JavaScript seems to be disabled in your browser. For the best experience on our site, be sure to turn on Javascript in your browser.

Home >> Signaling Pathways >> MAPK Signaling

MAPK Signaling(MAPK信号通路)

Products for MAPK Signaling

Cat.No. 产品名称 Information
GC30609 p38 MAPK-IN-2 p38MAPK-IN-2是一种p38kinase的抑制剂。
GC30545 Malantide Malantide是一种十二肽，能够被PKA磷酸化，并且能够增强PKA的活性。
GC30162 trans-Zeatin
反-玉米素

A cytokinin plant growth regulator
GC30158 p38-α MAPK-IN-1
p38-α MAPK-IN-1 is an inhibitor of p38-α, with IC50 value of 2300 nM in EFC displacement assay, and 5500 nM in HTRF assay.
GC30057 D-JNKI-1 (AM-111)
AM-111; XG-102
D-JNKI-1 (AM-111) (AM-111) 是一种高效且可渗透细胞的 JNK 肽抑制剂。
GC19479 AZ304 AZ304 是一种 ATP 竞争性双 BRAF 激酶抑制剂，有效抑制野生型 BRAF、V600E 突变型 BRAF 和野生型 CRAF，IC50 分别为 79 nM、38 nM 和 68 nM。 AZ304 对其他激酶也有显着影响，例如 p38 (IC50, 6 nM)、CSF1R (IC50, 35 nM)。抗肿瘤活性。
GC18156 MK8353
SCH900353
MK8353 (SCH900353) 是一种有效的、选择性的、可口服的 ERK1/2 抑制剂，IC50 分别为 23.0 nM 和 8.8 nM； MK8353 具有抗肿瘤活性。
GC19396 H 89
N-[2-[P-溴苯丙烯盐基氨基]乙基]-5-异喹啉磺酰胺

A PKA inhibitor
GC19366 UM-164
DAS-DFGO-II
An inhibitor of Src and p38 MAPK kinases
GC19325 SD 0006
3-[N-(2-羟基乙酰基)-4-哌啶基]-4-(4-嘧啶基)-5-(4-氯苯基)吡唑,SD-06
An inhibitor of p38α MAPK
GC19307 RAF709 A potent inhibitor of B-RAF and C-RAF
GC19304 R1487 Hydrochloride An inhibitor of p38α MAPK
GC19260 NCB-0846
顺式-4-((2-((1H-苯并[D]咪唑-6-基)氨基)喹唑啉-8-基)氧基)环己醇
A TNIK inhibitor
GC19235 LY3214996
LY3214996
An ERK1/2 inhibitor
GC19228 LXH254 A pan-RAF inhibitor
GC19173 GNE-3511 A selective and highly potent inhibitor of DLK
GC19131 Tomivosertib
6'-[(6-氨基-4-嘧啶基)氨基]-8'-甲基螺[环己烷-1,3'(2'H)-咪唑并[1,5-A]吡啶]-1',5'-二酮,eFT508
A potent inhibitor of MNK1 and MNK2
GC19091 CCT196969 A multi-kinase inhibitor
GC19090 CCG215022 A GRK inhibitor
GC19066 BGB-283 BGB-283 is a novel and potent Raf Kinase and EGFR inhibitor with IC50 values of 23 and 29 nM for recombinant BRafV600E and EGFR, respectively.
GC19048 AZD-0364
AZD0364
An inhibitor of ERK1/2
GC19041 ASK1-IN-1 ASK1-IN-1 是一种有效的、口服的、选择性的 ATP 竞争性凋亡信号调节激酶 1 (ASK1) 抑制剂，IC50 为 2.87 nM。
GC19019 Acumapimod
BCT197
An inhibitor of p38α MAPK
GC18951 Obscurolide A1 A phosphodiesterase inhibitor
GC18751 Reticulol
网状菌醇
A cAMP phosphodiesterase and DNA topoisomerase I inhibitor
GC18666 Debromohymenialdisine
DBH, SKF 108753
An inhibitor of Chk1 and Chk2
GC18602 p38 MAPK Inhibitor IV
2,2'-磺酰基双(3,4,6-三氯苯酚),p38 MAP Kinase Inhibitor IV
An inhibitor of p38 MAP kinases
GC18532 Skyrin
穗花衫双黄酮,Endothianin，Rhodophyscin
A fungal metabolite that blocks glucagon signaling
GC18273 SB 202190 (hydrochloride) A potent and selective p38 MAP kinase inhibitor
GC18257 GNE-495 An orally bioavailable, potent, and selective MAP4K4 inhibitor
GC18241 Lysophosphatidylcholines
L-溶血卵磷脂,Lyso-Lecithins (egg)
A glycerophospholipid
GC18178 BI-882370 A RAF inhibitor
GC14982 SD 169
1H-吲哚-5-甲酰胺,5-Carbamoylindole
A selective inhibitor of p38α and p38β MAP kinase
GC15352 8-CPT-Cyclic AMP (sodium salt)
8-(4-硫代氯苯基)腺苷-3',5'-环状磷酸钠,8-(p-Chlorophenylthio)-cAMP,8-CPT-cAMP
A cell-permeable cAMP analog
GC13142 RWJ 67657
4-(4-氟苯基)-2-(4-羟基-1-丁炔)-1-(3-苯基丙基)-5-(4-吡啶基)咪唑,JNJ-3026582
An orally active inhibitor of p38α and p38β
GC16723 MK2 Inhibitor IV
MK 25
A highly selective MAPKAPK2 (MK2) inhibitor
GC10593 BMS-582949 hydrochloride A p38α MAP kinase inhibitor
GC16678 UCN-02
7-epi-hydroxy Staurosporine
A PKC inhibitor
GC16019 SB 202474 A negative control for SB 202190 and SB 203580
GC11157 LL-Z 1640-4
Antibiotic LLZ1640-4,(5Z)-Zeaenol,Curvularia Sp.
A negative control for MAPK signaling
GC12799 H-8 (hydrochloride)
H-8二氢氯化物,Protein Kinase Inhibitor H-8
A potent, nonspecific kinase inhibitor
GC13640 Kemptide
肯普肽
A PKA substrate
GC15646 PD 184161 A potent MEK1/2 inhibitor
GC17265 AG-126
酪氨酸磷酸化抑制剂126,Tyrphostin AG-126
Tyrosine kinase inhibitor that blocks ERK1/2 phosphorylation
GC10428 Sp-5,6-dichloro-cBIMPS (sodium salt)
Sp-5,6-DCI-cBIMPS
A selective PKA activator
GC11422 Ulixertinib (hydrochloride)
BVD-523盐酸盐,BVD-523,VRT-752271
An ERK1/2 inhibitor
GC11307 ML-264
(2E)-3-(3-氯苯基)-N-[2-[甲基(四氢-1,1-二氧代-2H-噻喃-4-基)氨基]-2-氧代乙基]-2-丙烯酰胺
A selective KLF5 inhibitor
GC17693 Enniatin B
恩镰孢菌素 B
A natural inhibitor of Pdr5p in yeast
GC15240 APS-2-79 An inhibitor of KSR-dependent MAPK signaling
GC12124 Selonsertib (GS-4997)
GS-4997
An ASK1 inhibitor