Gutathione S-transferase(谷胱甘肽S-转移酶)
GSTs (Glutathione s-transferases)is a detoxification enzyme that catalyze the binding of electrophilic substrates to glutathione. They involved in removal of ROS, inhibition of Jun kinase and can conjugate non-catalytically to various ligands.
Products for Gutathione S-transferase
- Cat.No. 产品名称 Information
- GC64919 AZD9898 AZD9898 是一种口服有效的白三烯-C4 合成酶 (LTC4S) 抑制剂,IC50 值为 0.28 nM。AZD9898 减轻GABA 结合和肝毒性信号。AZD9898 可用于哮喘的研究。
-
GC35727
Coniferyl ferulate
阿魏酸松柏酯
A monolignal conjugate with diverse biological activities -
GC35759
Curzerene
莪术烯
Curzerene, a sesquiterpene isolated from the rhizome of Curculigo orchioides Gaertn with anti-cancer activity, inhibits glutathione S-transferase A1 (GSTA1) mRNA and protein expression and induces cell apoptosis. - GC10519 Ethacrynic acid - d5 An internal standard for the quantification of ethacrynic acid
-
GC18095
Ezatiostat
TER199;TLK199;Telintra
An inhibitor of GSTP1-1 -
GC13409
Ezatiostat hydrochloride
L-GAMMA-谷氨酰基-S-苄基-L-半胱氨酰基-2-苯基甘氨酸二乙酯盐酸盐,TER199; TLK199 hydrochloride
An inhibitor of GSTP1-1 - GC33342 GSTO-IN-2 GSTO-IN-2是一种谷胱甘肽S-转移酶(glutathioneS-transferase)抑制剂,对于GSTA2,GSTM1和GSTP1-1的IC50值分别为3.6,16.3,1.4μM。
- GC32971 GSTO1-IN-1 GSTO1-IN-1是一种有效的谷胱甘肽S-转移酶omega1(GSTO1)抑制剂,IC50为31nM。
-
GC17287
Iberin
3-甲基亚磺酰丙基异硫氰酸酯,NSC 321801
A natural isothiocyanate
-
GC63518
LAS17
LAS17 是一种强效的,不可逆的,选择性谷胱甘肽 S-转移酶 Pi (GSTP1) 抑制剂。LAS17 抑制 GSTP1 活性,IC50 为 0.5 µM.
-
GC44882
Seneciphylline
千里光菲灵碱
An alkaloid with diverse biological activities - GC65438 TK05 TK05 是一种有效选择性的白三烯 C4 合成酶 (LTC4S) 抑制剂,其 IC50 值为 95 nM。
-
GC30647
TLK117 (TER117)
TER117
TLK117 (TER117) 是 TLK199 的活性代谢物,选择性抑制谷胱甘肽 S-转移酶 P1-1 (GSTP1-1),Ki 为 0.4 ⋼M 用于 GSTP。