CYP3A/CYP450

CYP3A4 is an enzyme of cytochrome P450 superfamily found in human liver. It catalyzes the metabolism of endogenous and exogenous agents ( e.g. xenobiotics).

Products for CYP3A/CYP450

Cat.No. 产品名称 Information
GC10762 4β-hydroxy Cholesterol
4Β-羟基胆固醇
An oxysterol
GC14618 PPOH Selective inhibitor of epoxygenation reactions catalyzed by CYP4A2 and CYP4A3
GC10778 DDMS
Dibromo-dodecenyl-methylsulfimide
A potent inhibitor of 20-HETE synthesis
GC11731 4-phenyl-1,2,3-Thiadiazole
4-苯基-1,2,3-噻重氮,NSC 111906
Selective inhibitor of CYP2B4 and CYP2E1
GC11864 6,7-dihydroxy Bergamottin
二羟基香柠檬素,6,7-DHB
A potent CYP3A4 inhibitor
GC16550 Diosmetin
香叶木素
A flavonoid with diverse biological activities
GC13784 7-Ethoxyresorufin
乙氧基试卤灵,Resorufin ethyl ether
A fluorogenic substrate for, and inhibitor of, CYP1A1
GC16777 YM 511 YM 511 是一种高度特异性的非甾体芳香酶抑制剂。
GC10554 3-Cyano-7-ethoxycoumarin
3-氰基-7-乙氧基香豆素
A fluorogenic CYP450 substrate
GC15445 TMS
2,3',4,5'-四甲氧基二苯乙烯,(E)-2,3',4,5'-tetramethoxystilbene
A potent inhibitor of CYP1B1
GC17552 Pentoxyresorufin
7-羟基吩噁嗪酮二戊醚; Pentoxyresorufin
A fluorogenic substrate for CYP enzymes
GC10886 Methoxyresorufin
甲氧基试卤灵,Methoxyresorufin
A fluorogenic CYP1A1/2 substrate
GC14781 1-Aminobenzotriazole (ABT)
1-氨基苯并三唑,ABT; 3-Aminobenzotriazole
1-Aminobenzotriazole (ABT)是具有口服活性的细胞色素P450（CYP）的非特异性和不可逆抑制剂。
GC14382 VT-464 R enantiomer CYP17 lyase inhibitor
GC16073 Dronedarone
决奈达隆; SR 33589
An antiarrhythmic agent
GC16754 Clarithromycin
克拉霉素
A macrolide antibiotic
GC13079 Voriconazole
伏立康唑,(±)-UK-109496
A triazole antifungal agent
GC14269 Cobicistat (GS-9350)
可比司他,GS-9350
An inhibitor of CYP3A