Tyrosine Kinase(酪氨酸激酶)
- Bcr-Abl(64)
- Ack1(2)
- Axl(6)
- ALK(54)
- BMX Kinase(3)
- Broad Spectrum Protein Kinase Inhibitor(10)
- c-FMS(35)
- c-Kit(55)
- c-MET(82)
- c-RET(7)
- CSF-1R(3)
- DDR1/DDR2 Receptor(1)
- EGFR(225)
- EphB4(1)
- FAK(33)
- FGFR(94)
- FLT3(82)
- HER2(15)
- IGF1R(33)
- Insulin Receptor(42)
- IRAK(28)
- ITK(10)
- Lck(1)
- LRRK2(21)
- PDGFR(104)
- PTKs/RTKs(3)
- Pyk2(6)
- ROR(38)
- Spleen Tyrosine Kinase (Syk)(32)
- Src(95)
- Tie-2 (4)
- Trk(40)
- VEGFR(181)
- Discoidin Domain Receptor(15)
- DYRK(28)
- Ephrin Receptor(12)
- RET(28)
- ROS(14)
- TAM Receptor(28)
- IGFBR(1)
- Others(55)
- Cat.No. 产品名称 Information
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GC19044
Avitinib maleate
艾维替尼马来酸盐; Abivertinib maleate; AC0010 maleate
A selective inhibitor of mutant EGFR -
GC18718
bpV(pic) (potassium hydrate)
Bisperoxovanadium(pic)
A PTEN inhibitor -
GC18591
GSK805
N-(2,6-二氯-2'-(三氟甲氧基)-[1,1'-联苯]-4-基)-2-(4-(乙基磺酰基)苯基)乙酰胺
An RORγt inverse agonist - GC18580 B355252 A neuroprotective agent
-
GC18492
GSK3179106
RET Kinase Inhibitor 1
A RET kinase inhibitor - GC18438 CGP 77675 An inhibitor of Src family kinases
-
GC18211
Ningetinib
宁格替尼
A multi-kinase inhibitor -
GC19012
(R)-GNE-140
(R)-3-((2-氯苯基)硫基)-4-羟基-6-(4-吗啉苯基)-6-(噻吩-3-基)-5,6-二氢吡啶-2(1H)-酮
(R)-GNE-140 是一种有效的乳酸脱氢酶 A (LDHA) 抑制剂,对 LDHA 和 LDHB 的 IC50 分别为 3 nM 和 5 nM; (R)-GNE-140 的效力是 S 对映体的 18 倍。 -
GC18168
JI-101
CGI1842
An inhibitor of VEGFR2, PDGFRβ, and EphB4 -
GC18167
AC710
N-[4-[[[[5-(叔丁基)-3-异恶唑基]氨基]羰基]氨基]苯基]-5-[(1-乙基-2,2,6,6-四甲基-4-哌啶基)氧基]-2-吡啶甲酰胺
A PDGFR family kinase inhibitor -
GC11737
AG957
NSC 654705,Tyrphostin AG957
An inhibitor of Bcr-Abl and c-Abl -
GC16235
AG-1295
酪氨酸磷酸化抑制剂AG1295,NSC 380341,Tyrphostin AG-1295
A selective inhibitor of PDGF receptor kinase -
GC12864
AG-1557
Tyrphostin AG-1557
An EGFR inhibitor -
GC15365
N-Acetylserotonin
N-乙酰-5-羟色胺,N-Acetyl-5-hydroxytryptamine,NAS
The immediate precursor of melatonin -
GC14951
Meleagrin
6-O-Methyloxaline
A Fabl inhibitor -
GC12461
HA-100 (hydrochloride)
C-1
An inhibitor of PKA, PKC, and PKG -
GC14890
AG-183
酪氨酸磷酸化抑制剂A51,Tyrphostin 51
An inhibitor of EGF receptor kinase - GC12251 Tandutinib (MLN518) HCl FLT3 inhibitor,potent and selective
-
GC13988
HNMPA
Hydroxy-2-naphthalenylmethyl Phosphonic Acid
An insulin receptor tyrosine kinase inhibitor -
GC11024
AG-213
酪氨酸磷酸化抑制剂,Tyrphostin AG-213,Tyrphostin 47
An inhibitor of EGF receptor kinase -
GC10217
RG-14620
Tyrphostin RG14620
An inhibitor of EGF receptor kinase -
GC11845
AG-82
酪氨酸磷酸化抑制剂25,NSC 676484,RG-50875,Tyrphostin 25,Tyrphostin AG-82
An inhibitor of EGF receptor kinase -
GC16062
VEGFR Tyrosine Kinase Inhibitor II
Vascular Endothelial Growth Factor Tyrosine Kinase Inhibitor II
An inhibitor of KDR, FLT1, and c-Kit -
GC11712
AG-370
NSC 651712
A selective inhibitor of PDGF receptor kinase. -
GC16798
LDN-211904
N-(2-氯苯基)-6-(4-哌啶基)-咪唑并[1,2-A]吡啶-3-甲酰胺草酸盐
An EphB3 kinase inhibitor -
GC12370
IKK-16 (hydrochloride)
IKK Inhibitor VII
A potent inhibitor of IKKs -
GC17925
PKR-IN-C16
C16,GW 506033X,Protein Kinase RNA-activated
PKR-IN-C16 (Compound C16) is a specific double-stranded RNA-dependent protein kinase (PKR) inhibitor.
- GC14054 SR 0987 An agonist of RORγt
- GC10408 2-D08 An inhibitor of sumoylation
-
GC12818
4-methyl Erlotinib
埃罗替尼杂质G
A methylated analog of erlotinib -
GC10706
Rp-8-pCPT-Cyclic GMPS (sodium salt)
Rp-8-pCPT-cGMPS
A competitive inhibitor of cGK isoforms -
GC10517
Rp-8-bromo-Cyclic GMPS (sodium salt)
Rp-8-bromo-cGMPS
A competitive inhibitor of cGK - GC15145 CEP-28122 An orally active ALK inhibitor
- GC15314 PD 166326 An inhibitor of c-src and certain receptor tyrosine kinases, including c-abl
-
GC10938
AAL-993
VEGFR Tyrosine Kinase Inhibitor VI,ZK 260253
Inhibitor of VEGFR1, 2, and 3 - GC13905 GSK2981278 An inverse agonist of RORγ
-
GC14544
JNJ-10198409
3-氟-N-(6,7-二甲氧基-2,4-二氢茚并[1,2-C〕吡唑-3-基)苯基胺
A potent PDGF tyrosine kinase inhibitor -
GC10644
Neoruscogenin
新鲁斯可皂苷元
A bioavailable agonist of RORα - GC14418 SR 1555 (hydrochloride) inverse agonist of RORγ
-
GC15280
Tivozanib (hydrate)
AV-951,KRN 951
A VEGFR inhibitor - GC16483 MAZ51 MAZ51是一种选择性血管内皮生长因子受体3(VEGFR-3;FLT4)酪氨酸激酶抑制剂。
-
GC11312
EGFR Inhibitor
Epidermal Growth Factor Receptor Inhibitor
A selective antagonist of the EGFR - GC14856 EGFR/ErbB2 Inhibitor A dual inhibitor of EGFR and ErbB2
-
GC13961
ISCK03
STEM-CELLFACTOR/C-KIT抑制剂 ,c-Kit Inhibitor II,Stem-Cell Factor/c-Kit Inhibitor
An inhibitor of SCF/c-kit signaling - GC14103 NSC228155 An EGFR activator and inhibitor of KID-KIX interactions
-
GC15370
Olmutinib (HM61713, BI 1482694)
奥莫替尼
An inhibitor of mutant EGFR - GC12712 NT157 IRS-1/2 抑制剂,抑制 IGF-1R 和 STAT3 信号通路
-
GC11726
BAW2881 (NVP-BAW2881)
BAW2881
A VEGFR inhibitor - GC15340 BFH772 An inhibitor of VEGFR2
- GC15655 AMG 337 A selective c-Met inhibitor