GABA Receptor(γ-氨基丁酸受体)

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.

Products for GABA Receptor

Cat.No. 产品名称 Information
GC16564 Niflumic acid
氟尼酸
A selective COX-2 inhibitor
GC15960 Primidone
去氧苯比妥
An Analytical Reference Material
GC16691 Chlormezanone
氯美扎酮
A muscle relaxant
GC11901 Nefiracetam
奈非西坦; DM9384; DZL-221
An Analytical Reference Standard
GC12414 Bemegride
贝美格; 3-Ethyl-3-methylglutarimide; Bemegrid
Bemegride (3-Ethyl-3-methylglutarimide) 是一种中枢神经系统兴奋剂和巴比妥类中毒的解毒剂。
GC13792 Rufinamide
卢非酰胺; CGP 33101; E 2080; RUF 331
An anticonvulsant
GC14111 (R)-baclofen
(R)-巴氯芬; Arbaclofen; STX209
(R)-巴氯芬 (Arbaclofen) 是一种选择性 GABAB 受体激动剂。
GC10974 AWD 131-138
伊匹妥英,AWD 131-138
A partial agonist of the GABA_A receptor
GC13802 Riluzole
利鲁唑; PK 26124
Riluzole 是一种抗惊厥药，属于使用依赖性 Na+ 通道阻滞剂家族，它也可以抑制 GABA 摄取，IC50 为 43 μM。
GC12714 Gabapentin
加巴喷丁
An approved antiepileptic drug
GC10772 Flumazenil
氟马西尼; Ro 15-1788
A GABA_A receptor antagonist and partial agonist
GC12599 Retigabine dihydrochloride
瑞替加滨,D 20443 dihydrochloride;D-20443 dihydrochloride;D20443 dihydrochloride
An Analytical Reference Standard
GC15264 Etifoxine hydrochloride
盐酸艾替伏辛,Stresam;HOE 36-801
A positive allosteric modulator of GABA_A receptors
GC14916 Acamprosate calcium
阿坎酸钙,Calcium N-acetylhomotaurinate; Campral EC
An NMDA modulator
GC16149 Topiramate
托吡酯; McN 4853; RWJ 17021
An anticonvulsant
GN10254 Ginsenoside Rc
人参皂苷 Rc; Panaxoside Rc
A saponin with diverse biological activities
GN10251 Ginkgolide A
银杏内酯A; BN-52020
A terpenoid lactone with diverse biological activities
GN10086 Jujuboside A
酸枣仁皂苷 A
Jujuboside A 是一种从刺子中提取的糖苷，刺子是一种用于治疗失眠和焦虑的中草药。
GN10745 (+)-Bicuculline
(+)-荷包牡丹碱,Bucuculline
(+)-荷包牡丹碱((+)-Bicuculline ))是一种竞争性GABA_A受体拮抗剂，IC₅₀为2μM。
GA10664 H-Dab•HBr
L-2,4-二氨基丁酸氢溴酸盐,L-2,4-Diaminobutyric acid
H-Dab•HBr (L-2,4-Diaminobutyric acid) 是一周 GABA 转氨酶抑制剂，IC50 大于 500 μM;在体内和体外均表现出抗肿瘤活性。
GA10004 H-D-Met-OH
D-蛋氨酸,MRX-1024; D-Methionine
H-D-Met-OH (MRX-1024; D-H-D-Met-OH) 是一种有效的化学保护剂，还可以通过 GABAA 受体激活抑制神经元活性。