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Home >> Signaling Pathways >> Ubiquitination/ Proteasome

Ubiquitination/ Proteasome(泛素化/蛋白酶体)

  1. Cat.No. 产品名称 Information
  2. GC17995 Tacrolimus monohydrate

    他克莫司一水合物; FK506 monohydrate; Fujimycin monohydrate; FR900506 monohydrate

     他克莫司一水合物 (FK506 monohydrate) 是一种大环内酯，与 FK506 结合蛋白 (FKBP) 结合形成复合物并抑制钙调神经磷酸酶，从而抑制 T 淋巴细胞信号转导和 IL-2 转录。
  3. GC16993 PFK-015 A selective inhibitor of PFKFB3
  4. GC10441 Cabergoline

    卡麦角林; FCE-21336

     A potent and selective dopamine D2 receptor agonist
  5. GC16105 Iohexol

    碘海醇

     A contrast reagent
  6. GC13869 Fasudil

    法舒地尔; HA-1077; AT877

     Fasudil（法舒地尔；HA-1077；AT877）是一种非特异性RhoA/ROCK抑制剂，对ROCK1的Ki为0.33μM，IC50为0.158μM，对ROCK2和PKA、PKC、PKG的IC50分别为4.58μM、12.30μM、1.650μM。
  7. GC10356 DUBs-IN-3

    9-[(2-丙烯-1-氧基)亚氨基]-9H-茚并[1,2-B]吡嗪-2,3-二甲腈

     DUBs-IN-3 是一种有效的去泛素酶 (USP) 酶抑制剂，从参考化合物 22c 中提取，对 USP8 的 IC50 为 0.56 μM。
  8. GC17125 DUBs-IN-2

    9-乙氧基亚氨基-9H-茚并[1,2-B]吡嗪-2,3-二甲腈

     DUBs-IN-2 是一种有效的去泛素酶抑制剂，IC50 为 0.28 μM for USP8。
  9. GC17616 PPQ-102

    CFTR Inhibitor

     A CFTR channel inhibitor
  10. GC10579 Ouabain Octahydrate

    乌本(箭毒)苷,哇巴因,Acocantherine; G-Strophanthin

     Ouabain Octahydrate 是 Na+/K+-ATPase 的抑制剂，用于治疗充血性心力衰竭。
  11. GC16843 Hydroxyurea

    羟基脲; Hydroxycarbamide

     An antineoplastic agent
  12. GC15212 Divalproex Sodium

    双丙戊酸钠,VPA (sodium)

     A prodrug form of valproic acid
  13. GC10976 Noradrenaline bitartrate monohydrate

    酒石酸去甲肾上腺素; Levarterenol bitartrate monohydrate; L-Noradrenaline bitartrate monohydrate

     An adrenoceptor agonist
  14. GC14577 Sulfacetamide Sodium

    磺胺醋酰钠

     A sulfonamide antibiotic
  15. GC14142 Acetylcholine Chloride

    氯化乙酰胆碱; ACh chloride

     A neurotransmitter
  16. GC12017 Isoniazid

    异烟肼; INH; Isonicotinic acid hydrazide; Isonicotinic hydrazide

     An inhibitor of mycolic acid synthesis
  17. GC12226 Cisatracurium Besylate

    顺苯磺酸阿曲库铵; 51W89

     A competitive antagonist of nAChRs and non-depolarizing muscle relaxant
  18. GC15857 Sodium butyrate

    丁酸钠

     A short-chain fatty acid and HDAC inhibitor
  19. GC17082 Pirarubicin

    吡柔比星; THP

     An anthracycline antitumor antibiotic
  20. GC16486 Novobiocin Sodium

    新生霉素钠,Albamycin sodium; Cathomycin sodium

     An inhibitor of DNA gyrase
  21. GC14563 Ketanserin

    酮色林; R41468

     A potent 5-HT2 receptor antagonist
  22. GC17974 Latrepirdine dihydrochloride

    2,3,4,5-四氢-2,8-二甲基-5-[2-(6-甲基-3-吡啶基)乙基]-1H-吡啶并[4,3-B]吲哚二盐酸盐,Dimebolin dihydrochloride

     A neuroprotective agent
  23. GC12376 Maprotiline HCl

    盐酸马普替林

     A tricyclic antidepressant
  24. GC17229 Paroxetine HCl

    盐酸帕罗西汀; BRL29060 hydrochloride; BRL29060A

     A selective serotonin reuptake inhibitor
  25. GC16999 Nitrendipine

    尼群地平; BAY-E-5009

     An L-type calcium channel blocker
  26. GC14216 Chlorpromazine HCl

    盐酸氯丙嗪

     Chlorpromazine HCl是一种口服有效的、可透过血脑屏障的吩噻嗪类抗精神病药，能够有效抑制D2多巴胺受体和5-HT2A，具有很强的镇静作用。
  27. GC15024 Nifedipine

    硝苯地平; BAY-a-1040

     An L-type calcium channel blocker
  28. GC16921 Bromhexine HCl

    盐酸溴己新

     Bromhexine HCl 是一种有效且特异性的 TMPRSS2 蛋白酶抑制剂，IC50 为 0.75 μM。
  29. GC13974 Salbutamol Sulfate

    沙丁胺醇半硫酸盐; Albuterol hemisulfate; AH-3365 hemisulfate

     A β2-AR agonist
  30. GC10750 Dexmedetomidine HCl

    盐酸右美托咪定; (+)-Medetomidine hydrochloride; (S)-Medetomidine hydrochloride

     An α2-adrenoceptor agonist
  31. GC10132 Ciclopirox

    环吡酮胺; HOE296b

     An iron chelator, antifungal, and anticancer agent
  32. GC11885 Sevelamer HCl

    盐酸司维拉姆

     Sevelamer HCl 是一种磷酸盐结合药物，用于治疗慢性肾病患者的高磷血症；由与环氧氯丙烷交联的聚烯丙胺组成。
  33. GC14273 TTNPB (Arotinoid Acid)

    Ro 13-7410; Arotinoid acid; AGN191183

     A potent, selective RAR agonist
  34. GC13031 Trifluoperazine 2HCl

    盐酸三氟拉嗪；甲哌氟丙嗪；三氟吡拉嗪

     An anti-adrenergic and anti-dopaminergic agent
  35. GC10424 Tolbutamide

    甲苯磺丁脲

     A SUR1/Kir6.2 channel inhibitor
  36. GC12736 Thiamet G Thiamet G 是一种有效的 O-GlcNAcase 抑制剂 (Ki =21 nM)，用于提高 O-GlcNAcylation 水平。
  37. GC17151 Tempol

    阻聚剂701,4-Hydroxy-TEMPO

     A nitroxide and spin label with SOD mimetic activity
  38. GC15184 Taurine

    牛磺酸; 2-Aminoethanesulfonic acid

     A sulfur-containing amino acid
  39. GC13918 STF-62247

    N-(3-甲基苯基)-4-(4-吡啶)-2-噻唑胺

     Inducer of autophagy in renal cell carcinoma cells
  40. GC12516 Spironolactone

    螺内酯; SC9420

     An Analytical Reference Standard
  41. GC11033 Rupatadine Fumarate

    富马酸卢帕他定; UR-12592 Fumarate

     A histamine H1 and PAF receptor antagonist
  42. GC14263 Proflavine Hemisulfate

    硫酸原黄素,Proflavin hemisulfate; 3,6-Diaminoacridine hemisulfate

     Proflavine hemisulfate，一种吖啶染料，是一种已知的 DNA 嵌入剂。
  43. GC10458 Penfluridol

    五氟利多; R-16341

     A typical antipsychotic
  44. GC10678 Nicardipine HCl

    盐酸尼卡地平; YC-93

     An L-type calcium channel blocker
  45. GC13252 Meclizine 2HCl

    盐酸美克洛嗪; Meclozine dihydrochloride

     A histamine H1 receptor antagonist
  46. GC15929 Levosimendan

    左西孟旦; Simsndan; OR-1259

     A calcium sensitizer
  47. GC14764 Lamotrigine

    拉莫三嗪; LTG; BW430C

     An anticonvulsant
  48. GC15826 Isosorbide

    异山梨酯; D-Isosorbide; Dianhydro-D-glucitol

     A dianhydrohexitol
  49. GC10074 H 89 2HCl

    H-89二盐酸盐

     H-89 2HCl 是一种有效的选择性 camp 依赖性蛋白激酶 A 抑制剂，IC50 值为 48 nM，对 PKG、PKC、酪蛋白激酶和其他激酶表现出较弱的抑制作用 。
  50. GC17173 Felodipine

    非洛地平

     An L-type calcium channel inhibitor
  51. GC14968 Esmolol HCl

    盐酸艾司洛尔

     A β1-AR antagonist

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