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PKC(蛋白激酶C)

PKC (protein kinase C) is a serine/threonine protein kinase that mediates insulin signaling, actin cytoskeleton, cell mobility, apoptosis and tumorigenesis etc.

Products for  PKC

  1. Cat.No. 产品名称 Information
  2. GC43286 CMPD101 A GRK2 and GRK3 inhibitor
  3. GC43105 C8 Ceramide (d18:1.8:0)

    N-辛酰基-D-神经鞘氨醇; N-Octanoyl-D-erythro-sphingosine

    A cell-permeable ceramide analog
  4. GC42747 Afuresertib (hydrochloride)

    GSK2110183 hydrochloride

    A pan-Akt inhibitor
  5. GC40770 L-erythro Sphingosine (d18:1)

    双琥珀酰亚胺辛二酸酯

    A bioactive sphingolipid
  6. GC32870 Ingenol ((-)-Ingenol)

    巨大戟醇; (-)-Ingenol

    A PKC activator
  7. GC32811 LXS196

    LXS196; IDE196

    A PKC inhibitor
  8. GC32714 Mitoxantrone (mitozantrone)

    米托蒽醌; Mitozantrone; NSC 301739

    米托蒽醌Mitoxantrone是一种抗肿瘤的蒽醌衍生物。
  9. GC31959 AS2521780 AS2521780是新颖的PKCθ选择性抑制剂,IC50值为0.48nM。
  10. GC31912 VTX-27 A PKCθ inhibitor
  11. GC31892 Decursin ((+)-Decursin)

    紫花前胡素; (+)-Decursin

    A phytochemical with diverse biological activities
  12. GC31711 PKC-IN-1

    [(2S,5R)-2,5-二甲基-4-[(四氢-2H-吡喃-4-基)甲基]-1-哌嗪基][3-[(5-氟-2-甲基-4-嘧啶基)氨基]-4,6-二氢-6,6-二甲基吡咯并[3,4-C]吡唑-5(1H)-基]甲酮

    PKC-IN-1是一种有效的,ATP-竞争性的,可逆的PKC抑制剂,对人PKCβ和PKCα的Ki值分别为5.3和10.4nM,对人PKCα,PKCβI,PKCβII,PKCθ,PKCγ,PKCmu和PKCε的IC50值分别为2.3,8.1,7.6,25.6,57.5,314,808nM。
  13. GC31656 Ingenol Mebutate (Ingenol 3-angelate)

    巨大戟醇甲基丁烯酸酯; Ingenol 3-angelate; PEP005

    A natural cytotoxic diterpene ester
  14. GC30545 Malantide Malantide是一种十二肽,能够被PKA磷酸化,并且能够增强PKA的活性。
  15. GC30200 PKC-theta inhibitor PKC-theta inhibitor (compound 20) inhibits PKC-θ with an IC50 of 18 nM.
  16. GC18521 Cercosporin

    尾孢菌素

    A cytotoxic phytotoxin
  17. GC18354 Bisindolylmaleimide X (hydrochloride)

    BIM-X hydrochloride; Ro31-8425 hydrochloride

    A PKC inhibitor
  18. GC18246 R-59-949

    Diacylglycerol Kinase Inhibitor II, DKGI-II

    A DGK-α inhibitor
  19. GC14134 1,2-Dimyristoyl-sn-glycerol

    1,2-二肉豆蔻酸甘油酯,1,2-DMG

    A long-chain DAG
  20. GC18062 1,2-Dilauroyl-sn-glycerol

    1,2-二月桂酰-SN-甘油,1,2-DLG

    A long-chain DAG
  21. GC12662 1,2-Distearoyl-sn-glycerol

    1,2-Dioctadecanoyl-sn-glycerol,DSG

    A diacylglycerol
  22. GC10299 Hexadecyl Methyl Glycerol

    1-O-hexadecyl-2-O-methyl-sn-Glycerol

    A synthetic DAG
  23. GC16678 UCN-02

    7-epi-hydroxy Staurosporine

    A PKC inhibitor
  24. GC13877 1,2-Dipalmitoyl-sn-glycerol

    1,2-双棕榈酸甘油酯,1,2-DPG,NSC 269964

    A diacylglycerol
  25. GC17815 L-threo-Sphingosine C-18

    L-threo-Sphingosine C-18

    A D-erythro-sphingosine analog
  26. GC13226 Bisindolylmaleimide VIII (acetate)

    3-[1-(3-氨基丙基)-1H-吲哚-3-基]-4-(1-甲基-1H-吲哚-3-基)-1H-吡咯-2,5-二酮单乙酸盐,BIM VIII,Ro 31-7549

    A PKC inhibitor
  27. GC14716 Bisindolylmaleimide IV

    双吲哚马来酰亚胺IV,Arcyriarubin A,BIM IV

    A PKC inhibitor
  28. GC10343 α-Amyloid Precursor Protein Modulator α-Amyloid Precursor Protein Modulator 是一种细胞可渗透的苯并内酰胺衍生蛋白激酶 C (PKC) 激活剂,Ki 为 11.9 nM。
  29. GC15018 Hispidin

    6-[(1E)-2-(3,4-二羟基苯基)乙烯基]-4-羟基-2H-吡喃-2-酮

    A polyphenol with diverse biological activities
  30. GC16405 Safingol

    沙芬戈,L-threo-Dihydrosphingosine,L-threo-Sphinganine

    A dual inhibitor of PKC and SPHK
  31. GC11022 SB 218078 A potent Chk1 inhibitor
  32. GC13273 ZIP ZIP 是 PKMζ 的选择性肽抑制剂。
  33. GC17239 Bisindolylmaleimide V

    双吲哚马来酰亚胺,BIM V

    A S6K inhibitor
  34. GC10029 Ro 31-8220 methanesulfonate

    Ro 31-8220 methanesulfonate; Bisindolylmaleimide IX mesylate

    Inhibitor of protein kinase C
  35. GC17242 (-)-epigallocatechin

    (-)-表没食子儿茶素; Epigallocatechin; L-Epigallocatechin

    A green tea polyphenol
  36. GC10603 (-)-epicatechin gallate

    表儿茶素没食子酸酯; Epicatechin gallate; ECG; (-)-Epicatechin 3-O-gallate

    A natural polyphenol with diverse protective actions
  37. GC12695 Bryostatin 3 Bryostatin 3 是一种大环内酯,是一种蛋白激酶 C 激活剂,Ki 为 2.75 nM。 Bryostatin 3 可以阻断 12-O-tetradecanoylphorbol-13-acetate (TPA) 对细胞增殖的抑制作用,但不能阻断 TPA 增强的细胞-基质粘附。
  38. GC12842 Bryostatin 2 Protein kinase C (PKC) activator
  39. GC16475 Afuresertib

    GSK2110183

    A pan-Akt inhibitor
  40. GC14012 (-)-Indolactam V

    吲哚内酰胺V,Indolactam V

    A PKC activator
  41. GC10682 TAS 301

    3-(双(4-甲氧基苯基)亚甲基)吲哚啉-2-酮

    An inhibitor of Ca2+ mobilization and CaM kinase II
  42. GC12135 Bisindolylmaleimide II

    双吲哚马来酰亚胺II,Bis II

    A PKC inhibitor
  43. GC14583 R 59-022

    DKGI-I; Diacylglycerol kinase inhibitor I

    A DGK inhibitor
  44. GC10820 Rottlerin

    粗糠柴苦素,Mallotoxin; NSC 56346; NSC 94525

    An inhibitor of PKCδ and other protein kinases
  45. GC11605 C-1

    1-(5-异喹啉磺酰基)哌嗪盐酸盐

    C-1 是一种有效的蛋白激酶抑制剂,IC50 为 4 μM, 8 μM, 12 μM 和 240 μM 用于 cGMP 依赖性蛋白激酶 (PKG)、cAMP 依赖性蛋白激酶 (PKA) ,分别为蛋白激酶 C (PKC) 和 MLC 激酶。 C-1 也用作 ROCK 抑制剂。
  46. GC18055 SC-9

    NCM 119

    An activator of PKC
  47. GC13320 SC-10 Protein kinase C activator
  48. GC16510 ZIP, Biotinylated ZIP with a biotin moiety covalently attached
  49. GC15345 [Ala113]-MBP (104-118)

    肽抑制剂[ALA113]-MBP(104-118)

    [Ala113]-MBP (104-118) 是一种蛋白激酶 C (PKC) 的非竞争性肽抑制剂,IC50 范围为 28-62 μM。
  50. GC17727 [Ala107]-MBP (104-118)

    肽抑制剂[ALA107]-MBP(104-118)

    [Ala107]-MBP (104-118) 是一种蛋白激酶 C (PKC) 的非竞争性肽抑制剂,IC50 范围为 46-145 μM。
  51. GC11671 PKC fragment (530-558) Potent activator of protein kinase C

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