊布利特; U70226E

    A class III antiarrhythmic drug
  36. GC10458 Penfluridol

    五氟利多; R-16341

    A typical antipsychotic
  37. GC10678 Nicardipine HCl

    盐酸尼卡地平; YC-93

    An L-type calcium channel blocker
  38. GC13997 Lomerizine HCl

    盐酸洛美利嗪; KB-2796

    A voltage-dependent calcium channel blocker
  39. GC17173 Felodipine

    非洛地平

    An L-type calcium channel inhibitor
  40. GC17952 Zonisamide sodium

    唑尼沙胺钠; AD 810 sodium; CI 912 sodium

    A broad-spectrum sulfonamide antiepileptic agent
  41. GC15101 Azelnidipine

    阿折地平; CS 905

    A calcium channel blocker
  42. GC17106 Verapamil HCl

    盐酸维拉帕米; (±)-Verapamil hydrochloride; CP-16533-1 hydrochloride

    Verapamil是 L 型钙通道阻滞剂和肾上腺素能受体拮抗剂,常用于高血压、心律失常和心绞痛的研究。
  43. GC17316 Gabapentin HCl

    加巴喷丁盐酸盐

    An approved antiepileptic drug
  44. GC16128 Clevidipine Butyrate

    氯维地平

    An inhibitor of L-type calcium channels
  45. GC15293 Manidipine 2HCl

    盐酸马尼地平,CV-4093

    An L- and T-type calcium channel blocker
  46. GC16889 Nisoldipine

    尼索地平; BAY-k 5552

    A calcium channel inhibitor
  47. GC11070 Dehydroepiandrosterone (DHEA)

    脱氢表雄酮; Prasterone; Dehydroisoandrosterone; Dehydroepiandrosterone

    脱氢表雄酮 (DHEA) 及其硫酸酯 DHEAS 共同代表了人体内最丰富的类固醇激素。
  48. GC17690 Cromolyn sodium

    色甘酸钠; Disodium Cromoglycate; FPL-670

    A mast cell stabilizer
  49. GC11819 Strontium Ranelate

    雷尼酸锶; Distrontium renelate; S12911

    An antiosteoporotic agent
  50. GC14487 Ranolazine

    雷诺嗪; CVT 303; RS 43285-003

    Ranolazine (CVT 303) 是一种抗心绞痛药物,通过抑制内向钠电流(INa 和 IKr,IC50 值分别为 6 μM 和 12 μM)的晚期而不影响心率或血压 (BP) 来实现其效果。
  51. GC16587 Nimodipine

    尼莫地平; BAY-e 9736

    An L-type calcium channel inhibitor

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