Others
- Cat.No. 产品名称 Information
- GC60568 Afatinib N-Oxide AfatinibN-Oxide是Afatinibdimaleate氧化降解过程中的杂质。Afatinibdimaleate是一种不可逆的EGFR家族抑制剂。
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GC33728
Afegostat (D-Isofagomine)
D-Isofagomine; Isofagomine
Afegostat (D-Isofagomine) 是一种药理学伴侣,它以高亲和力特异性和可逆地结合内质网 (ER) 中的 acid-β-葡萄糖苷酶 (GCase)。 -
GC33503
Afegostat D-Tartrate (D-Isofagomine (D-Tartrate))
D-Isofagomine D-Tartrate; Isofagomine D-Tartrate
A β-glucosidase inhibitor -
GC18285
Aflatoxin M2
黄曲霉毒素 M2
A natural mycotoxin -
GC41360
Aflatoxin R0
黄曲霉毒醇; Aflatoxin R0
A mutagenic metabolite of aflatoxin B1 -
GC16348
Afobazole
CM346
A multi-targeted anxiolytic drug with neuroprotective activities
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GC30663
Agarotetrol
沉香四醇
A chromone derivative - GC33019 AGI-24512 AGI-24512是用于治疗癌症的甲硫氨酸腺苷转移酶2A(MATA2)抑制剂。AGI-24512在体外阻断MTAP缺失的癌细胞的生长。
- GC33307 AGI-25696 AGI-25696是蛋氨酸腺苷转移酶(MATA2)抑制剂,对研究癌症有用。AGI-25696阻断体内MTAP缺失的肿瘤的生长。
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GC32462
Aglafoline (Aglafolin)
Aglafolin; Rocaglamide U; (-)-Methyl rocaglate
Aglafoline (Aglafolin) 以选择性和浓度依赖性方式抑制 PAF(血小板激活因子)在洗涤过的兔血小板中诱导的聚集和 ATP 释放反应。 - GC38590 AGX51 AGX51, a first-in-class pan-Id (inhibitors of DNA-binding/differentiation proteins) antagonist and degrader, inhibits the Id1-E47 interaction, leading to ubiquitin-mediated degradation of Ids, cell growth arrest, and reduces viability, also inhibits pathologic ocular neovascularization.
- GC11189 AI-10-49 AI-10-49 是一种蛋白质-蛋白质相互作用抑制剂,选择性结合 CBFβ-SMMHC 并破坏其与 RUNX1 的结合,FRET IC50 为 0.26 uM。
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GC30756
AKOS B018304
AKOS B018304, an arylalkylidene derivative with polar substitution at para-position, is a potent inhibitor of chikungunya virus with low micro molar activity.
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GC30338
AKR1C3-IN-1
3-(3,4-二氢-1H-异喹啉-2-磺酰基)-苯甲酸
An inhibitor of prostaglandin F synthase/AKR1C3 -
GC60569
Aladorian
ARM036
Aladorian(ARM036)是一种苯并噻吩衍生物,具有抗心律失常作用。Aladorian被用于心力衰竭和儿茶酚胺能多态室性心动过速的研究。 -
GC33761
Alagebrium chloride (ALT711)
阿拉氯胺; ALT711
Alagebrium chloride (ALT711) (ALT711) 是一种晚期糖基化终产物 (AGE) 抑制剂。 -
GC14613
Aldicarb
NSC 379586, 2-methyl-2-(methylthio)-Propionaldehyde, UC-21149
cholinesterase inhibitor -
GC12004
Alendronate sodium
阿伦膦酸钠,Fosamax
An FPP synthase inhibitor -
GC10348
Alendronate sodium hydrate
阿仑膦酸钠; Alendronate; MK 217; G-704650 Adronat
An FPP synthase inhibitor -
GC39476
Alendronic acid
阿仑膦酸
Alendronic acid (alendronate) is a nitrogen-containing, second generation bisphosphonate used for osteoporosis, osteogenesis imperfecta, and several other bone diseases. -
GC16953
Alibendol
阿利苯多
Alibendol 是一种解痉剂、利胆剂和胆汁动力剂。 -
GC33692
Alimemazine hemitartrate (Trimeprazine hemitartrate)
酒石酸异丁嗪,Trimeprazine hemitartrate
A histamine H1 receptor antagonist -
GC38233
Alizarin Red S sodium
茜素红S,ARS sodium
Alizarin Red S sodium (Alizarin red S mono sodiumsalt, ARS sodium, C.I. Mordant Red 3, C.I 58005, Alizarin Carmine, Alizarin Red, Alizarin sodium monosulfonate, Alizarin sulfonate sodium, Alizarinsulfonic acid sodium salt, Sodium alizarinsulfonate) is an anthraquinone dye that has been used to evaluate calcium-rich deposits by cells in culture. -
GC39337
Allylestrenol
烯丙雌醇
Allylestrenol is an orally active progestagen of the 19-nortestosterone series resembling progesterone. -
GC35296
Alnustone
桤木酮
Alnustone 是一种在草药和香料中发现的非酚双苯庚烷类化合物,是姜黄的成分之一。Alnustone 具有抗吐、抗炎作用。 -
GC19510
Alovudine
3'-脱氧-3-氟胸苷,3'-Fluoro-3'-deoxythymidine
A nucleoside analog -
GC31195
Alpertine (Win 31665)
阿尔哌汀,Win 31665
Alpertine (Win 31665) 是一种从美国专利 5955459 A 中提取的抗精神病药物。 -
GC38357
Aluminum Hydroxide
氢氧化铝
Aluminium hydroxide (Aluminic), found in nature as the mineral gibbsite, is amphoteric (i.e., it has both basic and acidic properties). It is used to treat symptoms of increased stomach acid, such as heartburn, upset stomach, sour stomach, or acid indigestion; also reduce phosphate levels in people with certain kidney conditions. - GC63535 ALV2 ALV2 是一种有效和选择性的 Helios 降解剂。ALV2 可以结合 CRBN,IC50 为 0.57 μM。Helios 是一种锌指转录因子,可以在炎症性肿瘤微环境中维持稳定的 Treg 细胞表型。
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GC10943
AM 92016 hydrochloride
N-[4-[3-[[2-(3,4-二氯苯基)乙基]甲基氨基]-2-羟基丙氧基]苯基]甲磺酰胺盐酸盐
An IKr inhibitor -
GC30431
Amantanium bromide
金刚溴铵
Amantaniumbromide是季铵化合物,用作治疗功能的防腐/消毒剂。 -
GC30126
Ambroxol (NA-872)
氨溴索; NA-872
Ambroxol, a substituted benzylamine, is an active metabolite of bromhexine. It is a potent inhibitor of the neuronal Na+ channels. -
GC19027
Amcasertib
BBI503
Amcasertib (BBI503) 是一种具有口服活性的小分子多激酶抑制剂。 Amcasertib 对 PC-9/GR 细胞中的 NANOG 和 CD133 表达和细胞活力具有抑制活性。作为一种具有潜在抗肿瘤活性的口服癌细胞干细胞激酶抑制剂,它目前正在多种癌症的 I 期临床试验中进行研究。 -
GC33973
Amcinafal (SQ 15102)
安西法尔; SQ 15102
Amcinafal (SQ 15102) 是一种活性二醇,用于对抗病毒复制和干扰素产生。 -
GC60575
Ametryn
莠灭净
Ametryn,是一种抑制光合作用和其他酶的过程的除草剂。Ametryn对一年生阔叶杂草和草本植物是有效的。 - GC35312 AMG 487 S-enantiomer AMG 487 S-enantiomer 是 AMG 487 的 S 型异构体。AMG 487 是趋化因子受体 CXCR3 的有效拮抗剂。
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GC35317
Amicarbazone
胺唑草酮; BAY314666; BAY-MKH 3586
Amicarbazone(BAY-MKH3586; BAY314666) 通过与光系统II(PSII)的 Qb 结构域结合而成为光合电子传递的有效抑制剂;具有广谱杂草控制的除草剂。 -
GC35318
Amifampridine
3,4-二氨基吡啶; 3,4-Diaminopyridine
3,4-Diaminopyridine (Amifampridine, pyridine-3,4-diamine) blocks presynaptic potassium channels, and subsequently prolongs the action potential and increases presynaptic calcium concentrations. It is a drug predominantly used in the treatment of a number of rare muscle diseases. -
GC15473
Amifostine
氨磷汀; WR2721
A broad-spectrum radioprotective thiol -
GC32021
Aminochlorthenoxazin (ICI 350)
ICI 350
Aminochlorthenoxazin (ICI 350) 是一种解热镇痛剂。 -
GC15727
Aminoguanidine hydrochloride
氨基胍盐酸盐; Pimagedine hydrochloride; GER-11; Aminoguanidinium chloride
An iNOS inhibitor -
GC35326
Amotosalen hydrochloride
S-59
Amotosalen hydrochloride (S-59) 是一种光活化的 DNA 和 RNA 交联的补骨脂素化合物,可用于中和病原体。 -
GC13574
Amoxapine
阿莫沙平; CL-67772
A tetracyclic antidepressant - GC34470 AMXT-1501 tetrahydrochloride AMXT-1501tetrahydrochloride是一种新型的多胺转运系统抑制剂。AMXT1501可阻断免疫活性小鼠中的肿瘤生长,但不能阻断缺乏T细胞无胸腺裸鼠中的肿瘤生长。
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GC35330
Amylase
淀粉酶
Diastase, a natural enzyme, catalyses the breakdown of starch into maltose. - GC30122 AMZ30 AMZ30 (ML136, CS-2122) is a selective and covalent inhibitor of protein phosphatase methylesterase-1(PME-1) with IC50 of 0.60 μM. AMZ30 reduces the demethylated form of PP2A in living cells.
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GC39339
Anakinra
阿那白滞素; AMG-719
阿那白滞素(Anakinra)是一种重组的、非糖基化的人类白细胞介素-1受体拮抗剂(IL-1Ra)。
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GC33001
Anethole trithione
茴三硫
A dithiolthione with diverse biological activities -
GC35344
Angelic anhydride
当归酸酐
Angelic anhydride (2-Methylisocrotonic Anhydride, (Z)-2-Methylbut-2-enoic anhydride) is a synthetic chemical and usually used in content determination assays and pharmacological experiments. -
GC35346
Angelol A
当归酚A
Angelol A 是从当归根中分离得到的香豆素,在 Caco-2 单层细胞模型中以被动扩散的运输方式为主。