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HIV(人类免疫缺陷病毒)

HIV (human immunodeficiency virus) is a lentivirus that infect immune system. It cause immune system failure and lead to AIDS (acquired immnudeficiency syndrome).

Products for  HIV

  1. Cat.No. 产品名称 Information
  2. GC17040 DAPTA

    D-Ala-peptide T-amide; Adaptavir

    A CCR5 receptor antagonist
  3. GC12606 YYA-021 A small molecule CD4 mimetic
  4. GC16706 AMD 3465 hexahydrobromide

    GENZ-644494 hexahydrobromide

    A CXCR4 receptor antagonist
  5. GC10473 AMD 3465

    GENZ-644494

    A CXCR4 receptor antagonist
  6. GC16843 Hydroxyurea

    羟基脲; Hydroxycarbamide

    An antineoplastic agent
  7. GC18016 Salicylanilide

    水杨酰苯胺,2-Hydroxybenzanilide

    Salicylanilide 具有广泛的生物活性,包括抗病毒效力,可通过靶向 HIV-1 整合酶或逆转录酶来抑制 HIV 病毒。
  8. GC16825 Probenecid

    丙磺舒

    An inhibitor of OATs and MRP1 and an agonist of TRPV2
  9. GC10811 Miltefosine

    米替福新; HePC; Hexadecyl phosphocholine

    An inhibitor of CCT
  10. GC14314 Aloperine

    苦豆碱

    An alkaloid with diverse biological activities
  11. GC12830 Stavudine (d4T)

    司他夫定; d4T

    An inhibitor of HIV reverse transcriptase
  12. GC15996 Etravirine (TMC125)

    依曲韦林; R165335; TMC125

    An NNRTI
  13. GC10637 Zidovudine

    叠氮胸苷; Azidothymidine; AZT; ZDV

    A nucleoside reverse transcriptase inhibitor
  14. GC14720 Zalcitabine

    扎西他滨,2',3'-Dideoxycytidine; ddC; Dideoxycytidine

    A nucleoside reverse transcriptase inhibitor
  15. GC17709 Nelfinavir

    甲磺酸萘非那韦,AG1341

    Nelfinavir Mesylate 是强效的HIV protease抑制剂,Ki为2 nM。
  16. GC10263 BMS-378806 (BMS-806)

    1-[(2R)-4-苯甲酰基-2-甲基-1-哌嗪基]-2-(4-甲氧基-1H-吡咯并[2,3-B]吡啶-3-基)-1,2-乙二酮,BMS-806

    An HIV-1 entry inhibitor
  17. GC15488 Tenofovir maleate

    替诺福韦马来酸盐; GS 1278 maleate; PMPA maleate

    An HIV and HBV antiviral
  18. GC13846 Tenofovir hydrate

    替诺福韦水合物; GS 1278 hydrate; PMPA hydrate

    An HIV and HBV antiviral
  19. GC11688 Megestrol Acetate

    醋酸甲地孕酮

    A synthetic progestogen
  20. GC10570 BMS-538203 HIV integrase inhibitor,highly efficient
  21. GC11424 Valproic acid

    丙戊酸; VPA; 2-Propylpentanoic Acid

    A class I HDAC inhibitor
  22. GC12389 Efavirenz

    依法韦仑; DMP 266; EFV; L-743726

    A non-nucleoside reverse transcriptase inhibitor
  23. GC15452 Delavirdine mesylate

    U 90152 mesylate; BHAP-U 90152 mesylate

    A non-nucleoside reverse transcriptase inhibitor
  24. GC14199 RVX-208

    阿帕他隆; RVX-208; RVX000222

    A selective BET bromodomain antagonist
  25. GC16425 Flavopiridol hydrochloride

    (-)-2-(2-氯苯基)-5,7-二羟基-8-[(3S,4R)-3-羟基-1-甲基-4-哌啶基]-4H-1-苯并吡喃-4-酮盐酸盐,Alvocidib Hydrochloride; L86-8275 Hydrochloride; HMR-1275 Hydrochloride

    An inhibitor of cyclin-dependent kinases
  26. GC10295 Chloroquine diphosphate

    磷酸氯喹

    An aminoquinoline

  27. GC16215 GSK744 (S/GSK1265744)

    卡博特韦; GSK-1265744; S/GSK1265744

    An HIV-1 integrase inhibitor
  28. GC14452 Dapivirine (TMC120)

    达匹维林; TMC120; R147681

    A non-nucleoside reverse transcriptase inhibitor
  29. GC13653 Emtricitabine

    恩曲他滨; BW1592

    A nucleoside reverse transcriptase inhibitor
  30. GC15330 Didanosine

    地达诺辛; 2',3'-Dideoxyinosine; ddI

    An antiviral nucleoside analog and inhibitor of reverse transcriptase
  31. GC15392 Triciribine

    曲西瑞宾,API-2; NSC 154020; TCN

    A selective, potent inhibitor of Akt activation
  32. GC16387 Nevirapine

    奈韦拉平; BI-RG 587; NSC 641530; NVP

    An NNRTI
  33. GC10317 Lamivudine

    拉米夫定; BCH-189

    A nucleoside reverse transcriptase inhibitor
  34. GC15090 Maraviroc

    马拉维若,UK-427857; Selzentry; Celsentri

    马拉韦罗作为第一款CCR5拮抗剂已被批准用于治疗HIV感染,对hERG离子通道的IC50>10μM。

  35. GC14289 Fasudil (HA-1077) HCl

    盐酸法舒地尔; HA-1077 Hydrochloride; AT-877 Hydrochloride

    Fasudil(法舒地尔;HA-1077;AT877)是一种非特异性RhoA/ROCK抑制剂,对ROCK1的Ki为0.33μM,IC50为0.158μM,对ROCK2和PKA、PKC、PKG的IC50分别为4.58μM、12.30μM、1.650μM。
  36. GC12125 Tenofovir

    替诺福韦; GS 1278; PMPA

    An HIV and HBV antiviral
  37. GC15200 Aprepitant

    阿瑞匹坦; MK-0869; MK-869; L-754030

    An antiemetic and NK1 antagonist
  38. GC15067 Tenofovir Disoproxil Fumarate

    富马酸替诺福韦酯,Tenofovir DF; Bis(POC)-PMPA fumarate; GS 4331 fumarate

    A prodrug of the antiviral tenofovir
  39. GC17567 Doxorubicin (Adriamycin) HCl

    盐酸阿霉素; Hydroxydaunorubicin hydrochloride

    An anthracycline antitumor antibiotic

  40. GC17421 Vicriviroc maleate

    1-[(4,6-二甲基-5-嘧啶基)羰基]-4-[(3S)-4-[(1R)-2-甲氧基-1-[4-(三氟甲基)苯基]乙基]-3-甲基-1-哌嗪基]-4-甲基哌啶马来酸盐,Sch-417690; SCH-D

    A CCR5 antagonist
  41. GC14454 Tipranavir

    替拉那韦,Aptivus,Tipranavir

    A nonpeptidic HIV protease inhibitor
  42. GC15785 Saquinavir mesylate

    沙奎那韦甲磺酸盐; Ro 31-8959/003

    An HIV protease inhibitor
  43. GC15335 Saquinavir

    沙奎那韦; Ro 31-8959

    Saquinavir (Ro 31-8959) 是一种 HIV 蛋白酶抑制剂,用于抗逆转录病毒治疗。
  44. GC11059 Rilpivirine

    利匹韦林; R278474; TMC278; DB08864

    A non-nucleoside reverse transcriptase inhibitor
  45. GC14084 Nelfinavir Mesylate

    甲磺酸奈非那韦,AG 1343 Mesylate;AG1343 Mesylate;AG-1343 Mesylate,Nelfinavir

    An HIV-1 protease inhibitor
  46. GC16035 NBD-556

    N-(4-氯苯基)-N'-(2,2,6,6-四甲基哌啶-4-基)草酰胺,NBD 556;NBD556

    A small molecule CD4 mimetic
  47. GC16589 Limonin

    柠檬苦素; Limonoic acid 3,19

    柠檬苦素是一种天然的四环三萜类化合物,广泛存在于桉树、黄柏和黄连中。
  48. GC16596 Lersivirine

    3-氰基-5-[[3,5-二乙基-1-(2-羟基乙基)-1H-吡唑-4-基]氧基]苯腈,UK-453061;UK453061;UK 453061

    An NNRTI
  49. GC12998 HIV-1 integrase inhibitor

    4-[3-(叠氮基甲基)苯基]-2-羟基-4-氧代-2-丁烯酸

    HIV-1整合酶抑制剂可用于抗HIV。
  50. GC12555 GS-9620

    维沙莫德; GS-9620

    A TLR7 agonist
  51. GC11300 Fosamprenavir Calcium Salt

    福沙那伟钙,GW 433908G;Lexiva;GW433908G;GW-433908G

    A prodrug form of amprenavir

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