HIV(人类免疫缺陷病毒)
HIV (human immunodeficiency virus) is a lentivirus that infect immune system. It cause immune system failure and lead to AIDS (acquired immnudeficiency syndrome).
Products for HIV
- Cat.No. 产品名称 Information
-
GC17040
DAPTA
D-Ala-peptide T-amide; Adaptavir
A CCR5 receptor antagonist -
GC12606
YYA-021
A small molecule CD4 mimetic
-
GC16706
AMD 3465 hexahydrobromide
GENZ-644494 hexahydrobromide
A CXCR4 receptor antagonist -
GC10473
AMD 3465
GENZ-644494
A CXCR4 receptor antagonist -
GC16843
Hydroxyurea
羟基脲; Hydroxycarbamide
An antineoplastic agent -
GC18016
Salicylanilide
水杨酰苯胺,2-Hydroxybenzanilide
Salicylanilide 具有广泛的生物活性,包括抗病毒效力,可通过靶向 HIV-1 整合酶或逆转录酶来抑制 HIV 病毒。 -
GC16825
Probenecid
丙磺舒
An inhibitor of OATs and MRP1 and an agonist of TRPV2 -
GC10811
Miltefosine
米替福新; HePC; Hexadecyl phosphocholine
An inhibitor of CCT -
GC14314
Aloperine
苦豆碱
An alkaloid with diverse biological activities -
GC12830
Stavudine (d4T)
司他夫定; d4T
An inhibitor of HIV reverse transcriptase -
GC15996
Etravirine (TMC125)
依曲韦林; R165335; TMC125
An NNRTI -
GC10637
Zidovudine
叠氮胸苷; Azidothymidine; AZT; ZDV
A nucleoside reverse transcriptase inhibitor -
GC14720
Zalcitabine
扎西他滨,2',3'-Dideoxycytidine; ddC; Dideoxycytidine
A nucleoside reverse transcriptase inhibitor -
GC17709
Nelfinavir
甲磺酸萘非那韦,AG1341
Nelfinavir Mesylate 是强效的HIV protease抑制剂,Ki为2 nM。 -
GC10263
BMS-378806 (BMS-806)
1-[(2R)-4-苯甲酰基-2-甲基-1-哌嗪基]-2-(4-甲氧基-1H-吡咯并[2,3-B]吡啶-3-基)-1,2-乙二酮,BMS-806
An HIV-1 entry inhibitor -
GC15488
Tenofovir maleate
替诺福韦马来酸盐; GS 1278 maleate; PMPA maleate
An HIV and HBV antiviral -
GC13846
Tenofovir hydrate
替诺福韦水合物; GS 1278 hydrate; PMPA hydrate
An HIV and HBV antiviral -
GC11688
Megestrol Acetate
醋酸甲地孕酮
A synthetic progestogen -
GC10570
BMS-538203
HIV integrase inhibitor,highly efficient
-
GC11424
Valproic acid
丙戊酸; VPA; 2-Propylpentanoic Acid
A class I HDAC inhibitor -
GC12389
Efavirenz
依法韦仑; DMP 266; EFV; L-743726
A non-nucleoside reverse transcriptase inhibitor -
GC15452
Delavirdine mesylate
U 90152 mesylate; BHAP-U 90152 mesylate
A non-nucleoside reverse transcriptase inhibitor -
GC14199
RVX-208
阿帕他隆; RVX-208; RVX000222
A selective BET bromodomain antagonist -
GC16425
Flavopiridol hydrochloride
(-)-2-(2-氯苯基)-5,7-二羟基-8-[(3S,4R)-3-羟基-1-甲基-4-哌啶基]-4H-1-苯并吡喃-4-酮盐酸盐,Alvocidib Hydrochloride; L86-8275 Hydrochloride; HMR-1275 Hydrochloride
An inhibitor of cyclin-dependent kinases -
GC10295
Chloroquine diphosphate
磷酸氯喹
An aminoquinoline
-
GC16215
GSK744 (S/GSK1265744)
卡博特韦; GSK-1265744; S/GSK1265744
An HIV-1 integrase inhibitor -
GC14452
Dapivirine (TMC120)
达匹维林; TMC120; R147681
A non-nucleoside reverse transcriptase inhibitor -
GC13653
Emtricitabine
恩曲他滨; BW1592
A nucleoside reverse transcriptase inhibitor -
GC15330
Didanosine
地达诺辛; 2',3'-Dideoxyinosine; ddI
An antiviral nucleoside analog and inhibitor of reverse transcriptase -
GC15392
Triciribine
曲西瑞宾,API-2; NSC 154020; TCN
A selective, potent inhibitor of Akt activation -
GC16387
Nevirapine
奈韦拉平; BI-RG 587; NSC 641530; NVP
An NNRTI -
GC10317
Lamivudine
拉米夫定; BCH-189
A nucleoside reverse transcriptase inhibitor -
GC15090
Maraviroc
马拉维若,UK-427857; Selzentry; Celsentri
马拉韦罗作为第一款CCR5拮抗剂已被批准用于治疗HIV感染,对hERG离子通道的IC50>10μM。
-
GC14289
Fasudil (HA-1077) HCl
盐酸法舒地尔; HA-1077 Hydrochloride; AT-877 Hydrochloride
Fasudil(法舒地尔;HA-1077;AT877)是一种非特异性RhoA/ROCK抑制剂,对ROCK1的Ki为0.33μM,IC50为0.158μM,对ROCK2和PKA、PKC、PKG的IC50分别为4.58μM、12.30μM、1.650μM。 -
GC12125
Tenofovir
替诺福韦; GS 1278; PMPA
An HIV and HBV antiviral -
GC15200
Aprepitant
阿瑞匹坦; MK-0869; MK-869; L-754030
An antiemetic and NK1 antagonist -
GC15067
Tenofovir Disoproxil Fumarate
富马酸替诺福韦酯,Tenofovir DF; Bis(POC)-PMPA fumarate; GS 4331 fumarate
A prodrug of the antiviral tenofovir -
GC17567
Doxorubicin (Adriamycin) HCl
盐酸阿霉素; Hydroxydaunorubicin hydrochloride
An anthracycline antitumor antibiotic
-
GC17421
Vicriviroc maleate
1-[(4,6-二甲基-5-嘧啶基)羰基]-4-[(3S)-4-[(1R)-2-甲氧基-1-[4-(三氟甲基)苯基]乙基]-3-甲基-1-哌嗪基]-4-甲基哌啶马来酸盐,Sch-417690; SCH-D
A CCR5 antagonist -
GC14454
Tipranavir
替拉那韦,Aptivus,Tipranavir
A nonpeptidic HIV protease inhibitor -
GC15785
Saquinavir mesylate
沙奎那韦甲磺酸盐; Ro 31-8959/003
An HIV protease inhibitor -
GC15335
Saquinavir
沙奎那韦; Ro 31-8959
Saquinavir (Ro 31-8959) 是一种 HIV 蛋白酶抑制剂,用于抗逆转录病毒治疗。 -
GC11059
Rilpivirine
利匹韦林; R278474; TMC278; DB08864
A non-nucleoside reverse transcriptase inhibitor -
GC14084
Nelfinavir Mesylate
甲磺酸奈非那韦,AG 1343 Mesylate;AG1343 Mesylate;AG-1343 Mesylate,Nelfinavir
An HIV-1 protease inhibitor -
GC16035
NBD-556
N-(4-氯苯基)-N'-(2,2,6,6-四甲基哌啶-4-基)草酰胺,NBD 556;NBD556
A small molecule CD4 mimetic -
GC16589
Limonin
柠檬苦素; Limonoic acid 3,19
柠檬苦素是一种天然的四环三萜类化合物,广泛存在于桉树、黄柏和黄连中。 -
GC16596
Lersivirine
3-氰基-5-[[3,5-二乙基-1-(2-羟基乙基)-1H-吡唑-4-基]氧基]苯腈,UK-453061;UK453061;UK 453061
An NNRTI -
GC12998
HIV-1 integrase inhibitor
4-[3-(叠氮基甲基)苯基]-2-羟基-4-氧代-2-丁烯酸
HIV-1整合酶抑制剂可用于抗HIV。 -
GC12555
GS-9620
维沙莫德; GS-9620
A TLR7 agonist -
GC11300
Fosamprenavir Calcium Salt
福沙那伟钙,GW 433908G;Lexiva;GW433908G;GW-433908G
A prodrug form of amprenavir