Search Site
  • 0
    My Cart

    Click Here to Find How Many Items You Have Added:)

qq在线咨询
Home >> Signaling Pathways >> Tyrosine Kinase >> VEGFR

VEGFR(血管内皮生长因子受体)

VEGFR are receptors for vascular endothelial growth factor and belong to receptor tyrosine kinases.

Products for  VEGFR

  1. Cat.No. 产品名称 Information
  2. GC30242 Acrizanib

    LHA510

     Acrizanib是VEGFR-2的抑制剂，其IC50值为17.4nM。
  3. GC19332 Sitravatinib

    MGCD516; MG-516

     A multi-kinase inhibitor
  4. GC19108 SCR-1481B1

    麦他替尼胺丁三醇,c-Met inhibitor 2

     A pyridone
  5. GC18211 Ningetinib

    宁格替尼

     A multi-kinase inhibitor
  6. GC18168 JI-101

    CGI1842

     An inhibitor of VEGFR2, PDGFRβ, and EphB4
  7. GC16062 VEGFR Tyrosine Kinase Inhibitor II

    Vascular Endothelial Growth Factor Tyrosine Kinase Inhibitor II

     An inhibitor of KDR, FLT1, and c-Kit
  8. GC10938 AAL-993

    VEGFR Tyrosine Kinase Inhibitor VI,ZK 260253

     Inhibitor of VEGFR1, 2, and 3
  9. GC15280 Tivozanib (hydrate)

    AV-951,KRN 951

     A VEGFR inhibitor
  10. GC16483 MAZ51 MAZ51是一种选择性血管内皮生长因子受体3（VEGFR-3；FLT4）酪氨酸激酶抑制剂。
  11. GC11726 BAW2881 (NVP-BAW2881)

    BAW2881

     A VEGFR inhibitor
  12. GC15340 BFH772 An inhibitor of VEGFR2
  13. GC10165 Dovitinib (TKI258) Lactate

    多韦替尼,TKI258 lactate hydrate; CHIR-258 lactate hydrate

     A multi-kinase inhibitor
  14. GC10355 Fruquintinib(HMPL-013)

    呋喹替尼; HMPL-013

     An inhibitor of VEGF1, -2, and -3
  15. GC17959 AZD2932 A multi-kinase inhibitor
  16. GC16604 Altiratinib

    DCC-2701

     A multiple kinase inhibitor
  17. GC15801 ACTB-1003

    ACTB-1003

     A multi-kinase inhibitor
  18. GC17098 DMH4 A VEGFR2 inhibitor
  19. GC10195 Z-Guggulsterone

    孕二烯二酮

     Z-Guggulsterone 是阿育吠陀药用植物 Commiphora mukul 的一种成分，在体外和体内抑制血管生成，IC50 值为 1740、1000、220 和 >； 50000 nM 用于糖皮质激素、盐皮质激素、雄激素和法尼醇 X 受体 。
  20. GC13344 (Z)-FeCP-oxindole (Z)-FeCP-oxindole 是一种选择性人血管内皮生长因子受体 2 (VEGFR2) 抑制剂，IC50 值为 200 nM。 (Z)-FeCP-oxindole 在 10 μM 时可显着抑制 VEGFR1 和 PDGFRa 或 b。 (Z)-FeCP-oxindole 具有一定的抗癌活性，作用于 B16 鼠黑色素瘤系，IC50 小于 1 μM。
  21. GC17800 (E)-FeCP-oxindole VEGFR-2 inhibitor
  22. GC13944 (5Z)-7-Oxozeaenol

    FR148083,L-783,279,LL-Z 1640-2

     A selective TAK1 inhibitor
  23. GC11417 SU 4312

    NSC 86429

     A selective dual inhibitor of VEGFR2 and PDGFR
  24. GC16183 EG00229 An NRP-1 antagonist
  25. GC13833 BMS-794833 An inhibitor of c-Met and VEGFR2
  26. GC10758 Tyrphostin 9

    酪氨酸磷酸化抑制剂A9,Tyrphostin 9; Malonoben

     An inhibitor of EGF receptor kinase
  27. GC11555 ZM 323881 HCl

    5-[(7-苄氧基喹唑啉-4-基)氨基]-4-氟-2-甲基苯酚盐酸盐

     A potent and selective VEGFR2 inhibitor
  28. GC12586 SAR131675 An inhibitor of VEGFR3
  29. GC14292 Apatinib Mesylate

    阿帕替尼

    A selective VEGFR2 inhibitor
  30. GC17715 Golvatinib (E7050)

    N-[2-氟-4-[[2-[[[4-(4-甲基哌嗪-1-基)哌啶-1-基]羰基]氨基]吡啶-4-基]氧基]苯基]-N'-(4-氟苯基)环丙烷-1,1-二甲酰胺,E-7050

     A dual inhibitor of c-Met and VEGFR2
  31. GC12980 CP-673451 A selective PDGFRα/β kinase inhibitor
  32. GC12531 Cabozantinib malate (XL184)

    卡博替尼苹果酸盐; XL184 S-malate; BMS-907351 S-malate

     A VEGFR2 inhibitor
  33. GC11003 PP121 A potent dual inhibitor of tyrosine and phosphoinositide kinases
  34. GC17651 Sunitinib

    舒尼替尼; SU 11248

     舒尼替尼Sunitinib（SU 11248）是一种具口服活性的多靶点受体酪氨酸激酶抑制剂，对血管内皮生长因子受体（VEGFR2）和血小板衍生生长因子受体（PDGFRβ）的IC50分别为80nM和2nM。
  35. GC10220 TAK-593 TAK-593 是一种有效的 VEGFR 和 PDGFR 家族抑制剂，对 VEGFR1、VEGFR2、VEGFR3、PDFGRα 和 PDFGRβ 的 IC50 分别为 3.2、0.95、1.1、4.3 和 13 nM。
  36. GC13738 SKLB1002 A VEGFR2 inhibitor
  37. GC12185 ZM 306416

    CB 676475

     A VEGF receptor kinase inhibitor
  38. GC16000 WHI-P180

    3-[(6,7-二甲氧基-4-喹唑啉基)氨基]苯酚,Janex 3

     A multi-kinase inhibitor
  39. GC15022 Vandetanib (ZD6474)

    凡德他尼; ZD6474

     A multi-kinase inhibitor
  40. GC11763 Telatinib (BAY 57-9352)

    替拉替尼,BAY 579352;BAY 57 9352

     A multi-kinase inhibitor
  41. GC11372 Dovitinib Dilactic acid

    多韦替尼二乳酸

     FLT3 inhibitor
  42. GC12216 Axitinib (AG 013736)

    阿昔替尼; AG-013736

     Axitinib (AG 013736)是一种具有口服活性的特异性血管内皮生长因子受体（VEGFR）抑制剂，主要靶向VEGFR-1、VEGFR-2和VEGFR-3，IC50值分别为 0.1nM、0.2nM和0.1-0.3nM。
  43. GC12730 Pazopanib Hydrochloride

    盐酸帕唑帕尼; GW786034 (Hydrochloride)

     A multi-kinase inhibitor
  44. GC15818 RAF265

    CHIR-265;RAF 265;RAF-265;CHIR265

     A B-Raf and VEGFR2 inhibitor
  45. GC12590 KRN 633

    N-[2-氯-4-[(6,7-二甲氧基-4-喹唑啉基)氧基]苯基]-N'-丙基脲

     A VEGF receptor tyrosine kinase inhibitor
  46. GC14396 Ponatinib (AP24534)

    普纳替尼; AP24534

     An inhibitor of native and mutant Bcr-Abl
  47. GC16732 TSU-68 (SU6668,Orantinib)

    SU6668; TSU-68

     An inhibitor of select receptor tyrosine kinases
  48. GC17955 Vatalanib (PTK787) 2HCl

    瓦他拉尼,PTK787 dihydrochloride; CGP-797870 dihydrochloride; ZK-222584 dihydrochloride

     A potent and selective VEGF receptor inhibitor
  49. GC14238 Brivanib Alaninate (BMS-582664)

    1-[[4-[(4-氟-2-甲基-1H-吲哚-5-基)氧基]-5-甲基吡咯并[2,1-F][1,2,4]三嗪-6-基]氧基]-2-丙醇L-丙氨酸酯,BMS-582664

     A prodrug form of brivanib
  50. GC15735 Foretinib (GSK1363089)

    N-[3-氟-4-[[6-甲氧基-7-[[3-(吗啉-4-基)丙基]氧]喹啉-4-基]氧]苯基]-N'-(4-氟苯基)环丙烷-1,1-二甲酰胺,XL880; GSK1363089; GSK089; EXEL-2880

     A broad-spectrum tyrosine kinase inhibitor
  51. GC11336 Motesanib Diphosphate (AMG-706)

    二磷酸莫替沙尼,AMG 706 Diphosphate

     A multikinase inhibitor

Items 101 to 150 of 192 total

per page
  2. 1
  3. 2
  4. 3
  5. 4

Set Descending Direction