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Home >> Signaling Pathways >> Metabolism

Metabolism(代谢)

  1. Cat.No. 产品名称 Information
  2. GC61748 Betrixaban D6

    贝曲西班 d6

     BetrixabanD6是Betrixaban的氘代化合物。Betrixaban是一种口服有效的选择性factorXa(fXa)抑制剂。
  3. GC61747 Sp-cAMPS Sp-cAMPS，一种cAMP类似物，是一种依赖cAMP的PKAI和PKAII的有效激活剂。Sp-cAMPS还是一种有效的竞争性磷酸二酯酶(PDE3A)抑制剂，Ki为47.6µM。Sp-cAMPS以EC50为40μM来结合PDE10GAF域。
  4. GC61722 2,6-Dimethylquinoline

    2,6-二甲基喹啉

     2,6-Dimethylquinoline是一种来自Peucedantupraeruptorum根的天然成分，是CYP1A2的抑制剂，IC50为3.3µM。2,6-Dimethylquinoline也抑制CYP2B6的活性，IC50为480µM。
  5. GC61689 Alminoprofen

    阿明洛芬,EB-382

     Alminoprofen是苯丙酸类非甾体抗炎药(NSAID)。Alminoprofen同时具有抑制分泌磷脂酶A2(sPLA2)活性和抗环氧化酶(COX-2)的活性。
  6. GC61582 3-Phenyltoxoflavin 3-Phenyltoxoflavin是Toxoflavin的衍生物，是一种Hsp90抑制剂，抑制Hsp90-TPR2A之间相互作用的Kd值为585nM。3-Phenyltoxoflavin具有抗癌活性。
  7. GC61574 AS1810722 AS1810722是口服有效的STAT6抑制剂，IC50为1.9nM。AS1810722显示出良好的CYP3A4抑制作用。AS1810722是一种稠合双环嘧啶衍生物，具有用于过敏性疾病，例如哮喘和特应性疾病研究的潜力。
  8. GC61563 Aminohexylgeldanamycin

    AHGDM

     Aminohexylgeldanamycin(AHGDM)，Geldanamycin的衍生物，是一种热休克蛋白90(HSP90)抑制剂。Aminohexylgeldanamycin具有抗血管生成和抗肿瘤活性。
  9. GC61548 (Rac)-5-Keto Fluvastatin

    氟伐他汀EP杂质D,3-Hydroxy-5-Keto Fluvastatin

     (Rac)-5-KetoFluvastatin(3-Hydroxy-5-KetoFluvastatin)是Fluvastatin(XU62320)的杂质。Fluvastatin是HMG-CoA还原酶的抑制剂，IC50值为8nM。
  10. GC61508 CALP2 TFA CALP2TFA是一种钙调蛋白(CaM)拮抗剂(Kd为7.9µM)，以亲和力结合CaMEF-hand/Ca2+结合位点。CALP2TFA抑制CaM依赖性磷酸二酯酶(phosphodiesterase)活性并增加细胞内Ca2+浓度。CALP2TFA有效抑制粘附和脱粒。CALP2TFA还是肺泡巨噬细胞的强激活剂。
  11. GC61465 SDZ285428 SDZ285428是一种CYP51抑制剂。SDZ285428抑制Trypanosomacruzi(TC)CYP51，I/E2<1(5min)及I/E2=9(1h)。SDZ285428抑制Trypanosomabrucei(TB)CYP51，I/E2<1(5min)及I/E2=35(1h)。
  12. GC61436 Gallic acid hydrate

    没食子酸-水合物; 3,4,5-Trihydroxybenzoic acid hydrate

     A phenol with diverse biological activities
  13. GC19706 Propacetamol hydrochloride

    盐酸丙帕他莫

     A prodrug form of acetaminophen
  14. GC19691 Pyrene

    芘

     A polycyclic aromatic hydrocarbon
  15. GC19686 DL-Pyroglutamic acid

    DL-焦谷氨酸

      
  16. GC18252 Diallyl Sulfide

    二烯丙基硫醚

     An organosulfur compound
  17. GC19528 1,4-Benzoquinone

    对苯醌

     A toxic metabolite of benzene
  18. GC48954 CP21 An iron chelator
  19. GC48943 2-deoxy-2-fluoro-D-Glucose

    2-脱氧-2-氟-D-葡萄糖

     A glucose derivative with anticancer activity
  20. GC48932 Callosobruchusic Acid

    R-(–)-Callosobruchusic Acid

     An insect pheromone
  21. GC48895 Rufinamide-15N-d2

    [15N,2H2]-卢非酰胺

     An internal standard for the quantification of rufinamide
  22. GC48889 Methazolamide-d6

    L584601-d6

     An internal standard for the quantification of methazolamide
  23. GC48884 WF-3681

    抗生素WF-3681

     A fungal metabolite
  24. GC48872 Pyridindolol

    NSC 266530

     A bacterial metabolite
  25. GC48870 Anagrelide-13C3

    BL 4162A-13C3, BMY 26538-01-13C3

     An internal standard for the quantification of anagrelide
  26. GC48856 Fenspiride-d5

    Decaspiride-d5

     An internal standard for the quantification of fenspiride
  27. GC48843 5α-Androst-16-en-3α-ol

    (3α,5α)-16-烯-3-甾醇

     A pheromone with diverse biological activities
  28. GC48819 17-Epiestriol

    17-环雌三醇

     A metabolite of estrone
  29. GC48804 N-desmethyl Olanzapine

    N-去甲基奥氮平

     A major metabolite of olanzapine
  30. GC48803 Norethynodrel

    异炔诺酮,Enidrel; SC 4642; NSC 15432

     A synthetic progestin
  31. GC48788 Norethindrone-d6

    炔诺酮D6,Norethisterone-d6

     An internal standard for the quantification of norethindrone
  32. GC48782 10,13-epoxy-11-methyl-Octadecadienoic Acid

    F2 Furan Fatty Acid, 3-methyl-5-pentyl-2-Furannonanoic Acid, 9M5

     A furan fatty acid
  33. GC48778 Gadoleic Acid

    C20:1(9Z), cis-11-Eicosenoic Acid

     A monounsaturated fatty acid
  34. GC48763 Gestodene-d6

    SHB 331-d6; WL 70-d6

     An internal standard for the quantification of gestodene
  35. GC48738 (±)12-HETE-d8

    (±)12-Hydroxyeicosatetraenoic Acid-d8

     An internal standard for the quantification of 12-HETE
  36. GC48724 Pregnanetriol

    孕三醇

     A metabolite of 17α-hydroxyprogesterone
  37. GC48721 6-O-Demethyl Griseofulvin

    6-Demethylgriseofulvin

     A metabolite of griseofulvin
  38. GC48720 Griseofulvic Acid

    (±)-Griseofulvic Acid

     A metabolite of griseofulvin
  39. GC48719 (S)-Canadine

    四氢小檗碱,(-)-Canadine; (S)-(-)-Canadine

     An alkaloid with insecticidal activity
  40. GC48686 Prostaglandin E2-d4 MaxSpec® Standard

    Dinoprostoned4, PGE2d4

     A quantitative analytical standard guaranteed to meet MaxSpec identity, purity, stability, and concentration specifications
  41. GC48677 Sulindac-d3

    MK-231-d3

     An internal standard for the quantification of sulindac
  42. GC48650 DTUN A lipophilic hyponitrite radical initiator
  43. GC48649 7-hydroxy Chlorpromazine (hydrochloride) An active metabolite of chlorpromazine
  44. GC48645 1,3,4,6-Tetra-O-acetyl-2-azido-2-deoxy-α-D-Glucopyranose

    1,3,4,6-四-O-乙酰基-2-叠氮-2-脱氧-Α-D-吡喃葡萄糖

     A carbohydrate building block
  45. GC48617 2-Methylhexacosane

    2-Me-C26

     An insect pheromone
  46. GC48611 Ambroxol-d5

    盐酸氨溴索D5

     An internal standard for the quantification of ambroxol
  47. GC48553 Hyocholic Acid-d4

    HCA-d4, γ-MCA-d4, γ-Muricholic Acid-d4

     An internal standard for the quantification of hyocholic acid
  48. GC48528 Piericidin B A bacterial metabolite with insecticidal and antimicrobial activities
  49. GC48521 KRP 297

    MK-0767

     A dual agonist of PPARα and PPARγ
  50. GC48509 Apigenin 7-O-Glucuronide (hydrate) Apigenin 7-O-glucuronide is a flavonoid that has been found in J
  51. GC48508 (4-Carboxybutyl-d4)triphenylphosphonium (bromide)

    TPP-d4, 5-Triphenylphosphoniovaleric Acid-d4

     An internal standard for the quantification of (4-carboxybutyl)triphenylphosphonium

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