Phospholipase(磷脂酶)
Phospholipases are enzymes that catalyze the hydrolysis of phospholipids into fatty acids and other lipid mediators. It plays a variety of roles in tumorgenesis , inflammation and brain disorders etc.
Products for Phospholipase
- Cat.No. 产品名称 Information
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GC44549
Palmitoyl thio-PC
A chromogenic substrate for PLA2
-
GC44223
ML-299
CID 56593087
Dual inhibitor of PLD1 and PLD2 -
GC44222
ML-298
A selective inhibitor of PLD2
-
GC43815
Heptanoyl thio-PC
A thioester phospholipase substrate
-
GC43812
HEPC
2Hexadecanoylthio1Ethylphosphorylcholine
A thioester phospholipase substrate -
GC43756
GK187
A GVIA iPLA2 inhibitor
-
GC43701
FTY720 phenoxy-biotin
Biotin-tagged FTY720 analog
-
GC43695
Folipastatin
磷脂他汀
An inhibitor of PLA2 -
GC43671
FKGK 18
An inhibitor of GVIA iPLA2
-
GC43670
FKGK 11
A selective iPLA2 inhibitor
-
GC43305
Compound 48/80 (hydrochloride)
C48/80 trihydrochloride
复合物48/80三盐酸盐是N-甲基-p-甲氧基苯乙胺与甲醛缩合产物的混合物。 -
GC43179
CAY10590
GK115
A potent and selective sPLA2 inhibitor -
GC43161
CAY10502
A potent inhibitor of cPLA2α
-
GC42885
AX 048
A cPLA2 inhibitor
-
GC42855
ARN19874
An inhibitor of NAPE-PLD
-
GC42843
Arachidonoyl thio-PC
2-deoxy-2-thio Arachidonoyl PC
A PLA2 substrate -
GC42611
7-hydroxycoumarinyl-γ-Linolenate
UmbelliferylγLinolenate
A fluorogenic substrate -
GC42029
1-Palmitoyl-2-linoleoyl PE
1-Palmitoyl-2-Linoleoyl PE, PLPE, (1Palmitoyl, 2Linoleoyl)Phosphatidylethanolamine, (1Palmitoyl, 2Linoleoyl)Phosphoethanolamine
A product of lipid biosynthesis -
GC41808
1,2-Dioctanoyl PC
3-二(辛酰氧基)丙基2-(三甲基铵基)乙基磷酸酯
A short chain analog of phosphatidylcholine -
GC41782
1,2-bis(heptanoylthio) Glycerophosphocholine
Diheptanoyl ThioPC, 1,2bis(Heptanoylthio)1,2dideoxysnglycero3phosphorylcholine
A substrate for PLA2s -
GC41004
Rhamnetin
鼠李素
A flavonoid with diverse biological activities -
GC40794
Sphinganine (d18:0)
D-赤式-C18-二氢-D-神经鞘氨醇
Sphinganine (d18:0)是一种鞘脂代谢途径的中间体。 -
GC40679
(S)-Bromoenol lactone
(S)-BEL; (S,E)-Bromoenol lactone
A selective iPLA2β inhibitor -
GC40678
(R)-Bromoenol lactone
(R,E)-Bromoenol lactone
A selective iPLA2γ inhibitor -
GC40545
cis-Parinaric Acid
α-Parinaric Acid
A naturally-occurring PUFA -
GC33457
1-Naphthaleneacetic acid (1-Naphthylacetic acid)
1-萘乙酸; 1-Naphthylacetic acid
1-Naphthaleneacetic acid (α-Naphthaleneacetic acid) is a synthetic plant hormone in the auxin family. -
GC32768
Quinacrine dihydrochloride (Mepacrine dihydrochloride)
Quinacrine是一种荧光探针,使胆碱能受体蛋白发生构象转变,低μM水平对AML细胞具有作用活性,平均IC50为2.30μM。
-
GC32224
Lp-PLA2 -IN-1
Lp-PLA2-IN-1可以抑制beta-lactamase-IN-1的活性,例如动脉粥样硬化,阿尔茨海默氏症。
-
GC31825
Varespladib methyl (A-002)
A-002; LY333013
Varespladibmethyl (A-002) (A-002; LY333013) 是 II 组分泌型磷脂酶 A2 (PLA2) 的选择性抑制剂。 -
GC31355
AA26-9
AA26-9, KK007-N1
A pan-serine hydrolase inhibitor -
GC30610
LY 178002
LY178002是一种有效的5-lipoxygenase,phospholipaseA2抑制剂,对5-lipoxygenase的IC50值为0.6μM,能够抑制人多形核白细胞产生LTB4,同时可相对较弱地抑制cyclooxygenase的活性。
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GC30561
2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
2-(E-2-decenoylamino)ethyl2-(cyclohexylethyl)sulfide是一种由压力诱发的溃疡和低毒性抑制剂,可以在压力引起的溃疡大鼠中,维持磷脂酶A2(phospholipaseA2)和前列腺素E2(prostaglandinE2)的含量水平。
-
GC30464
Ecopladib (PLA 725)
PLA 725
Ecopladib (PLA 725) 是细胞溶质磷脂酶 A2α 的亚微摩尔抑制剂; (cPLA2α),在 GLU 胶束和大鼠全血试验中,IC50 分别为 0.15 μM 和 0.11 μM。 -
GC30180
ST271
ST271 is a tyrphostin-like protein tyrosine kinase (PTK) inhibitor which inhibits phospholipase D (PLD) activity.
-
GC11055
10-Pyrene-PC
1-Palmitoyl-2-pyrenedecanoyl Phosphatidylcholine
A substrate for some PLA2s -
GC19186
GW4869
GW4869是一种非竞争性中性鞘脂酶抑制剂,IC50为1微摩尔。
-
GC18691
CAY10594
CAY10594 是一种有效的磷脂酶 D2 (PLD2) 抑制剂(体外 IC50 为 140 nm,细胞内为 110 nm)。
-
GC18559
Lysophosphatidylethanolamines (egg)
溶血磷脂酰乙醇胺(鸡蛋)
A mixture of lysophosphatidylethanolamines isolated from egg -
GC18305
CAY10650
Potent cPLA2α inhibitor
-
GC11520
ST638
Α-氰基-(3-乙氧基-4-羟基-5-苯基硫代甲基)肉桂酰胺
Tyrosine kinase inhibitor -
GC14521
ONO-RS-082
A PLA2 inhibitor
-
GC10645
MJ33 (lithium salt)
An inhibitor of the PLA2 activity of Prdx6
-
GC18141
EA4
An inhibitor of PLA2 from red blood cells
-
GC11116
Thioetheramide-PC
1-Palmitylthio-2-palmitoylamido-1,2-dideoxy-sn-glycero-3-phosphorylcholine
A competitive, reversible inhibitor of sPLA2 -
GC11243
Halopemide
卤培米特,NSC 354856,R34301
Inhibitor of phospholipase D1 and D2 -
GC13276
Oleyloxyethyl Phosphorylcholine
磷酰胆碱
A PLA2 inhibitor
-
GC16770
Arachidonic Acid Leelamide
A novel fatty acid amide
-
GC13351
VU0359595
CID-53361951,ML-270
A selective PLD1 inhibitor -
GC11021
Bromoenol lactone
(6E)-Bromoenol lactone
A selective, potent, irreversible inhibitor of iPLA2 -
GC10565
7-hydroxycoumarinyl Arachidonate
Umbelliferyl Arachidonate
A substrate for cPLA2