NMDA Receptor(NMDA受体)

NMDA (N-methyl-D-aspartate) receptor is a glutamate-gated cation channels that plays a vital role in regulating synaptic transmission, neuroplasticity and central nervous system development. It is involved in a range of physiological processes such as learning, memory and pain etc.

Products for NMDA Receptor

Cat.No. 产品名称 Information
GC11335 DL-AP7
2-APH; 2-Amino-7-phosphonoheptanoic acid
DL-AP7 是一种竞争性 NMDA 拮抗剂和抗惊厥药。
GC13714 Conantokin G Conantokin G 是一种 17 个氨基酸的肽，是一种有效的、选择性的和竞争性的 N-甲基-D-天冬氨酸 (NMDA) 受体拮抗剂。
GC11585 TCN 237 dihydrochloride TCN 237 dihydrochloride 是一种有效的 NR2B 选择性 NMDA 拮抗剂，Ki 为 0.85 nM； NR2B Ca2+ 内流 IC50 为 9.7 nM；对 NR2A、NR2C、NR2D、hERG 通道和 α1-肾上腺素能受体无活性。
GC14121 GLYX 13
雷帕替奈; GLYX-13
A partial agonist of the NMDA receptor
GC12785 ZD 9379 ZD 9379 是一种有效的、具有口服活性的脑渗透性完全拮抗剂，作用于 NMDA 受体的甘氨酸位点。
GC12944 Conantokin-R non-competitive NMDA receptor antagonist
GC15156 Conantokin-T Non-competitive NMDA receptor antagonist
GC16240 MNI-caged-NMDA
NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group
GC10043 D-CPP-ene NMDA antagonist
GC10866 Spermidine trihydrochloride
三盐酸亚精胺
An endogenous polyamine
GC11064 Spermine tetrahydrochloride
精胺四盐酸盐
A natural polyamine
GC16915 (2R,3S)-Chlorpheg NMDA receptor antagonist
GC14470 Arcaine sulfate
硫酸魁蛤素
An NMDA receptor antagonist
GC17652 N-(4-Hydroxyphenylacetyl)spermine NMDA receptor antagonist
GC11715 Ibotenic acid
鹅膏氨酸,(RS)-Ibotenic acid; DL-Ibotenic acid
An excitotoxic NMDA and metabotropic glutamate receptor agonist
GC11286 ACBC
1-氨基环丁烷羧酸
ACBC 是一种 NMDA 受体部分激动剂，作用于甘氨酸位点 NR1。
GC14547 Quinolinic acid
喹啉酸
An excitotoxic agonist at NMDA receptors
GC17823 L-Cysteinesulfinic acid
L-半胱氨酸亚磺酸
L-半胱氨酸亚磺酸是几种大鼠代谢型谷氨酸受体 (mGluR) 的有效激动剂，对 mGluR1、mGluR5、mGluR2、mGluR4、mGluR6 和 mGluR8 的 pEC50 分别为 3.92、4.6、3.9、2.7、4.0 和 3.94 .
GC15363 Felbamate hydrate
W-554 hydrate; ADD-03055 hydrate
An inhibitor of NMDA receptors and a modulator of GABA_A receptors
GC10522 Felbamate
非尔氨酯; W-554; ADD-03055
An inhibitor of NMDA receptors and a modulator of GABA_A receptors
GC11470 Flupirtine maleate
氟吡啶马来酸
An activator of Kv7 channels
GC14039 MDL-29951
An NMDA receptor antagonist and GPR17 agonist
GC15270 (-)-MK 801
(-)-Dizocilpine Maleate
An NMDA receptor antagonist
GC16986 SDZ 220-581 hydrochloride
(S)-ALPHA-氨基-2'-氯-5-(膦酰甲基)-[1,1'-联苯]-3-丙酸盐酸盐
SDZ 220-581 hydrochloride 是一种口服有效的竞争性 NMDA 受体拮抗剂，pKi 值为 7.7。
GC18118 SDZ 220-581
(S)-ALPHA-氨基-2'-氯-5-(膦酰基甲基)-[1,1'-联苯]-3-丙酸,SDZ 220 581
SDZ 220-581 是一种具有口服活性、强效、竞争性 NMDA 受体拮抗剂，pKi 值为 7.7。
GC16616 (+)-MK 801
Dizocilpine maleate;Dizocilpine hydrogen maleate;(+)-MK 801;MK 801
强效 NMDA 拮抗剂