GABA Receptor(γ-氨基丁酸受体)
GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.
Products for GABA Receptor
- Cat.No. 产品名称 Information
-
GC10262
Tracazolate hydrochloride
ICI 136753 hydrochloride
Tracazolate (ICI 136753) hydrochloride 是一种有效的 GABAA 受体调节剂。 -
GC13374
CGP 13501
Positive modulator of GABAB receptors,allosteric
-
GC15563
CGP 7930
A positive allosteric modulator of GABAB receptors
-
GC16356
SB 205384
positive GABAA receptor modulator
-
GC17350
L-655,708
A ligand for α5 subunit-containing GABAA receptors with nootropic activity
-
GC14477
CI 966 hydrochloride
GABA transporter GAT-1 inhibitor
-
GC14045
Loreclezole
氯瑞唑,R 72063
Loreclezole是一种镇静剂和抗惊厥药,可作为 GABAA 受体正变构调节剂,选择性刺激含有β2或β3亚基的受体。 -
GC10101
SR 95531 hydrobromide
克他命,Gabazine
SR 95531 氢溴酸盐 (Gabazine) 是 GABAA 受体上 GABA 结合位点的选择性拮抗剂 。 -
GC13131
CGP 46381
GABAB受体拮抗剂
-
GC16947
CGP 52432
4-苄氧基苯基异硫氰酸酯
A GABAB receptor antagonist -
GC11153
CGP 35348
(3-氨丙基)(二乙氧基甲基)膦酸水合物
A brain-accessible GABAB receptor antagonist -
GC10489
CGP 54626 hydrochloride
TOCCGP54626盐酸盐
A selective GABAB receptor antagonist -
GC15226
SKF 89976A hydrochloride
1-(4,4-二苯基-3-丁烯基)-3-哌啶盐酸盐,d,l-SKF89976A hydrochloride
SKF 87699A hydrochloride 是一种选择性 GABA 转运蛋白 (GAT-1) 抑制剂,对 CHO 细胞中的 GAT-1、GAT-2 和 GAT-3 的 IC50 分别为 0.28 μM、137.34 μM 和 202.8 μM。 -
GC10183
TPMPA
A selective GABAA-ρ1 (ρ1 GABAC) receptor antagonist
-
GC16311
Chlormethiazole hydrochloride
氯美噻唑盐酸盐,Clomethiazole hydrochloride
A potentiator of GABAA receptors -
GC12169
NCS-382
A GHB receptor antagonist
-
GC16495
GBLD 345
GABAA receptor agonist
-
GC16569
PK 11195
1-(2-氯苯基)-N-甲基-N-(1-甲基丙基)-3-异喹啉甲酰胺,RP 52028
A high affinity ligand for peripheral benzodiazepine receptor, TSPO
-
GC16238
FGIN-1-43
ligand as probe for the mitochondial DBI receptor (peripheral benzodiazepine receptor)
-
GC14017
FGIN-1-27
N,N-二己基-2-(4-氟苯)吲哚-3-乙酰胺
A TSPO agonist -
GC17381
trans-4-Hydroxycrotonic acid
4-羟基巴豆酸
ligand of γ-hydroxybutyric acid (GHB) receptor -
GC11449
β-CCB
N-丁基-Β-咔啉-3-羧酸酯
benzodiazepine receptor ligand
-
GC12506
3-Methyl-GABA
3-Methyl-GABA 是一种有效的 GABA 氨基转移酶激活剂。
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GC14942
SKF 97541
GABAB激动剂
-
GC17257
Saclofen
3-氨基-2-(4-氯苯基-丙烷磺酸
A GABAB receptor antagonist -
GC11267
2-Hydroxysaclofen
3-氨基-2-4-氯苯基-2-羟基丙烷磺酸
2-Hydroxysaclofen 是一种有效的 γ-amino-butyric-acid-B (GABAB) 受体拮抗剂。 -
GC10967
TACA
7-氨基-3-[(1H-1,2,3-三唑-4-硫代)甲基]-8-氧代-5-硫杂-1-氮杂双环[4.2.0]辛-2-烯-2-甲酸,trans-4-Aminocrotonic acid
An agonist of homomeric GABAA receptors -
GC10313
ZAPA sulfate
GABAA receptors agonist
-
GC17691
Phaclofen
3-氨基-2-(4-氯苯基)丙基膦酸
Phaclofen 是一种选择性 GABAB 受体拮抗剂。 -
GC15636
(-)-Bicuculline methochloride
(-)-荷包牡丹碱甲氯化物,l-Bicuculline methochloride
An enantiomer of (+)-bicuculline methochloride -
GC16857
(-)-Bicuculline methobromide
(-)-荷包牡丹碱甲溴化物,l-Bicuculline methobromide
(-)-Bicuculline methobromide (l-Bicuculline methobromide) 是一种有效的 GABAA 受体拮抗剂。 -
GC11612
RuBi GABA trimethylphosphine
GABAB receptor agonist
-
GC17321
RuBi-GABA
RuBi-GABA 是一种新型的钌基笼状 GABA 化合物。
-
GC14150
DPNI-caged-GABA
activates GABAA receptor
-
GC14192
Allopregnanolone
四氢孕酮
Allopregnanolone 是一种 3alpha、5alpha 孕酮代谢物,可作为 γ-氨基丁酸 A 型 (GABAA) 受体的有效变构调节剂,发挥抗抑郁和神经保护作用 。 -
GC17399
Pregnanolone
孕烷醇酮
GABAA receptor positive allosteric modulator
-
GC11565
Bretazenil
溴他西尼,Ro 16-6028
A positive allosteric modulator of GABAA receptors -
GC11600
Valerenic acid
缬草素,(-)-Valerenic Acid
Valerenic acid ((-)-Valerenic Acid) 是一种倍半萜类化合物,是一种具有口服活性的 GABAA 受体正变构调节剂。 -
GC12357
Pentylenetetrazole
戊四唑
A seizure-inducing compound -
GC12359
Hispidulin
高车前素; Dinatin
A flavonoid with diverse biological activities -
GC10844
SCS
亚水杨基水杨基肼
GABAA receptor antagonist -
GC10856
THIP hydrochloride
GAB氧杂DOL盐酸盐
A GABAA receptor agonist and GABAC receptor antagonist -
GC12568
FG 7142
ZK 39106; LSU-65
A benzodiazepine receptor ligand -
GC10530
Dihydroergotoxine mesylate
甲磺酸二氢麦角碱; Ergoloid mesylates
A mixture of alkaloids with diverse biological activities -
GC14834
(±)-Nipecotic acid
3-哌啶甲酸; (±)-β-Homoproline; Hexahydronicotinic acid; 3-Carboxypiperidine
A GAT inhibitor -
GC13567
Isoguvacine hydrochloride
异四氢烟酸
A GABAA receptor agonist -
GC14659
Guvacine hydrochloride
去甲槟榔次碱
An inhibitor of GABA uptake -
GC10186
Tiagabine
噻加宾
A GAT-1 inhibitor -
GC17402
Tiagabine hydrochloride
盐酸噻加宾; NO050328 hydrochloride; NO328 hydrochloride; TGB hydrochloride
A GAT-1 inhibitor -
GC13387
Vigabatrin Hydrochloride
盐酸氨己烯酸; γ-Vinyl-GABA hydrochloride
Inhibitor of GABA transaminase